NO20074977L - Fuserte tiazolderivater med affinitet for histamin H3 receptoren - Google Patents
Fuserte tiazolderivater med affinitet for histamin H3 receptorenInfo
- Publication number
- NO20074977L NO20074977L NO20074977A NO20074977A NO20074977L NO 20074977 L NO20074977 L NO 20074977L NO 20074977 A NO20074977 A NO 20074977A NO 20074977 A NO20074977 A NO 20074977A NO 20074977 L NO20074977 L NO 20074977L
- Authority
- NO
- Norway
- Prior art keywords
- histamine
- affinity
- receptor
- thiazole derivatives
- fused thiazole
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Rheumatology (AREA)
- Child & Adolescent Psychology (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Obesity (AREA)
- Addiction (AREA)
- Hematology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Epidemiology (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Abstract
Foreliggende oppfinnelse angår nye sammensmeltede tiazolderivater som har farmakologisk aktivitet, fremgangsmåter for deres fremstilling, sammensetninger som inneholder dem og deres anvendelse ved behandling av neurologiske og psykiatriske forstyrrelser.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0505205A GB0505205D0 (en) | 2005-03-14 | 2005-03-14 | Novel compounds |
GB0525239A GB0525239D0 (en) | 2005-12-12 | 2005-12-12 | Novel compounds |
PCT/GB2006/000846 WO2006097691A1 (en) | 2005-03-14 | 2006-03-10 | Fused thiazole derivatives having affinity for the histamine h3 receptor |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20074977L true NO20074977L (no) | 2007-12-11 |
Family
ID=36283759
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20074977A NO20074977L (no) | 2005-03-14 | 2007-10-02 | Fuserte tiazolderivater med affinitet for histamin H3 receptoren |
Country Status (16)
Country | Link |
---|---|
US (1) | US20080161289A1 (no) |
EP (1) | EP1858900B1 (no) |
JP (1) | JP2008533117A (no) |
KR (1) | KR20070113225A (no) |
AT (1) | ATE420091T1 (no) |
AU (1) | AU2006224440A1 (no) |
BR (1) | BRPI0608437A2 (no) |
CA (1) | CA2601644A1 (no) |
DE (1) | DE602006004714D1 (no) |
EA (1) | EA200701984A1 (no) |
ES (1) | ES2321028T3 (no) |
IL (1) | IL185869A0 (no) |
MA (1) | MA29339B1 (no) |
MX (1) | MX2007011211A (no) |
NO (1) | NO20074977L (no) |
WO (1) | WO2006097691A1 (no) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0513886D0 (en) | 2005-07-06 | 2005-08-10 | Glaxo Group Ltd | Novel compounds |
US9108948B2 (en) | 2006-06-23 | 2015-08-18 | Abbvie Inc. | Cyclopropyl amine derivatives |
CN103382174A (zh) | 2006-06-23 | 2013-11-06 | 雅培制药有限公司 | 作为组胺h3受体调节物的环丙胺衍生物 |
EP2379565A1 (en) * | 2008-12-19 | 2011-10-26 | Schering Corporation | Piperidine and piperazine derivatives and methods of use thereof |
EP2379564A1 (en) | 2008-12-19 | 2011-10-26 | Schering Corporation | Bicyclic heterocyclic derivatives and methods of use thereof |
US9186353B2 (en) | 2009-04-27 | 2015-11-17 | Abbvie Inc. | Treatment of osteoarthritis pain |
RS54514B1 (en) * | 2010-09-02 | 2016-06-30 | Suven Life Sciences Limited | HETEROCYCLIC UNITS AS HISTAMINE H3 LEGANDS OF THE RECEPTOR |
WO2012037258A1 (en) | 2010-09-16 | 2012-03-22 | Abbott Laboratories | Processes for preparing 1,2-substituted cyclopropyl derivatives |
WO2013151982A1 (en) | 2012-04-03 | 2013-10-10 | Arena Pharmaceuticals, Inc. | Methods and compounds useful in treating pruritus, and methods for identifying such compounds |
EP2647377A1 (en) | 2012-04-06 | 2013-10-09 | Sanofi | Use of an h3 receptor antagonist for the treatment of alzheimer's disease |
EP3444239B1 (en) | 2016-04-06 | 2020-11-04 | Sumitomo Chemical Company, Limited | Heterocyclic compounds useful for controlling arthropods |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE4324580A1 (de) * | 1993-07-22 | 1995-01-26 | Thomae Gmbh Dr K | Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung |
DE4427838A1 (de) | 1994-08-05 | 1996-02-08 | Thomae Gmbh Dr K | Kondensierte Azepinderivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung |
JPH1017569A (ja) | 1996-07-05 | 1998-01-20 | Yamanouchi Pharmaceut Co Ltd | 置換チアゾール誘導体を有効成分とする医薬及び新規化合物 |
JP2002542245A (ja) | 1999-04-16 | 2002-12-10 | ノボ ノルディスク アクティーゼルスカブ | 置換イミダゾール、それらの製造および使用 |
GB0224083D0 (en) | 2002-10-16 | 2002-11-27 | Glaxo Group Ltd | Novel compounds |
US8466143B2 (en) | 2003-07-23 | 2013-06-18 | Exelixis, Inc. | Azepine derivatives as pharmaceutical agents |
-
2006
- 2006-03-10 AT AT06710058T patent/ATE420091T1/de not_active IP Right Cessation
- 2006-03-10 CA CA002601644A patent/CA2601644A1/en not_active Abandoned
- 2006-03-10 US US11/908,532 patent/US20080161289A1/en not_active Abandoned
- 2006-03-10 BR BRPI0608437-0A patent/BRPI0608437A2/pt not_active IP Right Cessation
- 2006-03-10 EA EA200701984A patent/EA200701984A1/ru unknown
- 2006-03-10 AU AU2006224440A patent/AU2006224440A1/en not_active Abandoned
- 2006-03-10 JP JP2008501397A patent/JP2008533117A/ja not_active Withdrawn
- 2006-03-10 EP EP06710058A patent/EP1858900B1/en active Active
- 2006-03-10 ES ES06710058T patent/ES2321028T3/es active Active
- 2006-03-10 KR KR1020077020994A patent/KR20070113225A/ko not_active Application Discontinuation
- 2006-03-10 MX MX2007011211A patent/MX2007011211A/es unknown
- 2006-03-10 WO PCT/GB2006/000846 patent/WO2006097691A1/en active Application Filing
- 2006-03-10 DE DE602006004714T patent/DE602006004714D1/de active Active
-
2007
- 2007-09-10 IL IL185869A patent/IL185869A0/en unknown
- 2007-09-24 MA MA30235A patent/MA29339B1/fr unknown
- 2007-10-02 NO NO20074977A patent/NO20074977L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
IL185869A0 (en) | 2008-01-06 |
AU2006224440A1 (en) | 2006-09-21 |
CA2601644A1 (en) | 2006-09-21 |
DE602006004714D1 (de) | 2009-02-26 |
WO2006097691A1 (en) | 2006-09-21 |
KR20070113225A (ko) | 2007-11-28 |
EP1858900A1 (en) | 2007-11-28 |
EA200701984A1 (ru) | 2008-02-28 |
EP1858900B1 (en) | 2009-01-07 |
BRPI0608437A2 (pt) | 2009-12-29 |
JP2008533117A (ja) | 2008-08-21 |
ATE420091T1 (de) | 2009-01-15 |
MX2007011211A (es) | 2007-10-17 |
MA29339B1 (fr) | 2008-03-03 |
US20080161289A1 (en) | 2008-07-03 |
ES2321028T3 (es) | 2009-06-01 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NO20074977L (no) | Fuserte tiazolderivater med affinitet for histamin H3 receptoren | |
ATE384050T1 (de) | Benzazepinderivate als histamin-h3-antagonisten | |
ATE467636T1 (de) | Pyrazoloä3 , 4-düazepinderivate als histamin-h3- antagonisten | |
ATE433966T1 (de) | Methylendipiperidinderivate | |
TW200621716A (en) | Novel compounds | |
CR9389A (es) | Compuestos de imidazopiridazina | |
TW200611701A (en) | Novel compounds | |
CY1112969T1 (el) | Ανταγωνιστες πιριδυλ πιπεριδινης του υποδοχεα ορεξινης | |
NZ592544A (en) | Isonicotinamide orexin receptor antagonists | |
UA96458C2 (ru) | Тиазолпиразолопиримидиновые соединения как антагонисты рецептора crf1 | |
MX2007006754A (es) | Derivados de indenilo y uso de los mismos para el tratamiento de trastornos neurologicos. | |
WO2005097778A8 (en) | Tetrahydrobenzazepines as histamine h3 receptor ligands | |
TW200514781A (en) | Novel compounds | |
SG166803A1 (en) | Novel processes for the preparation of cyclopropyl-amide derivatives | |
TW200621255A (en) | Novel compounds |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |