NO20052150L - Insekticid og anthelmintisk forbindelse samt fremstilling derav. - Google Patents

Insekticid og anthelmintisk forbindelse samt fremstilling derav.

Info

Publication number
NO20052150L
NO20052150L NO20052150A NO20052150A NO20052150L NO 20052150 L NO20052150 L NO 20052150L NO 20052150 A NO20052150 A NO 20052150A NO 20052150 A NO20052150 A NO 20052150A NO 20052150 L NO20052150 L NO 20052150L
Authority
NO
Norway
Prior art keywords
fki
substance
insecticide
preparation
activity
Prior art date
Application number
NO20052150A
Other languages
English (en)
Inventor
Satoshi Omura
Rokuro Masuma
Kazuro Shiomi
Original Assignee
Kitasato Inst
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kitasato Inst filed Critical Kitasato Inst
Publication of NO20052150L publication Critical patent/NO20052150L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K11/00Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12NMICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N1/00Microorganisms, e.g. protozoa; Compositions thereof; Processes of propagating, maintaining or preserving microorganisms or compositions thereof; Processes of preparing or isolating a composition containing a microorganism; Culture media therefor
    • C12N1/14Fungi; Culture media therefor
    • C12N1/145Fungal isolates
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P17/00Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
    • C12P17/14Nitrogen or oxygen as hetero atom and at least one other diverse hetero ring atom in the same ring
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12RINDEXING SCHEME ASSOCIATED WITH SUBCLASSES C12C - C12Q, RELATING TO MICROORGANISMS
    • C12R2001/00Microorganisms ; Processes using microorganisms
    • C12R2001/645Fungi ; Processes using fungi

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Genetics & Genomics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Engineering & Computer Science (AREA)
  • Microbiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Mycology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Botany (AREA)
  • Dentistry (AREA)
  • Virology (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

Det er beskrevet å dyrke en mikroorganisme som har egenskapen å danne FKI-1033-substans representert av formelen: i et medium, akkumulere FKI-1033-substans i dyrkningsmediet og isolere FKI-1033-substans fra den dyrkede masse. Den således fremstilte FKI-1033-substans har ryanodinebinding inhiberingsaktivitet, insekticid aktivitet og anthelmintisk aktivitet, og er ventet å være et anvendelig medikament som agrokjemikalium, veterinærmedisin og som medikamenter i effektivitet og toksisitet.
NO20052150A 2002-11-12 2005-05-02 Insekticid og anthelmintisk forbindelse samt fremstilling derav. NO20052150L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/JP2002/011777 WO2004044214A1 (ja) 2002-11-12 2002-11-12 新規fki−1033物質およびその製造法

Publications (1)

Publication Number Publication Date
NO20052150L true NO20052150L (no) 2005-06-10

Family

ID=32310251

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20052150A NO20052150L (no) 2002-11-12 2005-05-02 Insekticid og anthelmintisk forbindelse samt fremstilling derav.

Country Status (12)

Country Link
US (1) US7541336B2 (no)
EP (1) EP1561820B1 (no)
JP (1) JP4176077B2 (no)
AT (1) ATE419373T1 (no)
BR (1) BR0215937A (no)
CA (1) CA2504309A1 (no)
DE (1) DE60230686D1 (no)
ES (1) ES2318053T3 (no)
MX (1) MXPA05005032A (no)
NO (1) NO20052150L (no)
NZ (1) NZ539986A (no)
WO (1) WO2004044214A1 (no)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE602005014124D1 (de) * 2004-09-07 2009-06-04 Banyu Pharma Co Ltd Carbamoylsubstituiertes spiro-derivat
JP2014037351A (ja) * 2010-12-10 2014-02-27 Meiji Seikaファルマ株式会社 新規デプシペプチドpf1442物質およびその製造法
HUE042661T2 (hu) * 2012-06-13 2019-07-29 Meiji Seika Pharma Co Ltd Új ciklusos depszipeptid származék és ezt tartalmazó kártevõirtó szer
WO2015093558A1 (ja) * 2013-12-18 2015-06-25 Meiji Seikaファルマ株式会社 環状デプシペプチド誘導体およびそれを含んでなる有害生物防除剤
WO2018237394A1 (en) * 2017-06-23 2018-12-27 Vanderbilt University VERTICILIDE ENANTIOMER AND METHODS OF INHIBITING INTRACELLULAR CALCIUM RELEASE WITH RYANODINE RECEPTOR MEDIATION

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO176766C (no) * 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
DE4317432A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE10008128A1 (de) * 2000-02-22 2001-08-23 Bayer Ag Endoparasitizide Mittel
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere

Also Published As

Publication number Publication date
ATE419373T1 (de) 2009-01-15
EP1561820A1 (en) 2005-08-10
MXPA05005032A (es) 2008-02-05
NZ539986A (en) 2007-03-30
JP4176077B2 (ja) 2008-11-05
ES2318053T3 (es) 2009-05-01
JPWO2004044214A1 (ja) 2006-03-09
EP1561820B1 (en) 2008-12-31
EP1561820A4 (en) 2007-08-22
BR0215937A (pt) 2005-09-06
DE60230686D1 (de) 2009-02-12
CA2504309A1 (en) 2004-05-27
AU2002344494A1 (en) 2004-06-03
US20060111280A1 (en) 2006-05-25
US7541336B2 (en) 2009-06-02
WO2004044214A1 (ja) 2004-05-27

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