NL8005491A - Heterocyclische verbindingen met therapeutische wer- king. - Google Patents

Heterocyclische verbindingen met therapeutische wer- king. Download PDF

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Publication number
NL8005491A
NL8005491A NL8005491A NL8005491A NL8005491A NL 8005491 A NL8005491 A NL 8005491A NL 8005491 A NL8005491 A NL 8005491A NL 8005491 A NL8005491 A NL 8005491A NL 8005491 A NL8005491 A NL 8005491A
Authority
NL
Netherlands
Prior art keywords
group
compounds
formula
compound
preparation
Prior art date
Application number
NL8005491A
Other languages
English (en)
Dutch (nl)
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NL8005491A publication Critical patent/NL8005491A/nl

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NL8005491A 1979-10-03 1980-10-03 Heterocyclische verbindingen met therapeutische wer- king. NL8005491A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7934347 1979-10-03
GB7934347 1979-10-03

Publications (1)

Publication Number Publication Date
NL8005491A true NL8005491A (nl) 1981-04-07

Family

ID=10508267

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8005491A NL8005491A (nl) 1979-10-03 1980-10-03 Heterocyclische verbindingen met therapeutische wer- king.

Country Status (15)

Country Link
US (1) US4324792A (es)
JP (1) JPS5690063A (es)
AU (1) AU6294580A (es)
BE (1) BE885507A (es)
DE (1) DE3037313A1 (es)
DK (1) DK420480A (es)
ES (3) ES8203855A1 (es)
FI (1) FI803127L (es)
FR (1) FR2466461A1 (es)
GB (1) GB2062626B (es)
IT (1) IT1144007B (es)
NL (1) NL8005491A (es)
NZ (1) NZ195144A (es)
SE (1) SE8006953L (es)
ZA (1) ZA806146B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT78388B (en) * 1983-04-12 1986-09-15 Smithkline Beckman Corp Dopamine-beta-hydroxylase inhibitors
US4532331A (en) * 1983-04-12 1985-07-30 Smithkline Beckman Corporation 1-Benzyl-2-aminomethyl imidazole derivatives
US4602093A (en) * 1984-02-08 1986-07-22 Merck & Co., Inc. Novel substituted imidazoles, their preparation and use
US4661602A (en) * 1985-03-29 1987-04-28 G. D. Searle & Co. Substituted alkyl imidazole derivatives
NZ238688A (en) * 1990-06-28 1992-05-26 Smithkline Beecham Corp Substituted histidines: pharmaceutical compositions, preparation and uses thereof
US5807872A (en) * 1992-12-16 1998-09-15 Schering Corporation Imidazoylalkyl substituted with a six membered nitrogen containing heterocyclic ring
US5972984A (en) * 1995-06-06 1999-10-26 Merck & Co., Inc. Inhibitors of farnesyl-protein transferase
JP2001520222A (ja) * 1997-10-22 2001-10-30 ゼネカ・リミテッド イミダゾール誘導体およびファルネシルタンパク質トランスフェラーゼインヒビターとしてのそれらの使用
WO1999020611A1 (en) 1997-10-22 1999-04-29 Zeneca Limited Imidazole derivatives and their use as farnesyl protein transferase inhibitors
EP2447263A1 (en) * 2010-09-27 2012-05-02 Bioprojet Benzazole derivatives as histamine H4 receptor ligands

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2532547A (en) * 1950-12-05 Z-aminoalkyl-glyoxaline derivatives
GB1421792A (en) * 1973-05-17 1976-01-21 Smith Kline French Lab Heterocyclic substituted-1, 1-diamino-ethylene derivatives methods for their preparation and compositions containing them
US4152443A (en) * 1973-07-13 1979-05-01 Smith Kline & French Laboratories Limited Imidazolyl thioureas, ureas and guanidines
US4006137A (en) * 1975-08-21 1977-02-01 E. R. Squibb & Sons, Inc. 2-Ethenyl imidazolium derivatives

Also Published As

Publication number Publication date
ES495589A0 (es) 1981-12-16
NZ195144A (en) 1983-02-15
ES8205204A1 (es) 1982-06-01
FI803127L (fi) 1981-04-04
FR2466461B1 (es) 1983-05-20
ES505556A0 (es) 1982-12-01
BE885507A (fr) 1981-04-02
IT8049815A0 (it) 1980-10-03
DE3037313A1 (de) 1981-04-23
GB2062626B (en) 1983-10-05
ZA806146B (en) 1982-01-27
SE8006953L (sv) 1981-04-04
GB2062626A (en) 1981-05-28
FR2466461A1 (fr) 1981-04-10
ES8203855A1 (es) 1981-12-16
DK420480A (da) 1981-04-04
US4324792A (en) 1982-04-13
ES505555A0 (es) 1982-06-01
ES8301221A1 (es) 1982-12-01
JPS5690063A (en) 1981-07-21
AU6294580A (en) 1981-04-16
IT1144007B (it) 1986-10-29

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BV The patent application has lapsed