NO154194C - Analogifremgangsmaate til fremstilling av terapeutisk aktive diaryloktahydropyrazinopyrimidoner - Google Patents

Analogifremgangsmaate til fremstilling av terapeutisk aktive diaryloktahydropyrazinopyrimidoner

Info

Publication number
NO154194C
NO154194C NO782995A NO782995A NO154194C NO 154194 C NO154194 C NO 154194C NO 782995 A NO782995 A NO 782995A NO 782995 A NO782995 A NO 782995A NO 154194 C NO154194 C NO 154194C
Authority
NO
Norway
Prior art keywords
hydropyrazinopyrimidones
diarylocta
preparation
therapeutically active
analogue procedure
Prior art date
Application number
NO782995A
Other languages
English (en)
Norwegian (no)
Other versions
NO782995L (no
NO154194B (no
Inventor
Anders Karl Konrad Bjoerk
Bengt Eric Sigvard Kjellberg
Aina Lisbeth Abramo
Sven Erik Harry Hernestam
Original Assignee
Ferrosan Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferrosan Ab filed Critical Ferrosan Ab
Publication of NO782995L publication Critical patent/NO782995L/no
Publication of NO154194B publication Critical patent/NO154194B/no
Publication of NO154194C publication Critical patent/NO154194C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/12Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Anesthesiology (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO782995A 1977-09-05 1978-09-01 Analogifremgangsmaate til fremstilling av terapeutisk aktive diaryloktahydropyrazinopyrimidoner NO154194C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB3690477 1977-09-05

Publications (3)

Publication Number Publication Date
NO782995L NO782995L (no) 1979-03-06
NO154194B NO154194B (no) 1986-04-28
NO154194C true NO154194C (no) 1986-08-06

Family

ID=10392108

Family Applications (1)

Application Number Title Priority Date Filing Date
NO782995A NO154194C (no) 1977-09-05 1978-09-01 Analogifremgangsmaate til fremstilling av terapeutisk aktive diaryloktahydropyrazinopyrimidoner

Country Status (17)

Country Link
US (1) US4183933A (de)
JP (1) JPS5452097A (de)
AT (1) AT364365B (de)
BE (1) BE870227A (de)
CA (1) CA1102323A (de)
CH (1) CH637133A5 (de)
DE (1) DE2837089A1 (de)
DK (1) DK149365C (de)
ES (1) ES473070A1 (de)
FI (1) FI65621C (de)
FR (1) FR2401923A1 (de)
IT (1) IT1159108B (de)
LU (1) LU80192A1 (de)
MX (1) MX5281E (de)
NL (1) NL7809016A (de)
NO (1) NO154194C (de)
SE (1) SE442115B (de)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3560503A (en) * 1968-09-18 1971-02-02 Council Scient Ind Res Di-lower alkyl-substituted octahydropyrazinopyrimidinones
US3752816A (en) * 1969-06-10 1973-08-14 Sherwin Williams Co Certain 3-substituted-pyrido(3,2-d)pyrimidine 2,4-(1h,3h)-diones
GB1284582A (en) * 1969-11-10 1972-08-09 Council Scient Ind Res Substituted piperazinopyrimidinones
FR2103465A1 (en) * 1970-08-24 1972-04-14 Hokuriku Pharmaceutical Benzhydril-pyridodiazepines - as antihistaminics and anticholinergics from dihaloalkylpiperidines and arylalkylamines with condensing agent
US3965257A (en) * 1972-01-28 1976-06-22 Richardson-Merrell Inc. Compositions and methods for the treatment of the symptoms of histamine induced allergic reactions
US3922275A (en) * 1972-11-09 1975-11-25 Hisamitsu Pharmaceutical Co Pyrido{8 2,3-D{9 {0 pyrimidine-2,4(1H,3H)-diones
DE2523730A1 (de) * 1974-06-12 1976-02-12 Hisamitsu Pharmaceutical Co Pyrido eckige klammer auf 2,3-d eckige klammer zu pyrimidinonen

Also Published As

Publication number Publication date
BE870227A (fr) 1979-03-05
FI65621B (fi) 1984-02-29
ATA638178A (de) 1981-03-15
DE2837089A1 (de) 1979-03-22
MX5281E (es) 1983-06-02
IT7827103A0 (it) 1978-08-29
JPS5452097A (en) 1979-04-24
AT364365B (de) 1981-10-12
US4183933A (en) 1980-01-15
CH637133A5 (de) 1983-07-15
LU80192A1 (de) 1979-06-01
IT1159108B (it) 1987-02-25
FR2401923B1 (de) 1982-05-14
FI65621C (fi) 1984-06-11
SE7809288L (sv) 1979-03-06
FR2401923A1 (fr) 1979-03-30
JPS5725555B2 (de) 1982-05-29
FI782370A7 (fi) 1979-03-06
DK149365C (da) 1986-11-24
NO782995L (no) 1979-03-06
CA1102323A (en) 1981-06-02
DK149365B (da) 1986-05-20
NO154194B (no) 1986-04-28
DK386778A (da) 1979-03-06
SE442115B (sv) 1985-12-02
NL7809016A (nl) 1979-03-07
ES473070A1 (es) 1979-04-01

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