NL7801834A - NEW OXIMES OF 3-THIADIAZOLYL THIOMETHYL 7-AMINO THIAZOLYL ACEETAMIDO CEPHALOSPORIC ACID, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS. - Google Patents

NEW OXIMES OF 3-THIADIAZOLYL THIOMETHYL 7-AMINO THIAZOLYL ACEETAMIDO CEPHALOSPORIC ACID, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS.

Info

Publication number
NL7801834A
NL7801834A NL7801834A NL7801834A NL7801834A NL 7801834 A NL7801834 A NL 7801834A NL 7801834 A NL7801834 A NL 7801834A NL 7801834 A NL7801834 A NL 7801834A NL 7801834 A NL7801834 A NL 7801834A
Authority
NL
Netherlands
Prior art keywords
aceetamido
thiomethyl
thiadiazolyl
preparation
pharmaceutical preparations
Prior art date
Application number
NL7801834A
Other languages
Dutch (nl)
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of NL7801834A publication Critical patent/NL7801834A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36Methylene radicals, substituted by sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NL7801834A 1977-02-18 1978-02-17 NEW OXIMES OF 3-THIADIAZOLYL THIOMETHYL 7-AMINO THIAZOLYL ACEETAMIDO CEPHALOSPORIC ACID, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS. NL7801834A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7704745A FR2381053A1 (en) 1977-02-18 1977-02-18 NEW OXIMES DERIVED FROM 3-THIADIAZOLYL THIOMETHYL 7-AMINOTHIAZOLYL ACETAMIDO CEPHALOSPORANIC, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICINAL PRODUCTS

Publications (1)

Publication Number Publication Date
NL7801834A true NL7801834A (en) 1978-08-22

Family

ID=9186946

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7801834A NL7801834A (en) 1977-02-18 1978-02-17 NEW OXIMES OF 3-THIADIAZOLYL THIOMETHYL 7-AMINO THIAZOLYL ACEETAMIDO CEPHALOSPORIC ACID, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS.

Country Status (23)

Country Link
JP (1) JPS53108996A (en)
AT (1) AT355722B (en)
AU (1) AU516076B2 (en)
BE (1) BE864074A (en)
CA (1) CA1132537A (en)
CH (1) CH633016A5 (en)
DE (1) DE2806226A1 (en)
DK (1) DK68978A (en)
ES (2) ES467090A1 (en)
FI (1) FI69468C (en)
FR (1) FR2381053A1 (en)
GB (1) GB1575180A (en)
GR (1) GR71703B (en)
HU (1) HU181961B (en)
IE (1) IE46651B1 (en)
IL (1) IL54043A (en)
LU (1) LU79080A1 (en)
NL (1) NL7801834A (en)
PT (1) PT67673B (en)
SE (1) SE434268B (en)
SU (1) SU841590A3 (en)
YU (1) YU41583B (en)
ZA (1) ZA78847B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE878433A (en) * 1978-08-31 1980-02-25 Fujisawa Pharmaceutical Co PROCESS FOR THE PREPARATION OF 3-CEPHEM-4-CARBOXYLIC ACID DERIVATIVES 3,7-DISUBSTITUTED, NOVEL PRODUCTS THUS OBTAINED AND THEIR USE FOR THEIR ANTIBACTERIAL ACTIVITY
BE878514A (en) * 1978-09-04 1980-02-29 Fujisawa Pharmaceutical Co PROCESS FOR THE PREPARATION OF 3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS WITH DISUBSTITUTION IN POSITIONS 3 AND 7, NOVEL PRODUCTS THUS OBTAINED AND THEIR USE FOR THEIR ANTIBACTERIAL ACTIVITY
DE2714880A1 (en) * 1977-04-02 1978-10-26 Hoechst Ag CEPHEMDER DERIVATIVES AND PROCESS FOR THEIR PRODUCTION
US4341775A (en) * 1978-09-11 1982-07-27 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds
DE2945248A1 (en) * 1978-11-13 1980-05-22 Fujisawa Pharmaceutical Co CEPHEM COMPOUNDS, METHOD FOR THEIR PRODUCTION AND ANTIBACTERIAL PHARMACEUTICAL AGENTS CONTAINING THE SAME
US4399132A (en) * 1980-08-11 1983-08-16 American Cyanamid Company 7-Beta-[alpha-syn-methoxyimino-alpha-(2-aminothiazol-4-yl)-acetamido]-3-[(1,2,3-thiadiazol-5-ylthio)methyl]-3-cephem-4-carboxylic acid and C1 -C6 alkyl derivatives thereof
US4761409A (en) * 1984-08-16 1988-08-02 Sumitomo Pharmaceuticals Company, Limited Cephem derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1399086A (en) * 1971-05-14 1975-06-25 Glaxo Lab Ltd Cephalosporin compounds
DK154939C (en) * 1974-12-19 1989-06-12 Takeda Chemical Industries Ltd METHOD OF ANALOGUE FOR THE PREPARATION OF THIAZOLYLACETAMIDO-CEPHEM COMPOUNDS OR PHARMACEUTICAL ACCEPTABLE SALTS OR ESTERS THEREOF
DK162391C (en) * 1976-04-12 1992-03-09 Fujisawa Pharmaceutical Co ANALOGY PROCEDURE FOR PREPARING SYN-ISOMERS OF 3,7-DISUBSTITUTED 3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS
DE2715385A1 (en) * 1976-04-14 1977-11-10 Takeda Chemical Industries Ltd CEPHALOSPORIN DERIVATIVES, THE PROCESS FOR THEIR MANUFACTURING AND MEDICINAL PRODUCTS CONTAINING THEM

Also Published As

Publication number Publication date
DK68978A (en) 1978-08-19
PT67673A (en) 1978-03-01
CA1132537A (en) 1982-09-28
GB1575180A (en) 1980-09-17
ES467090A1 (en) 1979-06-01
FI69468C (en) 1986-02-10
AT355722B (en) 1980-03-25
JPS53108996A (en) 1978-09-22
ZA78847B (en) 1979-03-28
AU3337578A (en) 1979-08-23
YU33678A (en) 1983-01-21
GR71703B (en) 1983-06-21
PT67673B (en) 1980-03-03
YU41583B (en) 1987-10-31
AU516076B2 (en) 1981-05-14
DE2806226A1 (en) 1978-08-24
SU841590A3 (en) 1981-06-23
FI69468B (en) 1985-10-31
IE780364L (en) 1978-08-18
ES475956A1 (en) 1979-12-16
IL54043A0 (en) 1978-04-30
HU181961B (en) 1983-11-28
CH633016A5 (en) 1982-11-15
IE46651B1 (en) 1983-08-10
ATA120978A (en) 1979-08-15
FR2381053A1 (en) 1978-09-15
SE7800790L (en) 1978-08-18
FI780444A (en) 1978-08-19
LU79080A1 (en) 1978-09-28
IL54043A (en) 1983-02-23
FR2381053B1 (en) 1979-06-01
SE434268B (en) 1984-07-16
BE864074A (en) 1978-08-17

Similar Documents

Publication Publication Date Title
NL930045I2 (en) 7-Acylamino-3-vinyl cephalosporanic acid derivatives, methods of preparation thereof, pharmaceutical preparations containing them, their starting compounds and the preparation thereof.
NL7611394A (en) PROCESS FOR THE PREPARATION OF NEW PYRIDINE DERIVES AND PHARMACEUTICAL PREPARATIONS.
NL7608856A (en) PROCESS FOR THE PREPARATION OF NEW TETRAHYDROISOCHINOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE COMPOUNDS.
NL7604944A (en) PROCESS FOR PREPARING NEW THIENOPYRIDINE DERIVATIVES AND PROCESS FOR PREPARING PHARMACEUTICAL PREPARATIONS.
NL7607159A (en) METHODS FOR THE PREPARATION AND USE OF PHENYLAIC ACID DERIVATIVES.
NL7510535A (en) PROCESS FOR THE PREPARATION OF NEW ARYLPIPERIINES, AND PROCESS FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS.
NL7804230A (en) N-ALKYL-N-ACYL DERIVATIVES OF THIENAMYCIN, METHOD OF PREPARATION THEREOF, AND PHARMACEUTICAL PREPARATIONS.
NL7811220A (en) CEPHALOSPORANIC ACID DERIVATIVES, METHODS FOR THEIR PREPARATION, PHARMACEUTICAL PREPARATIONS.
NL163425B (en) PROCESS FOR THE PREPARATION OF AQUEOUS MIXTURES OF STEROL LYCOSIDES AND THEIR ESTERS.
NL7607254A (en) PROCESS FOR THE PREPARATION OF NEW THIENOPYRIDINE DERIVATIVES AND PROCESS FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS.
NL7606612A (en) PROCESS FOR THE PREPARATION OF NEW PHARMACEUTICAL PREPARATIONS.
NL7811823A (en) NEW OXIMES PROCESS FOR THE PREPARATION OF OXYDERES AND OXIMES CONTAINING THERAPEUTIC PREPARATION.
NL7700425A (en) PROCESS FOR THE PREPARATION OF PREPARATIONS AND SUBSTANCES AGAINST STOMACH ACID AND STOMACHES.
NL7801834A (en) NEW OXIMES OF 3-THIADIAZOLYL THIOMETHYL 7-AMINO THIAZOLYL ACEETAMIDO CEPHALOSPORIC ACID, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS.
NL7801887A (en) NEW 20,21-DINOREBURNAMENINE COMPOUNDS, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS.
NL7513336A (en) NEW AMINOPROPANOL DERIVATIVES, METHOD FOR THEIR PREPARATION AND PROCEDURE FOR THE PREPARATION OF THERAPEUTIC PREPARATIONS.
NL190700B (en) SULFURIC ISOCHINOLINE DERIVATIVES, CONTAINING THIS COMPOUND, PHARMACEUTICAL PREPARATIONS AND METHOD FOR PREPARING THESE NEW COMPOUNDS.
NL7612073A (en) PROCESS FOR PREPARING NEW PENICILLINS, AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE PENICILLINS.
NL7610057A (en) PROCESS FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS.
NL7508706A (en) PROCESS FOR THE PREPARATION OF PYRAZOFURINE DERIVATIVES AND PROCESS FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS.
NL7608164A (en) PROCESS FOR PREPARING CEFEM AND PENAM COMPOUNDS, AS WELL AS PROCEDURE FOR PREPARING PHARMACEUTICAL PREPARATIONS.
NL7900721A (en) NEW DERIVATIVES OF 1-NAPHYLACACIC ACID, METHOD OF PREPARATION THEREOF, AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE COMPOUNDS.
NL7902922A (en) NEW OXIM COMPOUNDS OF 3-AZIDOMETHYL-7-AMINOTHIA-ZOLYL-ACEETAMIDOCEPHALOSPORANIC ACID, METHOD FOR THEIR PREPARATION, THEIR USE AS MEDICINAL PRODUCTS AND PHARMA-CEUTIC COMPOUNDS CONTAINING THESE COMPOUNDS.
NL7606043A (en) PROCESS FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS, AND PROCESS FOR THE PREPARATION OF NEW AMINE DERIVATIVES.
NL186699C (en) KANAMYCIN DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF, PROCESS FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS AND FORMED PHARMACEUTICAL PREPARATIONS.

Legal Events

Date Code Title Description
BV The patent application has lapsed
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
A85 Still pending on 85-01-01
BC A request for examination has been filed
BV The patent application has lapsed