NO137692C - Analogifremgangsmaate ved fremstilling av terapeutisk aktive benzodiazepinderivater - Google Patents

Analogifremgangsmaate ved fremstilling av terapeutisk aktive benzodiazepinderivater

Info

Publication number
NO137692C
NO137692C NO742738A NO742738A NO137692C NO 137692 C NO137692 C NO 137692C NO 742738 A NO742738 A NO 742738A NO 742738 A NO742738 A NO 742738A NO 137692 C NO137692 C NO 137692C
Authority
NO
Norway
Prior art keywords
analogical
procedures
preparation
therapeutically active
benzodiazepin
Prior art date
Application number
NO742738A
Other languages
English (en)
Norwegian (no)
Other versions
NO742738L (fr
NO137692B (no
Inventor
Robert Ye-Fong Ning
Morton A Schwartz
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO742738L publication Critical patent/NO742738L/no
Publication of NO137692B publication Critical patent/NO137692B/no
Publication of NO137692C publication Critical patent/NO137692C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
NO742738A 1973-07-27 1974-07-26 Analogifremgangsmaate ved fremstilling av terapeutisk aktive benzodiazepinderivater NO137692C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US383228A US3925358A (en) 1973-07-27 1973-07-27 1-Lower alkyl-2-substituted-1,4-benzodiazepines

Publications (3)

Publication Number Publication Date
NO742738L NO742738L (fr) 1975-02-24
NO137692B NO137692B (no) 1977-12-27
NO137692C true NO137692C (no) 1978-04-05

Family

ID=23512244

Family Applications (1)

Application Number Title Priority Date Filing Date
NO742738A NO137692C (no) 1973-07-27 1974-07-26 Analogifremgangsmaate ved fremstilling av terapeutisk aktive benzodiazepinderivater

Country Status (24)

Country Link
US (1) US3925358A (fr)
JP (1) JPS5041884A (fr)
AR (1) AR210987A1 (fr)
AT (1) AT340430B (fr)
BE (1) BE818132A (fr)
CA (1) CA1024512A (fr)
CH (1) CH602673A5 (fr)
DD (1) DD116038A5 (fr)
DE (1) DE2436147A1 (fr)
DK (1) DK138320B (fr)
ES (1) ES428597A1 (fr)
FI (1) FI57256C (fr)
FR (1) FR2238498B1 (fr)
GB (1) GB1407585A (fr)
HU (1) HU169331B (fr)
IE (1) IE39631B1 (fr)
IL (1) IL45102A (fr)
LU (1) LU70603A1 (fr)
NL (1) NL7410101A (fr)
NO (1) NO137692C (fr)
PH (1) PH11991A (fr)
PL (1) PL89890B1 (fr)
SE (1) SE419445B (fr)
ZA (1) ZA743857B (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2952279A1 (de) * 1979-12-24 1981-06-25 Kali-Chemie Pharma Gmbh, 3000 Hannover Neue 2-acylaminomethyl-1,4-benzodiazepine und deren salze sowie verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
ATE4716T1 (de) * 1979-12-24 1983-10-15 Kali-Chemie Pharma Gmbh 2-acylaminomethyl-1,4-benzodiazepine und deren salze sowie verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel.
DE3048264A1 (de) * 1980-12-20 1982-09-09 Kali-Chemie Pharma Gmbh, 3000 Hannover 2-acylaminomethyl-1,4-benzodiazepine und deren salze sowie verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3124013A1 (de) * 1981-06-19 1982-12-30 Kali-Chemie Pharma Gmbh, 3000 Hannover 2-acylaminomethyl-1,4-benzodiazepin-verbindungen sowie verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3481921A (en) * 1965-10-22 1969-12-02 Hoffmann La Roche Benzodiazepines

Also Published As

Publication number Publication date
IE39631L (en) 1975-01-27
NO742738L (fr) 1975-02-24
PL89890B1 (fr) 1976-12-31
JPS5041884A (fr) 1975-04-16
CA1024512A (fr) 1978-01-17
FI224074A (fr) 1975-01-28
ATA617074A (de) 1977-04-15
HU169331B (fr) 1976-11-28
AU7169774A (en) 1976-01-29
IE39631B1 (en) 1978-11-22
CH602673A5 (fr) 1978-07-31
AT340430B (de) 1977-12-12
FI57256B (fi) 1980-03-31
NO137692B (no) 1977-12-27
AR210987A1 (es) 1977-10-14
IL45102A0 (en) 1974-09-10
PH11991A (en) 1978-10-05
FR2238498B1 (fr) 1977-07-08
SE7409734L (fr) 1975-01-28
BE818132A (fr) 1975-01-27
ES428597A1 (es) 1976-08-16
DD116038A5 (fr) 1975-11-05
FR2238498A1 (fr) 1975-02-21
DK138320C (fr) 1979-01-22
DK402774A (fr) 1975-04-01
FI57256C (fi) 1980-07-10
DK138320B (da) 1978-08-14
LU70603A1 (fr) 1976-06-11
GB1407585A (en) 1975-09-24
DE2436147A1 (de) 1975-02-13
IL45102A (en) 1978-01-31
NL7410101A (nl) 1975-01-29
SE419445B (sv) 1981-08-03
US3925358A (en) 1975-12-09
ZA743857B (en) 1975-06-25

Similar Documents

Publication Publication Date Title
NO793013L (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive benzodiazepinderivater
NO141407C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive etylenderivater
NO139560C (no) Analogifremgangsmaate til fremstilling av terapeutisk virksomme nonapeptidamid-derivater
NO145576C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive penicillinderivater
NO138565C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive piperazinyl-propyl-1,2,4-triazolinonderivater
NO149281C (no) Analogifremgangsmaate til fremstilling av terapeutisk aktive 7alfa-metoksycephalosporinderivater
NO145056C (no) (s)-1-aryloksy-2-propanolderivater for fremstilling av terapeutisk aktive (s)-1-aryloksy-3-amino-2-propanolderivater
NO140058C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive substituerte piperidinoalkanol-oxim-derivater
NO140597C (no) Analogifremgangsmaate ved fremstillingen av terapeutisk aktive 8-azapurin-6-on-derivater
NO142303C (no) Analogifremgangsmaate til fremstilling av terapeutisk virksomme oksazolderivater
NO140057C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive alfa-aryl-4-substituerte piperidinoalkanol-derivater
NO140978C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive isokinolinderivater
NO140821C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive pyrido-pyrimidin-derivater
NO140670C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive pyrazolodiazepinderivater
NO140596C (no) Analogifremgangsmaate for fremstilling av en terapeutisk aktive hydroksyalkylxantiner
NO139386C (no) Analogifremgangsmaate for fremstilling av farmakologisk aktive imidazopyridiner
NO142260C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive tienotriazolodiazepinderivater
NO140012C (no) Analogifremgangsmaate for fremstilling av nye terapeutisk aktive derivater av naftyridin
NO143499C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive indanderivater
NO137728C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive pyrasi-4-oksyd-derivater
NO138561C (no) Analogifremgangsmaate til fremstilling av terapeutisk virksomme cykloalkylfenoksykarboksylsyrederivater
NO137692C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive benzodiazepinderivater
NO140299C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive 4-aryl-5-aminoalkyl-4-oksazolin-2-oner
NO137696C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive benzodiazepin-derivater
NO138908C (no) Analogifremgangsmaate ved fremstilling av terapeutisk aktive imidazo- og pyrazolo-isokinolinderivater