NO20026194L - Selektive androgen-reseptor-modulatorer og fremgangsmåter for deres identifikasjon, utforming og anvendelse - Google Patents

Selektive androgen-reseptor-modulatorer og fremgangsmåter for deres identifikasjon, utforming og anvendelse

Info

Publication number
NO20026194L
NO20026194L NO20026194A NO20026194A NO20026194L NO 20026194 L NO20026194 L NO 20026194L NO 20026194 A NO20026194 A NO 20026194A NO 20026194 A NO20026194 A NO 20026194A NO 20026194 L NO20026194 L NO 20026194L
Authority
NO
Norway
Prior art keywords
identification
design
methods
androgen receptor
receptor modulators
Prior art date
Application number
NO20026194A
Other languages
English (en)
Norwegian (no)
Other versions
NO20026194D0 (no
Inventor
Mark Ernest Salvati
Marco M Gottardis
Jr Stanley R Krystek
Ricardo M Attar
John S Sack
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20026194D0 publication Critical patent/NO20026194D0/no
Publication of NO20026194L publication Critical patent/NO20026194L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/655—Azo (—N=N—), diazo (=N2), azoxy (>N—O—N< or N(=O)—N<), azido (—N3) or diazoamino (—N=N—N<) compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/28—Antiandrogens

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Diabetes (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Peptides Or Proteins (AREA)
NO20026194A 2000-06-28 2002-12-23 Selektive androgen-reseptor-modulatorer og fremgangsmåter for deres identifikasjon, utforming og anvendelse NO20026194L (no)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US21439200P 2000-06-28 2000-06-28
US23351900P 2000-09-19 2000-09-19
US28473001P 2001-04-18 2001-04-18
US28443801P 2001-04-18 2001-04-18
US28461701P 2001-04-18 2001-04-18
PCT/US2001/019665 WO2002000617A2 (en) 2000-06-28 2001-06-20 Selective androgen receptor modulators and methods for their identification, design and use

Publications (2)

Publication Number Publication Date
NO20026194D0 NO20026194D0 (no) 2002-12-23
NO20026194L true NO20026194L (no) 2003-02-26

Family

ID=27539683

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20026194A NO20026194L (no) 2000-06-28 2002-12-23 Selektive androgen-reseptor-modulatorer og fremgangsmåter for deres identifikasjon, utforming og anvendelse

Country Status (14)

Country Link
US (2) US6960474B2 (de)
EP (1) EP1299094A2 (de)
JP (1) JP2004509072A (de)
KR (1) KR20030016310A (de)
CN (1) CN1454083A (de)
AU (2) AU2001288213B2 (de)
BR (1) BR0111298A (de)
CA (1) CA2413417A1 (de)
CZ (1) CZ20024214A3 (de)
HU (1) HUP0303172A3 (de)
IL (1) IL152719A0 (de)
MX (1) MXPA02012605A (de)
NO (1) NO20026194L (de)
WO (1) WO2002000617A2 (de)

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JP2004509072A (ja) 2004-03-25
BR0111298A (pt) 2005-05-10
WO2002000617A3 (en) 2003-01-30
WO2002000617A2 (en) 2002-01-03
HUP0303172A3 (en) 2006-05-29
KR20030016310A (ko) 2003-02-26
US20020173445A1 (en) 2002-11-21
AU8821301A (en) 2002-01-08
CA2413417A1 (en) 2002-01-03
US6960474B2 (en) 2005-11-01
CZ20024214A3 (cs) 2003-04-16
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IL152719A0 (en) 2003-06-24
MXPA02012605A (es) 2003-05-14

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