NO147483C - Analogifremgangsmaate for fremstilling av farmakologisk aktive benzylpyrimidiner. - Google Patents

Analogifremgangsmaate for fremstilling av farmakologisk aktive benzylpyrimidiner.

Info

Publication number
NO147483C
NO147483C NO780743A NO780743A NO147483C NO 147483 C NO147483 C NO 147483C NO 780743 A NO780743 A NO 780743A NO 780743 A NO780743 A NO 780743A NO 147483 C NO147483 C NO 147483C
Authority
NO
Norway
Prior art keywords
benzylpyrimidines
preparation
pharmacologically active
analogue procedure
analogue
Prior art date
Application number
NO780743A
Other languages
English (en)
Norwegian (no)
Other versions
NO780743L (no
NO147483B (no
Inventor
Peter Scharwaechter
Klaus Gutsche
Friedrich-Wilhelm Kohlmann
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of NO780743L publication Critical patent/NO780743L/no
Publication of NO147483B publication Critical patent/NO147483B/no
Publication of NO147483C publication Critical patent/NO147483C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO780743A 1977-03-05 1978-03-03 Analogifremgangsmaate for fremstilling av farmakologisk aktive benzylpyrimidiner. NO147483C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19772709634 DE2709634A1 (de) 1977-03-05 1977-03-05 Benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Publications (3)

Publication Number Publication Date
NO780743L NO780743L (no) 1978-09-06
NO147483B NO147483B (no) 1983-01-10
NO147483C true NO147483C (no) 1983-04-20

Family

ID=6002850

Family Applications (1)

Application Number Title Priority Date Filing Date
NO780743A NO147483C (no) 1977-03-05 1978-03-03 Analogifremgangsmaate for fremstilling av farmakologisk aktive benzylpyrimidiner.

Country Status (20)

Country Link
US (1) US4189581A (de)
JP (1) JPS53130681A (de)
AT (1) AT361490B (de)
BE (1) BE864484A (de)
CA (1) CA1113932A (de)
CH (1) CH634566A5 (de)
DE (1) DE2709634A1 (de)
DK (1) DK142848C (de)
FI (1) FI780693A (de)
FR (1) FR2382444A1 (de)
GB (1) GB1596813A (de)
IE (1) IE46420B1 (de)
IL (1) IL54105A (de)
IN (1) IN149534B (de)
LU (1) LU79168A1 (de)
NL (1) NL7802380A (de)
NO (1) NO147483C (de)
SE (1) SE7802343L (de)
YU (1) YU47478A (de)
ZA (1) ZA781242B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3045720A1 (de) 1980-12-04 1982-07-08 Basf Ag, 6700 Ludwigshafen N-pyrimidinyl-carbaminsaeureester, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
US4672065A (en) * 1982-11-19 1987-06-09 Chevron Research Company N-substituted phenoxyacetamide fungicides
FR2609987A1 (fr) * 1987-01-26 1988-07-29 Carraz Gilbert Nouvel amide de l'amino-2-pyrimidine et compositions pharmaceutiques tranquillisantes et antisenescentes le contenant
ES2314106T3 (es) * 2001-10-17 2009-03-16 BOEHRINGER INGELHEIM PHARMA GMBH & CO.KG Derivados de pirimidina, agentes farmaceuticos que contiene dichos compuestos, uso y metodo para su obtencion.
US6884880B2 (en) * 2002-08-21 2005-04-26 Ash Stevens, Inc. Process for the preparation of 9-β-anomeric nucleoside analogs
RO122912B8 (ro) * 2005-02-18 2010-09-30 Arpida Ag Procedeu de preparare a unui derivat de 2h-cromen
US7855285B2 (en) * 2005-06-14 2010-12-21 Brigham Young University Methods for selective N-9 glycosylation of purines
CA2620129C (en) * 2005-09-01 2014-12-23 F. Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 modulators

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH507243A (it) * 1969-04-01 1971-05-15 Dompe Farmaceutici Spa Procedimento per la preparazione di 2,4-diamino-5-(-3,4,5-trimetossibenzil)-pirimidina
US3919229A (en) * 1973-07-19 1975-11-11 Labaz Pyrimidine derivatives and process for preparing the same

Also Published As

Publication number Publication date
DK142848C (da) 1981-08-24
IL54105A0 (en) 1978-04-30
CA1113932A (en) 1981-12-08
CH634566A5 (de) 1983-02-15
US4189581A (en) 1980-02-19
IN149534B (de) 1982-01-09
NO780743L (no) 1978-09-06
NL7802380A (nl) 1978-09-07
LU79168A1 (de) 1978-06-28
FI780693A (fi) 1978-09-06
ATA154278A (de) 1980-08-15
IE46420B1 (en) 1983-06-01
AT361490B (de) 1981-03-10
DK97578A (da) 1978-09-06
IL54105A (en) 1982-04-30
FR2382444A1 (fr) 1978-09-29
DE2709634A1 (de) 1978-09-07
IE780400L (en) 1978-09-05
BE864484A (fr) 1978-09-04
GB1596813A (en) 1981-09-03
FR2382444B1 (de) 1980-08-29
JPS53130681A (en) 1978-11-14
YU47478A (en) 1983-01-21
SE7802343L (sv) 1978-09-06
ZA781242B (en) 1979-03-28
DK142848B (da) 1981-02-09
NO147483B (no) 1983-01-10

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