NO20070157L - Substituerte diketopiperaziner som oksytocinantagonister - Google Patents
Substituerte diketopiperaziner som oksytocinantagonisterInfo
- Publication number
- NO20070157L NO20070157L NO20070157A NO20070157A NO20070157L NO 20070157 L NO20070157 L NO 20070157L NO 20070157 A NO20070157 A NO 20070157A NO 20070157 A NO20070157 A NO 20070157A NO 20070157 L NO20070157 L NO 20070157L
- Authority
- NO
- Norway
- Prior art keywords
- oxytocin antagonists
- methyl
- substituted diketopiperazines
- diketopiperazines
- substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/06—Antiabortive agents; Labour repressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Det er beskrevet forbindelser av formel (IA) hvor R1 er 2-indanyl, R2 er 1-metylpropyl, R3 er 1-metyl indazol-5-yl, R4 betyr metyl og R5 betyr hydrogen eller metyl, og farmasøytisk akseptable derivater derav, så vel som fremgangsmåter for deres fremstilling, farmasøytiske preparater inneholdende disse og anvendelse av disse innenfor medisin, spesielt anvendelse som oksytocinantagonister.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0414092.7A GB0414092D0 (en) | 2004-06-23 | 2004-06-23 | Novel compounds |
PCT/EP2005/006761 WO2006000400A1 (en) | 2004-06-23 | 2005-06-21 | Substituted diketopiperazines as oxytocin antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20070157L true NO20070157L (no) | 2007-01-23 |
Family
ID=32800052
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20070157A NO20070157L (no) | 2004-06-23 | 2007-01-09 | Substituerte diketopiperaziner som oksytocinantagonister |
Country Status (18)
Country | Link |
---|---|
US (1) | US20070208031A1 (no) |
EP (1) | EP1758893A1 (no) |
JP (1) | JP2008503535A (no) |
CN (1) | CN1989130A (no) |
AR (1) | AR049651A1 (no) |
AU (1) | AU2005256471A1 (no) |
BR (1) | BRPI0512359A (no) |
CA (1) | CA2571529A1 (no) |
GB (1) | GB0414092D0 (no) |
IL (1) | IL179912A0 (no) |
MA (1) | MA28698B1 (no) |
MX (1) | MXPA06014544A (no) |
NO (1) | NO20070157L (no) |
PE (1) | PE20060533A1 (no) |
RU (1) | RU2007102272A (no) |
TW (1) | TW200616635A (no) |
WO (1) | WO2006000400A1 (no) |
ZA (1) | ZA200610121B (no) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2641806B1 (fr) * | 1989-01-16 | 1992-05-07 | Diffusion Rech Tech Financ | Procede de stabilisation d'une aire de terrain meuble |
GB0130677D0 (en) * | 2001-12-21 | 2002-02-06 | Glaxo Group Ltd | Medicaments and novel compounds |
GB0314738D0 (en) * | 2003-06-24 | 2003-07-30 | Glaxo Group Ltd | Novel compounds |
GB0414093D0 (en) | 2004-06-23 | 2004-07-28 | Glaxo Group Ltd | Novel compounds |
GB0414100D0 (en) * | 2004-06-23 | 2004-07-28 | Glaxo Group Ltd | Novel compounds |
CA2695384A1 (en) | 2007-07-31 | 2009-02-05 | Burnham Institute For Medical Research | Bi-dentate compounds as kinase inhibitors |
US20100038143A1 (en) * | 2008-08-14 | 2010-02-18 | George Alexander Burnett | Drill cuttings treatment systems |
US8716286B2 (en) | 2009-10-30 | 2014-05-06 | Glaxo Group Limited | Crystalline forms of (3R, 6R)-3-(2,3-dihydro-1H-inden-2-yl)-1-[(1R)-1-(2,6-dimethyl-3-pyridinyl)-2-(4-morpholinyl)-2-oxoethyl]-6-[(1S)-1-methylpropyl]-2,5-piperazinedione |
CN109305969B (zh) * | 2017-07-27 | 2023-03-10 | 江苏恒瑞医药股份有限公司 | 哌嗪-2,5-二酮类衍生物、其制备方法及其在医药上的应用 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0130677D0 (en) * | 2001-12-21 | 2002-02-06 | Glaxo Group Ltd | Medicaments and novel compounds |
GB0414100D0 (en) * | 2004-06-23 | 2004-07-28 | Glaxo Group Ltd | Novel compounds |
-
2004
- 2004-06-23 GB GBGB0414092.7A patent/GB0414092D0/en not_active Ceased
-
2005
- 2005-06-21 JP JP2007517198A patent/JP2008503535A/ja active Pending
- 2005-06-21 AU AU2005256471A patent/AU2005256471A1/en not_active Abandoned
- 2005-06-21 CA CA002571529A patent/CA2571529A1/en not_active Abandoned
- 2005-06-21 TW TW094120516A patent/TW200616635A/zh unknown
- 2005-06-21 CN CNA200580024634XA patent/CN1989130A/zh active Pending
- 2005-06-21 EP EP05755377A patent/EP1758893A1/en not_active Withdrawn
- 2005-06-21 MX MXPA06014544A patent/MXPA06014544A/es not_active Application Discontinuation
- 2005-06-21 AR ARP050102538A patent/AR049651A1/es unknown
- 2005-06-21 WO PCT/EP2005/006761 patent/WO2006000400A1/en active Application Filing
- 2005-06-21 BR BRPI0512359-3A patent/BRPI0512359A/pt not_active IP Right Cessation
- 2005-06-21 RU RU2007102272/04A patent/RU2007102272A/ru not_active Application Discontinuation
- 2005-06-21 US US11/630,097 patent/US20070208031A1/en not_active Abandoned
- 2005-06-22 PE PE2005000713A patent/PE20060533A1/es not_active Application Discontinuation
-
2006
- 2006-12-04 ZA ZA200610121A patent/ZA200610121B/xx unknown
- 2006-12-07 IL IL179912A patent/IL179912A0/en unknown
- 2006-12-29 MA MA29584A patent/MA28698B1/fr unknown
-
2007
- 2007-01-09 NO NO20070157A patent/NO20070157L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AR049651A1 (es) | 2006-08-23 |
JP2008503535A (ja) | 2008-02-07 |
BRPI0512359A (pt) | 2008-03-04 |
US20070208031A1 (en) | 2007-09-06 |
GB0414092D0 (en) | 2004-07-28 |
CN1989130A (zh) | 2007-06-27 |
CA2571529A1 (en) | 2006-01-05 |
AU2005256471A1 (en) | 2006-01-05 |
RU2007102272A (ru) | 2008-07-27 |
MA28698B1 (fr) | 2007-06-01 |
WO2006000400A1 (en) | 2006-01-05 |
IL179912A0 (en) | 2007-05-15 |
ZA200610121B (en) | 2008-08-27 |
EP1758893A1 (en) | 2007-03-07 |
PE20060533A1 (es) | 2006-09-03 |
MXPA06014544A (es) | 2007-03-12 |
TW200616635A (en) | 2006-06-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |