NO20011654D0 - Benzamidderivater som trombininhibitorer - Google Patents
Benzamidderivater som trombininhibitorerInfo
- Publication number
- NO20011654D0 NO20011654D0 NO20011654A NO20011654A NO20011654D0 NO 20011654 D0 NO20011654 D0 NO 20011654D0 NO 20011654 A NO20011654 A NO 20011654A NO 20011654 A NO20011654 A NO 20011654A NO 20011654 D0 NO20011654 D0 NO 20011654D0
- Authority
- NO
- Norway
- Prior art keywords
- thrombin inhibitors
- benzamide derivatives
- benzamide
- derivatives
- thrombin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9821483.6A GB9821483D0 (en) | 1998-10-03 | 1998-10-03 | Chemical compounds |
| PCT/EP1999/007194 WO2000020394A1 (en) | 1998-10-03 | 1999-09-30 | Benzamide derivatives as thrombin inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20011654D0 true NO20011654D0 (no) | 2001-04-02 |
| NO20011654L NO20011654L (no) | 2001-05-30 |
Family
ID=10839873
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20011654A NO20011654L (no) | 1998-10-03 | 2001-04-02 | Benzamidderivater som trombininhibitorer |
Country Status (21)
| Country | Link |
|---|---|
| US (2) | US6441008B1 (no) |
| EP (1) | EP1117644A1 (no) |
| JP (1) | JP3457281B2 (no) |
| KR (1) | KR20010075546A (no) |
| CN (1) | CN1328548A (no) |
| AR (1) | AR023332A1 (no) |
| AU (1) | AU758007B2 (no) |
| BR (1) | BR9914267A (no) |
| CA (1) | CA2345997A1 (no) |
| CO (1) | CO5140085A1 (no) |
| CZ (1) | CZ20011216A3 (no) |
| GB (1) | GB9821483D0 (no) |
| HU (1) | HUP0103744A3 (no) |
| IL (1) | IL142301A0 (no) |
| MA (1) | MA26695A1 (no) |
| NO (1) | NO20011654L (no) |
| NZ (1) | NZ510839A (no) |
| PE (1) | PE20001059A1 (no) |
| PL (1) | PL347152A1 (no) |
| TR (1) | TR200100906T2 (no) |
| WO (1) | WO2000020394A1 (no) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0117144D0 (en) * | 2001-07-13 | 2001-09-05 | Glaxo Group Ltd | Process |
| EP1637141B1 (en) | 2004-09-21 | 2011-11-16 | Trobio AB | Stabilized protease composition comprising a serine protease, morpholino derivatives and reversible inhibitors of said serine protease |
| AU2005336535B2 (en) * | 2005-09-22 | 2012-05-24 | Trobio Ab | Stabilized protease composition |
| TWI808055B (zh) | 2016-05-11 | 2023-07-11 | 美商滬亞生物國際有限公司 | Hdac 抑制劑與 pd-1 抑制劑之組合治療 |
| TWI794171B (zh) | 2016-05-11 | 2023-03-01 | 美商滬亞生物國際有限公司 | Ｈｄａｃ抑制劑與ｐｄ-ｌ１抑制劑之組合治療 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW257757B (no) | 1993-03-03 | 1995-09-21 | Boehringer Mannheim Gmbh | |
| IL109144A (en) | 1993-03-29 | 2000-02-29 | Zeneca Ltd | Glycoprotein IIB/IIIA inhibiting 4-pyridylamino heterocyclic derivatives process for their preparation and pharmaceutical compositions containing them |
| GB9525620D0 (en) * | 1995-12-15 | 1996-02-14 | Glaxo Group Ltd | Chemical compounds |
-
1998
- 1998-10-03 GB GBGB9821483.6A patent/GB9821483D0/en not_active Ceased
-
1999
- 1999-09-29 AR ARP990104910A patent/AR023332A1/es not_active Application Discontinuation
- 1999-09-30 IL IL14230199A patent/IL142301A0/xx unknown
- 1999-09-30 CO CO99061898A patent/CO5140085A1/es unknown
- 1999-09-30 NZ NZ510839A patent/NZ510839A/en unknown
- 1999-09-30 PL PL99347152A patent/PL347152A1/xx not_active Application Discontinuation
- 1999-09-30 BR BR9914267-8A patent/BR9914267A/pt not_active IP Right Cessation
- 1999-09-30 CZ CZ20011216A patent/CZ20011216A3/cs unknown
- 1999-09-30 TR TR2001/00906T patent/TR200100906T2/xx unknown
- 1999-09-30 CA CA002345997A patent/CA2345997A1/en not_active Abandoned
- 1999-09-30 PE PE1999000995A patent/PE20001059A1/es not_active Application Discontinuation
- 1999-09-30 JP JP2000574511A patent/JP3457281B2/ja not_active Expired - Fee Related
- 1999-09-30 HU HU0103744A patent/HUP0103744A3/hu unknown
- 1999-09-30 EP EP99952472A patent/EP1117644A1/en not_active Withdrawn
- 1999-09-30 AU AU64670/99A patent/AU758007B2/en not_active Ceased
- 1999-09-30 KR KR1020017004191A patent/KR20010075546A/ko not_active Application Discontinuation
- 1999-09-30 US US09/806,407 patent/US6441008B1/en not_active Expired - Fee Related
- 1999-09-30 CN CN99813786A patent/CN1328548A/zh active Pending
- 1999-09-30 WO PCT/EP1999/007194 patent/WO2000020394A1/en not_active Application Discontinuation
- 1999-10-01 MA MA25797A patent/MA26695A1/fr unknown
-
2001
- 2001-04-02 NO NO20011654A patent/NO20011654L/no not_active Application Discontinuation
-
2002
- 2002-01-10 US US10/044,769 patent/US6670381B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP2002526531A (ja) | 2002-08-20 |
| HUP0103744A3 (en) | 2002-03-28 |
| MA26695A1 (fr) | 2004-12-20 |
| CZ20011216A3 (cs) | 2001-09-12 |
| BR9914267A (pt) | 2001-07-03 |
| AU758007B2 (en) | 2003-03-13 |
| US20020169189A1 (en) | 2002-11-14 |
| KR20010075546A (ko) | 2001-08-09 |
| IL142301A0 (en) | 2002-03-10 |
| AU6467099A (en) | 2000-04-26 |
| CA2345997A1 (en) | 2000-04-13 |
| JP3457281B2 (ja) | 2003-10-14 |
| NO20011654L (no) | 2001-05-30 |
| PE20001059A1 (es) | 2000-10-23 |
| CN1328548A (zh) | 2001-12-26 |
| AR023332A1 (es) | 2002-09-04 |
| US6670381B2 (en) | 2003-12-30 |
| PL347152A1 (en) | 2002-03-25 |
| TR200100906T2 (tr) | 2001-07-23 |
| CO5140085A1 (es) | 2002-03-22 |
| NZ510839A (en) | 2003-08-29 |
| WO2000020394A1 (en) | 2000-04-13 |
| GB9821483D0 (en) | 1998-11-25 |
| EP1117644A1 (en) | 2001-07-25 |
| US6441008B1 (en) | 2002-08-27 |
| HUP0103744A2 (hu) | 2002-02-28 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK2253620T3 (da) | Substituerede 3-cyanoquinoliner som protein-tyrosinkinase-inhibitorer | |
| NO20030867D0 (no) | Hydroksamderivater anvendelig som deacetylaseinhibitorer | |
| DK1244647T3 (da) | Quinzolinderivater som VIGF-inhibitorer | |
| NO20014483D0 (no) | Aminderivater som proteaseinhibitorer | |
| NO992725L (no) | 6-Fenylpyridyl-2-amin-derivater anvendelige som NOS-inhibitorer | |
| NO20010686D0 (no) | Hydroksypipecolathydroksaminsyrederivater som MMP inhibitorer | |
| NO20031540D0 (no) | Benzamidforbindelser som Apo-B-sekresjonsinhibitorer | |
| NO20002958D0 (no) | Benzamidinderivater som koagulasjonsfaktor Xa-hemmere | |
| NO20021239D0 (no) | Pteridinoner som kinase-inhibitorer | |
| NO20012980D0 (no) | Proteaseinhibitorer | |
| DK1460066T3 (da) | Piperazinforbindelse som tachykinin-inhibitorer | |
| NO20015065D0 (no) | Pyrazolobenzodiazepiner som CDK2-inhibitorer | |
| DK1097127T3 (da) | Diacylhydrazinderivater som integrininhibitorer | |
| ATE460424T1 (de) | Factor viia inhibitore | |
| NO20024997D0 (no) | 2-guanidino-4-arylkinazoliner som NHE-3-inhibitorer | |
| NO20004696L (no) | Kinoloner som serinproteaseinhibitorer | |
| NO20021407D0 (no) | Bifenylderivater anvendt som NHE-3-inhibitorer | |
| NO994103D0 (no) | Reverse hydroksamatderivater som metallproteaseinhibitorer | |
| NO20001924L (no) | Isoquinoliner som urokinase-inhibitorer | |
| NO20016201D0 (no) | Tienopyrimidiner som fosfodiesteraseinhibitorer | |
| NO20003814D0 (no) | Trombininhibitorer | |
| NO20014875D0 (no) | Promedikamenter for trombin inhibitorer | |
| NO20021959L (no) | Tetrahydrotiopyranftalazinon-derivater som PDE4-inhibitorer | |
| NO991994D0 (no) | Substituerte 4-bifenyl-4-hydroksysm°rsyrederivater som matriks-metalloproteaseinhibitorer | |
| NO20005301D0 (no) | Pyrrolidiner som inhibitorer av neuraminidaser |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |