NO20002800L - Cyklosporinholdig mikroemulsjon, for konsentratsammensetning - Google Patents

Cyklosporinholdig mikroemulsjon, for konsentratsammensetning

Info

Publication number
NO20002800L
NO20002800L NO20002800A NO20002800A NO20002800L NO 20002800 L NO20002800 L NO 20002800L NO 20002800 A NO20002800 A NO 20002800A NO 20002800 A NO20002800 A NO 20002800A NO 20002800 L NO20002800 L NO 20002800L
Authority
NO
Norway
Prior art keywords
cyclosporin
concentrate composition
containing microemulsion
microemulsion
concentrate
Prior art date
Application number
NO20002800A
Other languages
English (en)
Other versions
NO20002800D0 (no
Inventor
Ii Chung Hong
Jung Woo Kim
Nam Hee Choi
Hee Jong Shin
Su Geun Yang
Original Assignee
Chong Kun Dang Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from KR1019980015309A external-priority patent/KR19990076462A/ko
Priority claimed from KR1019980024207A external-priority patent/KR19990066706A/ko
Application filed by Chong Kun Dang Corp filed Critical Chong Kun Dang Corp
Publication of NO20002800D0 publication Critical patent/NO20002800D0/no
Publication of NO20002800L publication Critical patent/NO20002800L/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13Cyclosporins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Dispersion Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Transplantation (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO20002800A 1997-12-05 2000-05-31 Cyklosporinholdig mikroemulsjon, for konsentratsammensetning NO20002800L (no)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
KR19970066454 1997-12-05
KR19980010046 1998-03-24
KR1019980015309A KR19990076462A (ko) 1997-12-05 1998-04-29 사이클로스포린-함유 마이크로에멀젼 예비농축액 조성물
KR1019980024207A KR19990066706A (ko) 1997-03-24 1998-06-25 사이클로스포린-함유 마이크로에멀젼 예비농축액 조성물
PCT/KR1998/000315 WO1999000002A2 (en) 1997-12-05 1998-10-16 Cyclosporin-containing microemulsion preconcentrate composition

Publications (2)

Publication Number Publication Date
NO20002800D0 NO20002800D0 (no) 2000-05-31
NO20002800L true NO20002800L (no) 2000-08-03

Family

ID=27483248

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20002800A NO20002800L (no) 1997-12-05 2000-05-31 Cyklosporinholdig mikroemulsjon, for konsentratsammensetning

Country Status (15)

Country Link
US (1) US6063762A (no)
EP (1) EP1035862B1 (no)
JP (1) JP2001517602A (no)
CN (1) CN1280502A (no)
AR (1) AR017801A1 (no)
AT (1) ATE244573T1 (no)
AU (1) AU9465898A (no)
BR (1) BR9815350A (no)
CA (1) CA2313015A1 (no)
DE (1) DE69816335T2 (no)
HU (1) HUP0004379A2 (no)
IL (1) IL136444A0 (no)
NO (1) NO20002800L (no)
NZ (1) NZ504844A (no)
WO (1) WO1999000002A2 (no)

Families Citing this family (36)

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Publication number Priority date Publication date Assignee Title
GB9325445D0 (en) 1993-12-13 1994-02-16 Cortecs Ltd Pharmaceutical formulations
US5858401A (en) * 1996-01-22 1999-01-12 Sidmak Laboratories, Inc. Pharmaceutical composition for cyclosporines
US6465016B2 (en) * 1996-08-22 2002-10-15 Research Triangle Pharmaceuticals Cyclosporiine particles
AU729724B2 (en) * 1997-04-18 2001-02-08 Taisho Pharmaceutical Co., Ltd. Microemulsion
CA2313024C (en) * 1997-12-10 2008-06-03 Severson, Mary L. Pharmaceutical compositions containing an omega-3 fatty acid oil
ID25908A (id) * 1998-03-06 2000-11-09 Novartis Ag Prakonsentrat-prakonsentrat emulsi yang mengandung siklosporin atau makrolida
GB2380674B (en) * 1998-03-06 2003-05-28 Novartis Ag Emulsion preconcentrates containing cyclosporin or a macrolide
JP2002516267A (ja) 1998-05-29 2002-06-04 アールティーピー・ファーマ・インコーポレーテッド 熱的に保護された微粒子組成物及びその最終蒸気滅菌
EE05190B1 (et) 1998-11-20 2009-08-17 Rtp Pharma Inc. Dispergeeruvad fosfolipiididega stabiliseeritud mikroosakesed
SE9804192D0 (sv) * 1998-12-03 1998-12-03 Scotia Lipidteknik Ab New formulation
US6267985B1 (en) * 1999-06-30 2001-07-31 Lipocine Inc. Clear oil-containing pharmaceutical compositions
GB9912476D0 (en) 1999-05-28 1999-07-28 Novartis Ag Organic compounds
JP2003501376A (ja) * 1999-06-04 2003-01-14 スカイファーマ インコーポレーテッド 疎水性薬物の持続性放出のための油コア組成物
AU2003254754B2 (en) * 1999-08-17 2006-01-12 Ivax Pharmaceuticals, S.R.O. Pharmaceutical compositions for oral and topical administration
GB2355656B (en) * 1999-08-17 2004-04-07 Galena As Pharmaceutical compositions for oral and topical administration
EP1214059B1 (en) * 1999-09-21 2005-05-25 Skyepharma Canada Inc. Surface modified particulate compositions of biologically active substances
AU7638300A (en) * 1999-10-20 2001-04-30 Vesifact Ag Microemulsion preconcentrates and microemulsions
US7732404B2 (en) * 1999-12-30 2010-06-08 Dexcel Ltd Pro-nanodispersion for the delivery of cyclosporin
US6623765B1 (en) * 2000-08-01 2003-09-23 University Of Florida, Research Foundation, Incorporated Microemulsion and micelle systems for solubilizing drugs
JP4391673B2 (ja) * 2000-08-08 2009-12-24 花王株式会社 油脂組成物
EA200301139A1 (ru) 2001-06-21 2004-12-30 Пфайзер Продактс Инк. Самоэмульгирующиеся препараты ингибиторов белка-переносчика эфиров холестерина
US6960563B2 (en) * 2001-08-31 2005-11-01 Morton Grove Pharmaceuticals, Inc. Spontaneous emulsions containing cyclosporine
US6479060B1 (en) 2001-09-04 2002-11-12 Healthpoint, Ltd. Elegant hydrogenated castor oil ointments
IL160761A0 (en) * 2001-10-19 2004-08-31 Isotechnika Inc Novel cyclosporin analog microemulsion preconcentrates
ITBS20010111A1 (it) * 2001-12-20 2003-06-20 Paoli Ambrosi Gianfranco De Composizione per uso topico a base dell'estere etilico dell'acido linoleico e e del trietil estere dell'acido citrico associati con opportun
US7182950B2 (en) * 2002-06-12 2007-02-27 Nutralease Ltd. Nano-sized self-assembled liquid dilutable vehicles
DE10226990A1 (de) * 2002-06-18 2004-03-18 Sanguibiotech Ag Topisch applizierbare Mikro-Emulsionen mit binärer Phasen- und Wirkstoffdifferenzierbarkeit, deren Herstellung und deren Verwendung, insbesondere zur Versorgung der Haut mit bioverfügbarem Sauerstoff
MX2007011250A (es) * 2005-03-21 2007-11-14 Ivax Pharmaceuticals Sro Inhibidor de la cristalizacion y su uso en capsulas de gelatina.
CN100478025C (zh) * 2005-03-25 2009-04-15 中国科学院上海药物研究所 一种环孢菌素a眼用微乳制剂及其制备方法
JP4842553B2 (ja) * 2005-03-30 2011-12-21 株式会社ナリス化粧品 ヒドロキシカルボン酸エステルを用いてナノ乳化粒子を安定化させる方法及びナノ乳化粒子を含有する皮膚外用剤
JP2009517410A (ja) * 2005-11-30 2009-04-30 ジェネレクス ファーマシューティカルズ インコーポレイテッド 経口吸収される医薬製剤および投与方法
US11311477B2 (en) 2006-03-07 2022-04-26 Sgn Nanopharma Inc. Ophthalmic preparations
AU2007224006A1 (en) * 2006-03-07 2007-09-13 Novavax, Inc. Nanoemulsions of poorly soluble pharmaceutical active ingredients and methods of making the same
US10137083B2 (en) 2006-03-07 2018-11-27 SGN Nanopharma Inc Ophthalmic preparations
WO2008058366A1 (en) * 2006-09-28 2008-05-22 Université de Montréal Oil-in-water emulsions, methods of use thereof, methods of preparation thereof and kits thereof
EP2200613B1 (en) 2007-09-21 2018-09-05 The Johns Hopkins University Phenazine derivatives and uses thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2907460A1 (de) * 1978-03-07 1979-09-13 Sandoz Ag Neue resorbierbare galenische kompositionen
US5639724A (en) * 1984-07-24 1997-06-17 Sandoz Ltd. Cyclosporin galenic forms
KR0148748B1 (ko) * 1988-09-16 1998-08-17 장 크라메르, 한스 루돌프 하우스 사이클로스포린을 함유하는 약학조성물
US5342625A (en) * 1988-09-16 1994-08-30 Sandoz Ltd. Pharmaceutical compositions comprising cyclosporins
IT1256386B (it) * 1992-11-13 1995-12-04 Luigi Boltri Composizioni farmaceutiche comprendenti un farmaco,una sostanza polimerica reticolata,un olio ed un agente tensioattivo
US5639474A (en) * 1993-07-01 1997-06-17 Hanmi Pharm. Ind., Ltd. Cyclosporin soft capsule composition
GB9405304D0 (en) * 1994-03-16 1994-04-27 Scherer Ltd R P Delivery systems for hydrophobic drugs
HU215966B (hu) * 1994-11-21 1999-07-28 BIOGAL Gyógyszergyár Rt. Orálisan alkalmazható, ciklosporint tartalmazó, összetett emulzió-előkoncentrátum
EP0760237A1 (en) * 1995-08-30 1997-03-05 Cipla Limited Oil-in-water microemulsions

Also Published As

Publication number Publication date
BR9815350A (pt) 2001-10-16
HUP0004379A2 (hu) 2001-08-28
CN1280502A (zh) 2001-01-17
ATE244573T1 (de) 2003-07-15
CA2313015A1 (en) 1999-01-07
DE69816335D1 (de) 2003-08-14
IL136444A0 (en) 2001-06-14
NZ504844A (en) 2001-11-30
EP1035862B1 (en) 2003-07-09
US6063762A (en) 2000-05-16
DE69816335T2 (de) 2004-04-15
JP2001517602A (ja) 2001-10-09
WO1999000002A2 (en) 1999-01-07
WO1999000002A3 (en) 1999-03-25
EP1035862A2 (en) 2000-09-20
NO20002800D0 (no) 2000-05-31
AR017801A1 (es) 2001-10-24
AU9465898A (en) 1999-01-19

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