GB2380674B - Emulsion preconcentrates containing cyclosporin or a macrolide - Google Patents

Emulsion preconcentrates containing cyclosporin or a macrolide

Info

Publication number
GB2380674B
GB2380674B GB0229289A GB0229289A GB2380674B GB 2380674 B GB2380674 B GB 2380674B GB 0229289 A GB0229289 A GB 0229289A GB 0229289 A GB0229289 A GB 0229289A GB 2380674 B GB2380674 B GB 2380674B
Authority
GB
United Kingdom
Prior art keywords
macrolide
containing cyclosporin
emulsion preconcentrates
preconcentrates containing
emulsion
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Revoked
Application number
GB0229289A
Other versions
GB0229289D0 (en
GB2380674A (en
Inventor
Michael Ambuehl
Barbara Lueckel
Friedrich Richter
Barbara Haeberlin
Armin Meinzer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27447881&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GB2380674(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9804742.6A external-priority patent/GB9804742D0/en
Priority claimed from GBGB9805104.8A external-priority patent/GB9805104D0/en
Priority claimed from GBGB9805199.8A external-priority patent/GB9805199D0/en
Application filed by Novartis AG filed Critical Novartis AG
Priority claimed from GB0021495A external-priority patent/GB2350791B/en
Publication of GB0229289D0 publication Critical patent/GB0229289D0/en
Publication of GB2380674A publication Critical patent/GB2380674A/en
Application granted granted Critical
Publication of GB2380674B publication Critical patent/GB2380674B/en
Anticipated expiration legal-status Critical
Revoked legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13Cyclosporins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Dispersion Chemistry (AREA)
  • Transplantation (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Medicinal Preparation (AREA)
GB0229289A 1998-03-06 1999-03-04 Emulsion preconcentrates containing cyclosporin or a macrolide Revoked GB2380674B (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GBGB9804742.6A GB9804742D0 (en) 1998-03-06 1998-03-06 Organic compounds
GBGB9805104.8A GB9805104D0 (en) 1998-03-10 1998-03-10 Organic compounds
GBGB9805199.8A GB9805199D0 (en) 1998-03-11 1998-03-11 Organic compounds
GB0021495A GB2350791B (en) 1998-03-06 1999-03-04 Emulsion preconcentrates containing cyclosporin or a macrolide

Publications (3)

Publication Number Publication Date
GB0229289D0 GB0229289D0 (en) 2003-01-22
GB2380674A GB2380674A (en) 2003-04-16
GB2380674B true GB2380674B (en) 2003-05-28

Family

ID=27447881

Family Applications (2)

Application Number Title Priority Date Filing Date
GB0229289A Revoked GB2380674B (en) 1998-03-06 1999-03-04 Emulsion preconcentrates containing cyclosporin or a macrolide
GB0229284A Expired - Fee Related GB2380673B (en) 1998-03-06 1999-03-04 Emulsion preconcentrates containing cyclosporin or a macrolide

Family Applications After (1)

Application Number Title Priority Date Filing Date
GB0229284A Expired - Fee Related GB2380673B (en) 1998-03-06 1999-03-04 Emulsion preconcentrates containing cyclosporin or a macrolide

Country Status (1)

Country Link
GB (2) GB2380674B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8535716B2 (en) 2004-04-01 2013-09-17 Tsrl, Inc. Methods and composition of extended delivery of water insoluble drugs
EP2204167A1 (en) * 2009-01-05 2010-07-07 Azad Pharma AG Pharmaceutical microemulsion for preventing supramolecular aggregation of amphiphilic molecules
JP5717034B2 (en) * 2012-08-27 2015-05-13 丸和バイオケミカル株式会社 Soil nematode control agent containing macrolide compounds

Citations (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2222770A (en) * 1988-09-16 1990-03-21 Sandoz Ltd Cyclosporin emulsion compositions
GB2278780A (en) * 1993-05-27 1994-12-14 Sandoz Ltd Macrolide antibiotic emulsions
WO1996013273A1 (en) * 1994-10-26 1996-05-09 Novartis Ag Pharmaceutical compositions
US5639724A (en) * 1984-07-24 1997-06-17 Sandoz Ltd. Cyclosporin galenic forms
EP0793966A1 (en) * 1996-03-05 1997-09-10 Hanmi Pharm. Co. Ltd Cyclosporin-containing topical pharmaceutical composition
WO1998010747A1 (en) * 1996-09-12 1998-03-19 Galena As Immunomodulatory formulation
WO1998041225A1 (en) * 1997-03-14 1998-09-24 Novartis Ag Pharmaceutical compositions
WO1999000002A2 (en) * 1997-12-05 1999-01-07 Chong Kun Dang Corp. Cyclosporin-containing microemulsion preconcentrate composition
EP1142568A1 (en) * 1992-09-25 2001-10-10 Novartis AG Pharmaceutical compositions containing cyclosporins

Patent Citations (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5639724A (en) * 1984-07-24 1997-06-17 Sandoz Ltd. Cyclosporin galenic forms
GB2222770A (en) * 1988-09-16 1990-03-21 Sandoz Ltd Cyclosporin emulsion compositions
EP1142568A1 (en) * 1992-09-25 2001-10-10 Novartis AG Pharmaceutical compositions containing cyclosporins
GB2278780A (en) * 1993-05-27 1994-12-14 Sandoz Ltd Macrolide antibiotic emulsions
WO1996013273A1 (en) * 1994-10-26 1996-05-09 Novartis Ag Pharmaceutical compositions
EP0793966A1 (en) * 1996-03-05 1997-09-10 Hanmi Pharm. Co. Ltd Cyclosporin-containing topical pharmaceutical composition
WO1998010747A1 (en) * 1996-09-12 1998-03-19 Galena As Immunomodulatory formulation
WO1998041225A1 (en) * 1997-03-14 1998-09-24 Novartis Ag Pharmaceutical compositions
WO1999000002A2 (en) * 1997-12-05 1999-01-07 Chong Kun Dang Corp. Cyclosporin-containing microemulsion preconcentrate composition

Also Published As

Publication number Publication date
GB2380673A (en) 2003-04-16
GB0229289D0 (en) 2003-01-22
GB2380673B (en) 2003-05-28
GB0229284D0 (en) 2003-01-22
GB2380674A (en) 2003-04-16

Similar Documents

Publication Publication Date Title
GB2350791B (en) Emulsion preconcentrates containing cyclosporin or a macrolide
PL348333A1 (en) Macrolides
CZ20011273A3 (en) Stabilized shampoo containing siloxysilicates
DE69818977D1 (en) 3'-n-oxid,3'-n-dimethylamin,9-oxime erythromycin a derivate
EP1091212A4 (en) Acceleration sensor
ZA989835B (en) Erythromycin a derivatives
GB2380673B (en) Emulsion preconcentrates containing cyclosporin or a macrolide
IL139501A0 (en) Microemulsion preconcentrates containing a piperidin substance p antagonist
SI1059913T1 (en) Emulsion preconcentrates containing cyclosporin or a macrolide
PL335369A1 (en) Acarbosic claster from actinoplanes sp. se 50/110
HK1056310A1 (en) Emulsion preconcentrates containing cyclosporin ora macrolide.
GB2315216B (en) Microemulsion preconcentrates comprising FK506 or 33-epi-chloro-33-desoxy-ascomycin
DK1059913T3 (en) Emulsion preconcentrates containing cyclosporin or a macrolide
DE19882184T1 (en) Preparation containing cyclosporin
PL342742A1 (en) Emulsion-type pre-concentrates containing cyclosporin or macrolyde
GB2313642B (en) Bucket tappet guide
SI1066304T1 (en) Macrolide lhrh antagonists
SI1082119T1 (en) Microemulsion preconcentrates containing a piperidine substance p antagonist
AU139241S (en) A console
AU139648S (en) A console
GB9824413D0 (en) A map device
TW397234U (en) A map capable of distinguishing a direction
TW325092U (en) Retaining block structure having water-drainage function for us
GB9817874D0 (en) Navigation plotter
AU134353S (en) A grommet

Legal Events

Date Code Title Description
REG Reference to a national code

Ref country code: HK

Ref legal event code: GR

Ref document number: 1056310

Country of ref document: HK

7276 Counter claim for revocation lodged in the pat. court (section 72)
772B Case decided by the comptroller ** patent revoked (sect. 72/1977)

Free format text: PATENT REVOKED