NO20065179L - Polysykliske pyridiner som kalsium-kanalmodulatorer - Google Patents
Polysykliske pyridiner som kalsium-kanalmodulatorerInfo
- Publication number
- NO20065179L NO20065179L NO20065179A NO20065179A NO20065179L NO 20065179 L NO20065179 L NO 20065179L NO 20065179 A NO20065179 A NO 20065179A NO 20065179 A NO20065179 A NO 20065179A NO 20065179 L NO20065179 L NO 20065179L
- Authority
- NO
- Norway
- Prior art keywords
- calcium channel
- channel modulators
- pyridines
- polycyclic
- polycyclic pyridines
- Prior art date
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- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Abstract
Foreliggende oppfinnelse tilveie-bringer en familie av polysykliske pyridiner som er anvendbare som modu-latorer av kaliumionekanaler. Modu-latorene ifølge oppfinnelsen kan anvendes i både terapeutiske og diagnostiske fremgangsmåter.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US56203504P | 2004-04-13 | 2004-04-13 | |
PCT/US2005/012837 WO2005100349A2 (en) | 2004-04-13 | 2005-04-13 | Polycyclic pyridines as potassium ion channel modulators |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20065179L true NO20065179L (no) | 2007-01-15 |
Family
ID=35149256
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20065179A NO20065179L (no) | 2004-04-13 | 2006-11-10 | Polysykliske pyridiner som kalsium-kanalmodulatorer |
Country Status (12)
Country | Link |
---|---|
US (1) | US20080108600A1 (no) |
EP (1) | EP1737852A2 (no) |
JP (1) | JP2007532676A (no) |
KR (1) | KR20070030196A (no) |
CN (1) | CN1980923A (no) |
AU (1) | AU2005233642A1 (no) |
CA (1) | CA2560346A1 (no) |
IL (1) | IL178174A0 (no) |
MX (1) | MXPA06011807A (no) |
NO (1) | NO20065179L (no) |
RU (1) | RU2006139933A (no) |
WO (1) | WO2005100349A2 (no) |
Families Citing this family (32)
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GB0220581D0 (en) | 2002-09-04 | 2002-10-09 | Novartis Ag | Organic Compound |
US20050089559A1 (en) | 2003-10-23 | 2005-04-28 | Istvan Szelenyi | Combinations of potassium channel openers and sodium channel inhibitors or sodium channel-influencing active compounds for treating pains |
AR049401A1 (es) | 2004-06-18 | 2006-07-26 | Novartis Ag | Aza-biciclononanos |
GB0415746D0 (en) * | 2004-07-14 | 2004-08-18 | Novartis Ag | Organic compounds |
GB0521508D0 (en) * | 2005-10-21 | 2005-11-30 | Novartis Ag | Organic compounds |
GB0525672D0 (en) * | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
GB0525673D0 (en) * | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
US7960436B2 (en) | 2006-06-05 | 2011-06-14 | Valeant Pharmaceuticals International | Substituted arylamino-1,2,3,4-tetrahydro naphthalenes and-2,3-dihydro-1H-indenes as potassium channel modulators |
US8993593B2 (en) | 2006-08-23 | 2015-03-31 | Valeant Pharmaceuticals International | N-(4-(6-fluoro-3,4-dihydroisoquinolin-2(1H)-yl)-2,6-dimethylphenyl)-3,3-dimethylbutanamide as potassium channel modulators |
PT2061465E (pt) | 2006-08-23 | 2013-07-15 | Valeant Pharmaceuticals Int | Derivados de 4-(n-azacicloalquil)anilidas como moduladores do canal de potássio |
US8030518B2 (en) | 2006-11-28 | 2011-10-04 | Valeant Pharmaceuticals International | 1,4 diamino bicyclic retigabine analogues as potassium channel modulators |
US8367684B2 (en) | 2007-06-13 | 2013-02-05 | Valeant Pharmaceuticals International | Derivatives of 4-(N-azacycloalkyl) anilides as potassium channel modulators |
US8563566B2 (en) * | 2007-08-01 | 2013-10-22 | Valeant Pharmaceuticals International | Naphthyridine derivatives as potassium channel modulators |
US7786146B2 (en) | 2007-08-13 | 2010-08-31 | Valeant Pharmaceuticals International | Derivatives of 5-amino-4,6-disubstituted indole and 5-amino-4,6-disubstituted indoline as potassium channel modulators |
CN101868459B (zh) | 2007-09-21 | 2013-12-18 | 阿雷生物药品公司 | 用于治疗糖尿病的、作为葡糖激酶激活剂的吡啶-2-基-氨基-1,2,4-噻二唑衍生物 |
WO2009119528A1 (ja) * | 2008-03-24 | 2009-10-01 | 武田薬品工業株式会社 | 複素環化合物 |
RU2011103451A (ru) * | 2008-07-01 | 2012-08-10 | Вертекс Фармасьютикалз Инкорпорейтед (Us) | Гетероциклические производные в качестве модуляторов ионных каналов |
GB0812969D0 (en) * | 2008-07-15 | 2008-08-20 | Sentinel Oncology Ltd | Pharmaceutical compounds |
GB0821307D0 (en) * | 2008-11-21 | 2008-12-31 | Summit Corp Plc | Compounds for treatment of duchenne muscular dystrophy |
US8932842B2 (en) | 2009-02-11 | 2015-01-13 | Northwestern University | Aminopyridine dimer compounds, compositions and related methods for neuronal nitric oxide synthase inhibition |
US8278084B2 (en) | 2009-02-11 | 2012-10-02 | Northwestern University | Aminopyridine dimer compounds, compositions and related methods for neuronal nitric oxide synthase inhibition |
US8247436B2 (en) | 2010-03-19 | 2012-08-21 | Novartis Ag | Pyridine and pyrazine derivative for the treatment of CF |
GB201209587D0 (en) | 2012-05-30 | 2012-07-11 | Takeda Pharmaceutical | Therapeutic compounds |
CN103372016A (zh) * | 2013-07-04 | 2013-10-30 | 丁圣雨 | Chukrasone A在降低血糖药物中的应用 |
CN103372000B (zh) * | 2013-07-04 | 2015-09-16 | 丁圣雨 | Chukrasone B在制备治疗或预防慢性心衰的药物中的应用 |
GB201320905D0 (en) * | 2013-11-27 | 2014-01-08 | Takeda Pharmaceutical | Therapeutic compounds |
EP3189038B1 (en) * | 2014-09-05 | 2022-11-23 | Celgene Quanticel Research, Inc. | Inhibitors of lysine specific demethylase-1 |
US10913734B2 (en) * | 2016-07-11 | 2021-02-09 | Baruch S. Blumberg Institute | Substituted aminothiazoles |
EP3846793B1 (en) | 2018-09-07 | 2024-01-24 | PIC Therapeutics, Inc. | Eif4e inhibitors and uses thereof |
SI3921030T1 (sl) | 2019-02-06 | 2024-03-29 | Eli Lilly And Company | Derivati 1-((2-(2,2,2-trifluoroetoksi)piridin-4-il)metil)sečnine kot ojačevalci kcnq |
TW202317106A (zh) | 2021-08-27 | 2023-05-01 | 南韓商柳韓洋行 | 作為egfr抑制劑之取代胺基吡啶化合物 |
TW202317105A (zh) | 2021-08-27 | 2023-05-01 | 南韓商柳韓洋行 | 作為egfr抑制劑之含六員雜芳基之胺基吡啶化合物 |
Family Cites Families (14)
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BE559196A (no) * | 1956-07-13 | |||
JPS5335579B2 (no) * | 1973-04-11 | 1978-09-28 | ||
US3923773A (en) * | 1973-04-25 | 1975-12-02 | Dainippon Ink & Chemicals | Method for preparing isoindolenone pigments |
JPS54119531A (en) * | 1978-03-10 | 1979-09-17 | Nippon Soda Co Ltd | Bispyrrolopyrazine compound, its preparation, and method of using it as pigment |
JPS5650965A (en) * | 1979-10-03 | 1981-05-08 | Dainippon Ink & Chem Inc | Preparation of isoindolinone pigment |
JPS57155242A (en) * | 1981-03-20 | 1982-09-25 | Dainippon Ink & Chem Inc | Colorant for polyolefin resin |
DE68926082T2 (de) * | 1988-09-07 | 1996-11-28 | Minnesota Mining & Mfg | Photoinitiator enthaltende Halogenmethyl-1,3,5-Triazine |
EP0596126A4 (en) * | 1991-12-27 | 1994-06-08 | Wakunaga Seiyaku Kk | Novel quinolone derivative or salt thereof and antibacterial containing the same. |
TW327171B (en) * | 1994-02-18 | 1998-02-21 | Boehringer Ingelheim Pharma | 2-heteroaryl-5 for prevention or treatment of HIV infection |
US5705499A (en) * | 1995-10-06 | 1998-01-06 | Boehringer Ingelheim Pharmaceuticals, Inc. | 8-arylalkyl- and 8-arylheteroalkyl-5,11-dihydro-6H-dipyrido 3,2-B:2',3'-e! 1!diazepines and their use in the treatment of HIV-1 infection |
JP3991376B2 (ja) * | 1996-02-22 | 2007-10-17 | 三菱化学株式会社 | カラー画像の形成方法 |
PL359416A1 (en) * | 2000-07-18 | 2004-08-23 | Yamanouchi Pharmaceutical Co, Ltd. | Medicine comprising dicyanopyridine derivative |
JP4177561B2 (ja) * | 2001-03-30 | 2008-11-05 | 富士フイルム株式会社 | ビストリアジン誘導体を含有する写真処理組成物及び画像形成方法 |
JP2003050447A (ja) * | 2001-08-06 | 2003-02-21 | Fuji Photo Film Co Ltd | ハロゲン化銀写真感光材料用固体処理剤及びその製造方法 |
-
2005
- 2005-04-13 EP EP05734869A patent/EP1737852A2/en not_active Withdrawn
- 2005-04-13 AU AU2005233642A patent/AU2005233642A1/en not_active Abandoned
- 2005-04-13 US US10/592,985 patent/US20080108600A1/en not_active Abandoned
- 2005-04-13 CA CA002560346A patent/CA2560346A1/en not_active Abandoned
- 2005-04-13 KR KR1020067023733A patent/KR20070030196A/ko not_active Application Discontinuation
- 2005-04-13 RU RU2006139933/04A patent/RU2006139933A/ru not_active Application Discontinuation
- 2005-04-13 CN CNA2005800111395A patent/CN1980923A/zh active Pending
- 2005-04-13 WO PCT/US2005/012837 patent/WO2005100349A2/en active Application Filing
- 2005-04-13 MX MXPA06011807A patent/MXPA06011807A/es not_active Application Discontinuation
- 2005-04-13 JP JP2007508563A patent/JP2007532676A/ja not_active Withdrawn
-
2006
- 2006-09-19 IL IL178174A patent/IL178174A0/en unknown
- 2006-11-10 NO NO20065179A patent/NO20065179L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
CA2560346A1 (en) | 2005-10-27 |
KR20070030196A (ko) | 2007-03-15 |
CN1980923A (zh) | 2007-06-13 |
WO2005100349A2 (en) | 2005-10-27 |
EP1737852A2 (en) | 2007-01-03 |
IL178174A0 (en) | 2006-12-31 |
RU2006139933A (ru) | 2008-05-20 |
MXPA06011807A (es) | 2007-02-21 |
AU2005233642A1 (en) | 2005-10-27 |
WO2005100349A3 (en) | 2006-03-16 |
US20080108600A1 (en) | 2008-05-08 |
JP2007532676A (ja) | 2007-11-15 |
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