NO20074254L - Krystallinsk og amorf 4-cyano-N[(2R)-2-[4-(2,3-dihydro-benzo[1,4]dioksin-5-yl)-piperazin-1-yl]-propyl)-N-pyridin-2-yl-benzamid-hydroklorid - Google Patents
Krystallinsk og amorf 4-cyano-N[(2R)-2-[4-(2,3-dihydro-benzo[1,4]dioksin-5-yl)-piperazin-1-yl]-propyl)-N-pyridin-2-yl-benzamid-hydrokloridInfo
- Publication number
- NO20074254L NO20074254L NO20074254A NO20074254A NO20074254L NO 20074254 L NO20074254 L NO 20074254L NO 20074254 A NO20074254 A NO 20074254A NO 20074254 A NO20074254 A NO 20074254A NO 20074254 L NO20074254 L NO 20074254L
- Authority
- NO
- Norway
- Prior art keywords
- dioxin
- piperazin
- benzo
- dihydro
- cyano
- Prior art date
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/06—Antimigraine agents
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A61P25/00—Drugs for disorders of the nervous system
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/22—Anxiolytics
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A61P25/00—Drugs for disorders of the nervous system
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
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- A61P25/36—Opioid-abuse
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- A61P5/00—Drugs for disorders of the endocrine system
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- A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Anesthesiology (AREA)
- Gynecology & Obstetrics (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
(I) Foreliggende oppfinnelse omhandler krystallinske og amorfe former av 5-HT1A reseptorantagonisten 4-cyano-N-{(2R)-2-[4-(2,3-dihydro-benzo[1,4]dioksin-5-yl)-piperazin-1-yl]-propyl}-N-pyridin-2-yl-benzamidhydroklorid, så vel som sammensetninger derav og fremgangsmåter for anvendelse av disse. ?? ?? ?? ?? 38
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US65757505P | 2005-03-01 | 2005-03-01 | |
PCT/US2006/006802 WO2006093853A1 (en) | 2005-03-01 | 2006-02-27 | Crystalline and amorphous 4-cyano-n{(2r)-2-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-n-pyridin-2-yl-benzamide hydrochloride |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20074254L true NO20074254L (no) | 2007-09-24 |
Family
ID=36659970
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20074254A NO20074254L (no) | 2005-03-01 | 2007-08-21 | Krystallinsk og amorf 4-cyano-N[(2R)-2-[4-(2,3-dihydro-benzo[1,4]dioksin-5-yl)-piperazin-1-yl]-propyl)-N-pyridin-2-yl-benzamid-hydroklorid |
Country Status (19)
Country | Link |
---|---|
US (2) | US20070027162A1 (no) |
EP (1) | EP1853593A1 (no) |
JP (1) | JP2008531694A (no) |
KR (1) | KR20070112797A (no) |
CN (1) | CN101137648A (no) |
AR (1) | AR053152A1 (no) |
AU (1) | AU2006218845A1 (no) |
BR (1) | BRPI0609370A2 (no) |
CA (1) | CA2599588A1 (no) |
CR (1) | CR9319A (no) |
GT (1) | GT200600098A (no) |
IL (1) | IL185267A0 (no) |
MX (1) | MX2007010524A (no) |
NI (1) | NI200700217A (no) |
NO (1) | NO20074254L (no) |
PE (1) | PE20061344A1 (no) |
RU (1) | RU2007131044A (no) |
TW (1) | TW200700413A (no) |
WO (1) | WO2006093853A1 (no) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20070334A1 (es) * | 2005-09-09 | 2007-05-08 | Wyeth Corp | Composiciones y formas de dosificacion farmaceuticas que comprende lecozotan |
Family Cites Families (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL101722A (en) * | 1991-05-02 | 1996-05-14 | Wyeth John & Brother Ltd | History of piperazine, their preparation and pharmaceutical preparations containing them |
GB9125900D0 (en) * | 1991-12-05 | 1992-02-05 | Wyeth John & Brother Ltd | Piperazine derivatives |
CA2134038C (en) * | 1994-06-16 | 1997-06-03 | David Taiwai Wong | Potentiation of drug response |
EP0714663A3 (en) * | 1994-11-28 | 1997-01-15 | Lilly Co Eli | Potentiation of drug responses by serotonin 1A receptor antagonists |
US5568992A (en) * | 1995-05-19 | 1996-10-29 | Caterpillar Paving Products Inc. | Screed control system for an asphalt paver and method of use |
US5756532A (en) * | 1995-11-06 | 1998-05-26 | American Home Products Corporation | Aminomethyl-2 3 8 9-tetrahydro-7H-1 4-dioxino 2 3-E!-indol-8-ones and derivatives |
US5776969A (en) * | 1997-02-27 | 1998-07-07 | Eli Lilly And Company | Treatment of sleep disorders |
US6287839B1 (en) * | 1997-11-19 | 2001-09-11 | Genencor International, Inc. | Cellulase producing actinomycetes, cellulase produced therefrom and method of producing same |
US6127062A (en) * | 1998-03-24 | 2000-10-03 | Duracell Inc | End cap seal assembly for an electrochemical cell |
EP1112270B1 (en) * | 1998-09-10 | 2007-03-21 | F. Hoffmann-La Roche Ag | Dihydrobenzodioxine carboxamide and ketone derivatives as 5-ht4 receptor antagonists |
IT1318394B1 (it) * | 2000-03-17 | 2003-08-25 | Enichem Spa | Processo per la preparazione di 1-esene. |
US6469007B2 (en) * | 2000-11-28 | 2002-10-22 | Wyeth | Serotonergic agents |
AU2003220122A1 (en) * | 2002-03-12 | 2003-09-29 | Wyeth | Preparation of n1-(2'-pyridyl)-1,2-propanediamine sulfamic acid and its use in the synthesis of biologically active piperazines |
US7091349B2 (en) * | 2002-03-12 | 2006-08-15 | Wyeth | Process for synthesizing N-aryl piperazines with chiral N′-1-[benzoyl(2-pyridyl)amino]-2-propane substitution |
WO2003078417A1 (en) * | 2002-03-12 | 2003-09-25 | Wyeth, A Corporation Of The State Of Delaware | Process for synthesizing chiral n-aryl piperazines |
US20050215561A1 (en) * | 2004-03-19 | 2005-09-29 | Krishnendu Ghosh | Pharmaceutical dosage forms and compositions |
PA8626301A1 (es) * | 2004-03-19 | 2006-12-07 | Wyeth Wyeth | Proceso para preparar derivados de n-aril-piperazina |
TWI257220B (en) * | 2005-03-25 | 2006-06-21 | Ind Tech Res Inst | Cross-layer rate adaptation mechanism for WLAN |
-
2006
- 2006-02-27 CN CNA2006800068775A patent/CN101137648A/zh active Pending
- 2006-02-27 KR KR1020077021157A patent/KR20070112797A/ko not_active Application Discontinuation
- 2006-02-27 CA CA002599588A patent/CA2599588A1/en not_active Abandoned
- 2006-02-27 TW TW095106572A patent/TW200700413A/zh unknown
- 2006-02-27 AU AU2006218845A patent/AU2006218845A1/en not_active Abandoned
- 2006-02-27 JP JP2007558092A patent/JP2008531694A/ja not_active Withdrawn
- 2006-02-27 EP EP06736178A patent/EP1853593A1/en not_active Withdrawn
- 2006-02-27 WO PCT/US2006/006802 patent/WO2006093853A1/en active Application Filing
- 2006-02-27 US US11/364,902 patent/US20070027162A1/en not_active Abandoned
- 2006-02-27 BR BRPI0609370-1A patent/BRPI0609370A2/pt not_active Application Discontinuation
- 2006-02-27 MX MX2007010524A patent/MX2007010524A/es unknown
- 2006-02-27 RU RU2007131044/04A patent/RU2007131044A/ru not_active Application Discontinuation
- 2006-03-01 GT GT200600098A patent/GT200600098A/es unknown
- 2006-03-01 PE PE2006000236A patent/PE20061344A1/es not_active Application Discontinuation
- 2006-03-01 AR ARP060100776A patent/AR053152A1/es not_active Application Discontinuation
-
2007
- 2007-08-14 IL IL185267A patent/IL185267A0/en unknown
- 2007-08-16 CR CR9319A patent/CR9319A/es not_active Application Discontinuation
- 2007-08-21 NO NO20074254A patent/NO20074254L/no not_active Application Discontinuation
- 2007-08-21 NI NI200700217A patent/NI200700217A/es unknown
-
2009
- 2009-02-03 US US12/365,156 patent/US20090192311A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
TW200700413A (en) | 2007-01-01 |
US20070027162A1 (en) | 2007-02-01 |
BRPI0609370A2 (pt) | 2010-03-30 |
CR9319A (es) | 2008-01-21 |
MX2007010524A (es) | 2008-01-16 |
RU2007131044A (ru) | 2009-04-10 |
CN101137648A (zh) | 2008-03-05 |
IL185267A0 (en) | 2008-02-09 |
GT200600098A (es) | 2006-11-09 |
EP1853593A1 (en) | 2007-11-14 |
AR053152A1 (es) | 2007-04-25 |
AU2006218845A1 (en) | 2006-09-08 |
JP2008531694A (ja) | 2008-08-14 |
WO2006093853A1 (en) | 2006-09-08 |
PE20061344A1 (es) | 2007-01-03 |
US20090192311A1 (en) | 2009-07-30 |
NI200700217A (es) | 2008-07-24 |
KR20070112797A (ko) | 2007-11-27 |
CA2599588A1 (en) | 2006-09-08 |
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NO20074254L (no) | Krystallinsk og amorf 4-cyano-N[(2R)-2-[4-(2,3-dihydro-benzo[1,4]dioksin-5-yl)-piperazin-1-yl]-propyl)-N-pyridin-2-yl-benzamid-hydroklorid | |
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