NL8202847A - Werkwijze voor het bereiden van 6-fluorsteroiden. - Google Patents
Werkwijze voor het bereiden van 6-fluorsteroiden. Download PDFInfo
- Publication number
- NL8202847A NL8202847A NL8202847A NL8202847A NL8202847A NL 8202847 A NL8202847 A NL 8202847A NL 8202847 A NL8202847 A NL 8202847A NL 8202847 A NL8202847 A NL 8202847A NL 8202847 A NL8202847 A NL 8202847A
- Authority
- NL
- Netherlands
- Prior art keywords
- formula
- fluoro
- dien
- dione
- group
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0003—Androstane derivatives
- C07J1/0033—Androstane derivatives substituted in position 17 alfa and 17 beta
- C07J1/004—Androstane derivatives substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
- C07J1/0048—Alkynyl derivatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0003—Androstane derivatives
- C07J1/0011—Androstane derivatives substituted in position 17 by a keto group
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Rheumatology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Pain & Pain Management (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US28630681 | 1981-07-24 | ||
US06/286,306 US4383947A (en) | 1981-07-24 | 1981-07-24 | Introduction of a fluorine atom |
Publications (1)
Publication Number | Publication Date |
---|---|
NL8202847A true NL8202847A (nl) | 1983-02-16 |
Family
ID=23097997
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NL8202847A NL8202847A (nl) | 1981-07-24 | 1982-07-14 | Werkwijze voor het bereiden van 6-fluorsteroiden. |
Country Status (8)
Country | Link |
---|---|
US (1) | US4383947A (xx) |
JP (3) | JPS5824595A (xx) |
CH (1) | CH651053A5 (xx) |
DE (1) | DE3226164A1 (xx) |
FR (1) | FR2530641B1 (xx) |
GB (2) | GB2102805B (xx) |
IT (1) | IT1157224B (xx) |
NL (1) | NL8202847A (xx) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS6126648U (ja) * | 1984-07-23 | 1986-02-17 | トヨタ自動車株式会社 | 室内鏡取付構造 |
JPS6126647U (ja) * | 1984-07-23 | 1986-02-17 | トヨタ自動車株式会社 | 室内鏡取付構造 |
DE3573576D1 (en) * | 1984-07-23 | 1989-11-16 | Toyota Motor Co Ltd | A rear view mirror assembly |
JPS6126649U (ja) * | 1984-07-23 | 1986-02-17 | トヨタ自動車株式会社 | 室内鏡取付構造 |
US5352809A (en) * | 1986-10-10 | 1994-10-04 | Gist-Brocades N.V. | 9-alpha-hydroxy steroids, process for their preparation, process for the preparation of the corresponding 9(11)-dehydro derivatives and pharmaceutical preparations containing such steroids |
US4936533A (en) * | 1988-11-15 | 1990-06-26 | Donnelly Corporation | Mounting assembly for vehicle accessories |
JPH0523412Y2 (xx) * | 1989-07-14 | 1993-06-15 | ||
US5100095A (en) * | 1991-03-01 | 1992-03-31 | Donnelly Corporation | Breakaway vehicle accessory mount |
CN114195844B (zh) * | 2021-12-29 | 2023-03-17 | 湖北武当安泰药业有限公司 | 一种去氢表雄酮的制备方法 |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3126375A (en) * | 1964-03-24 | Chioacyl | ||
NL245860A (xx) * | 1958-11-28 | |||
US2961441A (en) * | 1959-08-07 | 1960-11-22 | Pfizer & Co C | Process for producing 6beta-fluorosteroids |
US3014938A (en) * | 1959-09-07 | 1961-12-26 | Syntex Sa | Preparation of 16, 21-diacetate derivative of cyclopentanophenanthrene compounds |
BE642575A (xx) * | 1963-01-16 | |||
US3127428A (en) * | 1963-01-16 | 1964-03-31 | Schering Corp | Process for converting a 3-keto-delta-steroid to the corresponding 3-keto delta-compound |
US3221033A (en) * | 1964-07-07 | 1965-11-30 | Schering Corp | Novel process for the preparation of 1,5-bis-dehydro steroids |
US3980778A (en) * | 1973-10-25 | 1976-09-14 | The Upjohn Company | Anti-inflammatory steroid |
US4041055A (en) * | 1975-11-17 | 1977-08-09 | The Upjohn Company | Process for the preparation of 17α-hydroxyprogesterones and corticoids from androstenes |
DE2558088C2 (de) * | 1975-12-19 | 1985-05-30 | Schering AG, 1000 Berlin und 4709 Bergkamen | Verfahren zur Herstellung von 4-Androsten-3,17-dion-Derivaten |
US4102907A (en) * | 1977-03-07 | 1978-07-25 | The Upjohn Company | Desulfinylation process for preparing androsta-4,9(11)-diene-3,17-dione |
US4127596A (en) * | 1977-04-11 | 1978-11-28 | The Upjohn Company | Non-aromatic oxygenated strong acid dehydration of 9α-hydroxyandrostenediones |
US4188322A (en) * | 1978-04-28 | 1980-02-12 | Blasinachim S.P.A. | Process for the preparation of 6-halo-pregnanes |
FR2433536A1 (fr) * | 1978-08-16 | 1980-03-14 | Roussel Uclaf | Nouveaux derives de l'androst 4-ene, leur procede de preparation et leur application comme medicament |
-
1981
- 1981-07-24 US US06/286,306 patent/US4383947A/en not_active Expired - Lifetime
-
1982
- 1982-07-06 GB GB08219484A patent/GB2102805B/en not_active Expired
- 1982-07-13 DE DE19823226164 patent/DE3226164A1/de active Granted
- 1982-07-14 NL NL8202847A patent/NL8202847A/nl not_active Application Discontinuation
- 1982-07-16 JP JP57124289A patent/JPS5824595A/ja active Granted
- 1982-07-19 IT IT48845/82A patent/IT1157224B/it active
- 1982-07-23 CH CH4522/82A patent/CH651053A5/de not_active IP Right Cessation
- 1982-07-23 FR FR8212932A patent/FR2530641B1/fr not_active Expired
-
1984
- 1984-08-31 GB GB08421987A patent/GB2152058B/en not_active Expired
-
1989
- 1989-08-15 JP JP1211208A patent/JPH0276896A/ja active Granted
-
1991
- 1991-10-04 JP JP3257524A patent/JPH0689021B2/ja not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
CH651053A5 (de) | 1985-08-30 |
DE3226164C2 (xx) | 1992-07-02 |
JPH0517497A (ja) | 1993-01-26 |
JPH0689021B2 (ja) | 1994-11-09 |
GB2152058B (en) | 1986-01-02 |
IT1157224B (it) | 1987-02-11 |
US4383947A (en) | 1983-05-17 |
FR2530641B1 (fr) | 1987-03-06 |
JPS5824595A (ja) | 1983-02-14 |
IT8248845A0 (it) | 1982-07-19 |
GB2152058A (en) | 1985-07-31 |
DE3226164A1 (de) | 1983-02-03 |
GB2102805B (en) | 1985-09-04 |
JPH0480038B2 (xx) | 1992-12-17 |
JPH0211600B2 (xx) | 1990-03-14 |
GB2102805A (en) | 1983-02-09 |
GB8421987D0 (en) | 1984-10-03 |
JPH0276896A (ja) | 1990-03-16 |
FR2530641A1 (fr) | 1984-01-27 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
A85 | Still pending on 85-01-01 | ||
BA | A request for search or an international-type search has been filed | ||
BB | A search report has been drawn up | ||
BC | A request for examination has been filed | ||
DNT | Communications of changes of names of applicants whose applications have been laid open to public inspection |
Free format text: PHARMACIA & UPJOHN COMPANY |
|
BV | The patent application has lapsed |