NO20035313D0 - Fremgangsmåte for fremstilling av tialzol PPAR-ligand og polymorfer derav - Google Patents

Fremgangsmåte for fremstilling av tialzol PPAR-ligand og polymorfer derav

Info

Publication number
NO20035313D0
NO20035313D0 NO20035313A NO20035313A NO20035313D0 NO 20035313 D0 NO20035313 D0 NO 20035313D0 NO 20035313 A NO20035313 A NO 20035313A NO 20035313 A NO20035313 A NO 20035313A NO 20035313 D0 NO20035313 D0 NO 20035313D0
Authority
NO
Norway
Prior art keywords
polymorphs
tialzole
preparation
ppar ligand
compound
Prior art date
Application number
NO20035313A
Other languages
English (en)
Other versions
NO20035313L (no
Inventor
Thierry Boyer
Caroline Jane Day
Andrew Jonathan Whitehead
Richard Anthony Henson
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NO20035313D0 publication Critical patent/NO20035313D0/no
Publication of NO20035313L publication Critical patent/NO20035313L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Nutrition Science (AREA)
  • Child & Adolescent Psychology (AREA)
  • Vascular Medicine (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Physical Or Chemical Processes And Apparatus (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
NO20035313A 2001-05-31 2003-11-28 Fremgangsmåte for fremstilling av tialzol PPAR-ligand og polymorfer derav NO20035313L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0113232.3A GB0113232D0 (en) 2001-05-31 2001-05-31 Chemical process
PCT/EP2002/005884 WO2002096893A1 (en) 2001-05-31 2002-05-29 Process for preparing a thialzole ppar-ligand and polymorphs thereof

Publications (2)

Publication Number Publication Date
NO20035313D0 true NO20035313D0 (no) 2003-11-28
NO20035313L NO20035313L (no) 2003-12-09

Family

ID=9915637

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20035313A NO20035313L (no) 2001-05-31 2003-11-28 Fremgangsmåte for fremstilling av tialzol PPAR-ligand og polymorfer derav

Country Status (22)

Country Link
US (1) US7244849B2 (no)
EP (1) EP1395572B1 (no)
JP (1) JP2004532265A (no)
KR (1) KR20040007631A (no)
CN (1) CN1551871A (no)
AT (1) ATE315556T1 (no)
AU (1) AU2002317764B2 (no)
BR (1) BR0209892A (no)
CA (1) CA2448101A1 (no)
CO (1) CO5540298A2 (no)
CZ (1) CZ20033256A3 (no)
DE (1) DE60208682T2 (no)
ES (1) ES2256493T3 (no)
GB (1) GB0113232D0 (no)
HU (1) HUP0400117A3 (no)
IL (1) IL158641A0 (no)
MX (1) MXPA03010943A (no)
NO (1) NO20035313L (no)
NZ (1) NZ529486A (no)
PL (1) PL367114A1 (no)
WO (1) WO2002096893A1 (no)
ZA (1) ZA200308570B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7105551B2 (en) * 2000-12-20 2006-09-12 Smithkline Beecham Corporation Thiazole derivatives for treating PPAR related disorders
CN1662487A (zh) 2002-06-19 2005-08-31 伊莱利利公司 酰胺连接基过氧化物酶体增殖物激活受体调节剂
TW200400816A (en) 2002-06-26 2004-01-16 Lilly Co Eli Tricyclic steroid hormone nuclear receptor modulators
US7553867B2 (en) 2002-09-06 2009-06-30 Takeda Pharmaceutical Company Limited Furan or thiophene derivative and medicinal use thereof
EA010422B1 (ru) 2003-08-01 2008-08-29 Янссен Фармацевтика Н.В. Замещённые индол-о-глюкозиды
WO2005097076A2 (en) * 2004-04-09 2005-10-20 Smithkline Beecham Corporation Low dose pharmaceutical products
CN101400663A (zh) * 2006-01-10 2009-04-01 史密丝克莱恩比彻姆公司 {2-甲基-4-[4-甲基-2-(4-三氟甲基苯基)噻唑-5-基甲硫基]苯氧基}-乙酸的多晶型
WO2012168948A2 (en) * 2011-06-06 2012-12-13 Hetero Research Foundation Process for febuxostat

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1067109B1 (en) 1998-03-10 2009-12-09 Ono Pharmaceutical Co., Ltd. Carboxylic acid derivatives and drugs containing the same as the active ingredient
PE20011010A1 (es) 1999-12-02 2001-10-18 Glaxo Group Ltd Oxazoles y tiazoles sustituidos como agonista del receptor activado por el proliferador de peroxisomas humano
JP2004517100A (ja) * 2000-12-20 2004-06-10 グラクソ グループ リミテッド hPPARアルファアゴニストとしての置換オキサゾールおよびチアゾール
GB0111523D0 (en) * 2001-05-11 2001-07-04 Glaxo Group Ltd Chemical compounds
GB0113233D0 (en) * 2001-05-31 2001-07-25 Glaxo Group Ltd Chemical compounds

Also Published As

Publication number Publication date
EP1395572B1 (en) 2006-01-11
CA2448101A1 (en) 2002-12-05
JP2004532265A (ja) 2004-10-21
PL367114A1 (en) 2005-02-21
WO2002096893A1 (en) 2002-12-05
US20040242657A1 (en) 2004-12-02
CO5540298A2 (es) 2005-07-29
US7244849B2 (en) 2007-07-17
AU2002317764B2 (en) 2005-01-06
ATE315556T1 (de) 2006-02-15
ES2256493T3 (es) 2006-07-16
CZ20033256A3 (en) 2004-04-14
KR20040007631A (ko) 2004-01-24
BR0209892A (pt) 2004-06-08
IL158641A0 (en) 2004-05-12
GB0113232D0 (en) 2001-07-25
EP1395572A1 (en) 2004-03-10
HUP0400117A3 (en) 2005-09-28
DE60208682T2 (de) 2006-08-24
ZA200308570B (en) 2005-02-03
NO20035313L (no) 2003-12-09
NZ529486A (en) 2005-12-23
CN1551871A (zh) 2004-12-01
MXPA03010943A (es) 2004-02-27
HUP0400117A2 (hu) 2005-03-29
DE60208682D1 (de) 2006-04-06

Similar Documents

Publication Publication Date Title
MY134892A (en) Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines and their use
CY1110631T1 (el) Διαλυτοποιημενα δηλητηρια τοποϊσομερασης
YU59001A (sh) 16-halogen-epotilon-derivati, postupak za njihovo dobijanje i njihova farmaceutska primena
HK1070063A1 (en) Stable polymorph of flibanserin, technical processfor its preparation and the use thereof for prepa ring medicaments
GB9822473D0 (en) Chemical compounds
CY1106743T1 (el) Μεθοδος παρασκευης θειαμεθοξαμης
WO2005021544A3 (en) N3-substituted imidazopyridine-derivatives as c-kit inhibitors
YU61103A (sh) Postupci za produkciju supstituisanih 2-(2-piridilmetil) sulfinil-1h-benzimidazola
JO2413B1 (en) Benzoxazine derivatives and their use
PL371127A1 (en) 6-aminomorphinane derivatives, method for the production and use thereof
MXPA03004426A (es) Proceso quimico y nuevos intermediarios.
CY1107635T1 (el) Μεθοδος για την παρασκευη σιταλοπραμης
BR0209901A (pt) Processos para a sìntese de derivados de 2,3-dihidro-1,4-dioxino-[2,3-f] quinolina
MXPA05005790A (es) Aminoalcoxiindoles como ligandos del receptor 5-ht6 para el tratamiento de enfermedades del sistema nervioso central.
NO20035313D0 (no) Fremgangsmåte for fremstilling av tialzol PPAR-ligand og polymorfer derav
WO2007014839A3 (en) Cathepsin k inhibitors
NO20032401D0 (no) Fremgangsmåte ved fremstilling av taksanderivater
FI952420A (fi) Glukopyranosidibentsotiofeenit
WO2002072567A3 (en) Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them
WO2004039776A3 (en) A process for the preparation of benzyl 2-oxo-4- (heteroaryl) dithio-alpha-isoprenyl-1- azetidineazetate derivatives
SG149005A1 (en) Process for the preparation of thiazolopyrimidines
EA200100157A3 (ru) Новые производные арил- или гетероарилхинолинилфосфоновой кислоты, способ их получения и содержащие их фармацевтические композиции
MXPA04001852A (es) Uso de sistemas indan-1-ol c2-sustituidas para la produccion de medicamentos para la profilaxis o tratamiento de obesidad.
MXPA04001856A (es) Indan-1-oles c2-sustituidos y sus derivados, metodo para su produccion y su uso como medicamentos.
MXPA04001851A (es) Inda-1-onas c2-disustituidas y sus derivados, metodo para su produccion y su uso como medicamentos.

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application