NO20015892D0 - Inhibitorer av metallproteinaser - Google Patents
Inhibitorer av metallproteinaserInfo
- Publication number
- NO20015892D0 NO20015892D0 NO20015892A NO20015892A NO20015892D0 NO 20015892 D0 NO20015892 D0 NO 20015892D0 NO 20015892 A NO20015892 A NO 20015892A NO 20015892 A NO20015892 A NO 20015892A NO 20015892 D0 NO20015892 D0 NO 20015892D0
- Authority
- NO
- Norway
- Prior art keywords
- inhibitors
- metal proteinases
- proteinases
- metal
- arylpiperazines
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/26—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms
- C07D211/28—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms to which a second hetero atom is attached
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP99401350 | 1999-06-04 | ||
PCT/GB2000/002085 WO2000075108A1 (en) | 1999-06-04 | 2000-05-31 | Inhibitors of metalloproteinases |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20015892D0 true NO20015892D0 (no) | 2001-12-03 |
NO20015892L NO20015892L (no) | 2001-12-19 |
Family
ID=8241999
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20015892A NO20015892L (no) | 1999-06-04 | 2001-12-03 | Inhibitorer av metallproteinaser |
Country Status (17)
Country | Link |
---|---|
US (1) | US6916817B1 (no) |
EP (1) | EP1187811B1 (no) |
JP (1) | JP2003501414A (no) |
KR (1) | KR20020005769A (no) |
CN (1) | CN1159295C (no) |
AT (1) | ATE356114T1 (no) |
AU (1) | AU773967B2 (no) |
BR (1) | BR0011339A (no) |
CA (1) | CA2374460A1 (no) |
DE (1) | DE60033809T2 (no) |
ES (1) | ES2281346T3 (no) |
IL (1) | IL146543A0 (no) |
MX (1) | MXPA01012322A (no) |
NO (1) | NO20015892L (no) |
NZ (1) | NZ515829A (no) |
WO (1) | WO2000075108A1 (no) |
ZA (1) | ZA200109675B (no) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0119474D0 (en) | 2001-08-09 | 2001-10-03 | Astrazeneca Ab | Compounds |
EP1431285B1 (en) | 2001-09-07 | 2009-01-07 | Kaken Pharmaceutical Co., Ltd. | Reverse hydroxamic acid derivatives |
SE0301922D0 (sv) | 2003-06-27 | 2003-06-27 | Astrazeneca Ab | Novel compounds |
GB0427403D0 (en) * | 2004-12-15 | 2005-01-19 | Astrazeneca Ab | Novel compounds I |
KR20080064880A (ko) * | 2005-10-26 | 2008-07-09 | 라보라뚜와르 세로노 에스. 에이. | 술폰아미드 유도체 및 금속단백분해효소를 조정하기 위한그것의 용도 |
KR100673015B1 (ko) | 2005-11-14 | 2007-01-24 | 삼성전자주식회사 | 캐패시터를 갖는 반도체 소자 및 그 형성 방법 |
GB0617367D0 (en) * | 2006-09-02 | 2006-10-11 | Astrazeneca Ab | Novel process |
WO2008147763A1 (en) * | 2007-05-23 | 2008-12-04 | Array Biopharma Inc. | Mmp inhibitors and methods of use thereof |
EA201792443A1 (ru) | 2015-05-06 | 2018-10-31 | Дзе Риджентс Оф Дзе Юниверсити Оф Калифорния | МОДУЛЯТОРЫ K-Ras |
MX2019012532A (es) | 2017-04-20 | 2019-12-02 | Univ California | Moduladores de k-ras. |
WO2019204449A1 (en) * | 2018-04-18 | 2019-10-24 | Theras, Inc. | K-ras modulators with a vinyl sulfone moiety |
AU2019352741A1 (en) | 2018-10-04 | 2021-05-06 | Assistance Publique-Hôpitaux De Paris (Aphp) | EGFR inhibitors for treating keratodermas |
CN111117990B (zh) * | 2020-02-26 | 2023-03-28 | 中国医科大学 | 一种抑制mmp9活性的多肽及其应用 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5817822A (en) | 1994-06-24 | 1998-10-06 | Novartis Corporation | Certain alpha-azacycloalkyl substituted arylsulfonamido acetohydroxamic acids |
HUP0000941A3 (en) * | 1997-01-23 | 2002-06-28 | Hoffmann La Roche | Sulfamide derivatives, process for producing them, pharmaceutical compositions containing them and their use |
WO1999002510A1 (en) * | 1997-07-10 | 1999-01-21 | Pharmacia & Upjohn S.P.A. | Matrix metalloproteinase inhibitors |
ZA988967B (en) * | 1997-10-03 | 2000-04-03 | Du Pont Pharm Co | Lactam metalloprotease inhibitors. |
ATE346041T1 (de) * | 1998-01-30 | 2006-12-15 | Darwin Discovery Ltd | N-hydroxyformamid-derivate |
GB9919776D0 (en) * | 1998-08-31 | 1999-10-27 | Zeneca Ltd | Compoujnds |
-
2000
- 2000-05-31 EP EP00935363A patent/EP1187811B1/en not_active Expired - Lifetime
- 2000-05-31 ES ES00935363T patent/ES2281346T3/es not_active Expired - Lifetime
- 2000-05-31 BR BR0011339-5A patent/BR0011339A/pt not_active IP Right Cessation
- 2000-05-31 WO PCT/GB2000/002085 patent/WO2000075108A1/en active IP Right Grant
- 2000-05-31 AU AU50909/00A patent/AU773967B2/en not_active Ceased
- 2000-05-31 NZ NZ515829A patent/NZ515829A/en unknown
- 2000-05-31 IL IL14654300A patent/IL146543A0/xx unknown
- 2000-05-31 MX MXPA01012322A patent/MXPA01012322A/es unknown
- 2000-05-31 DE DE60033809T patent/DE60033809T2/de not_active Expired - Fee Related
- 2000-05-31 CA CA002374460A patent/CA2374460A1/en not_active Abandoned
- 2000-05-31 AT AT00935363T patent/ATE356114T1/de not_active IP Right Cessation
- 2000-05-31 CN CNB008112231A patent/CN1159295C/zh not_active Expired - Fee Related
- 2000-05-31 JP JP2001501589A patent/JP2003501414A/ja active Pending
- 2000-05-31 KR KR1020017015430A patent/KR20020005769A/ko not_active Application Discontinuation
- 2000-05-31 US US09/980,593 patent/US6916817B1/en not_active Expired - Fee Related
-
2001
- 2001-11-23 ZA ZA200109675A patent/ZA200109675B/en unknown
- 2001-12-03 NO NO20015892A patent/NO20015892L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
ATE356114T1 (de) | 2007-03-15 |
DE60033809T2 (de) | 2007-12-06 |
CN1390200A (zh) | 2003-01-08 |
AU773967B2 (en) | 2004-06-10 |
US6916817B1 (en) | 2005-07-12 |
NZ515829A (en) | 2003-10-31 |
JP2003501414A (ja) | 2003-01-14 |
ZA200109675B (en) | 2003-02-24 |
ES2281346T3 (es) | 2007-10-01 |
AU5090900A (en) | 2000-12-28 |
MXPA01012322A (es) | 2002-07-22 |
DE60033809D1 (de) | 2007-04-19 |
EP1187811B1 (en) | 2007-03-07 |
CA2374460A1 (en) | 2000-12-14 |
WO2000075108A1 (en) | 2000-12-14 |
NO20015892L (no) | 2001-12-19 |
KR20020005769A (ko) | 2002-01-17 |
CN1159295C (zh) | 2004-07-28 |
EP1187811A1 (en) | 2002-03-20 |
IL146543A0 (en) | 2002-07-25 |
BR0011339A (pt) | 2002-03-19 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |