NL7315350A - Nieuwe aminoguanidine verbindingen. - Google Patents

Nieuwe aminoguanidine verbindingen.

Info

Publication number
NL7315350A
NL7315350A NL7315350A NL7315350A NL7315350A NL 7315350 A NL7315350 A NL 7315350A NL 7315350 A NL7315350 A NL 7315350A NL 7315350 A NL7315350 A NL 7315350A NL 7315350 A NL7315350 A NL 7315350A
Authority
NL
Netherlands
Prior art keywords
aminoguanidine compounds
new
new aminoguanidine
compounds
aminoguanidine
Prior art date
Application number
NL7315350A
Other languages
English (en)
Dutch (nl)
Original Assignee
Akzo Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nv filed Critical Akzo Nv
Priority to NL7315350A priority Critical patent/NL7315350A/xx
Priority to AR256431A priority patent/AR205358A1/es
Priority to ZA00746701A priority patent/ZA746701B/xx
Priority to IE2173/74A priority patent/IE40409B1/xx
Priority to GB45874/74A priority patent/GB1487852A/en
Priority to US05/517,554 priority patent/US3972932A/en
Priority to DK579774AA priority patent/DK138791B/da
Priority to HU74AO00000394A priority patent/HU171856B/hu
Priority to DE19742452691 priority patent/DE2452691A1/de
Priority to CH1484974A priority patent/CH616656A5/de
Priority to FI3243/74A priority patent/FI62064C/fi
Priority to JP12882574A priority patent/JPS5546389B2/ja
Priority to BE150356A priority patent/BE822019A/xx
Priority to FR7437192A priority patent/FR2250521B1/fr
Priority to SE7414045A priority patent/SE420720B/xx
Priority to CA213,351A priority patent/CA1032962A/en
Priority to ES431775A priority patent/ES431775A1/es
Publication of NL7315350A publication Critical patent/NL7315350A/xx
Priority to US05/653,318 priority patent/US4101675A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C281/00Derivatives of carbonic acid containing functional groups covered by groups C07C269/00 - C07C279/00 in which at least one nitrogen atom of these functional groups is further bound to another nitrogen atom not being part of a nitro or nitroso group
    • C07C281/16Compounds containing any of the groups, e.g. aminoguanidine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NL7315350A 1973-11-09 1973-11-09 Nieuwe aminoguanidine verbindingen. NL7315350A (nl)

Priority Applications (18)

Application Number Priority Date Filing Date Title
NL7315350A NL7315350A (nl) 1973-11-09 1973-11-09 Nieuwe aminoguanidine verbindingen.
AR256431A AR205358A1 (es) 1973-11-09 1974-01-01 Procedimiento para la preparacion de compuestos de 1-(2,6-disubstituido fenil) - 2 - aminoguanidina
ZA00746701A ZA746701B (en) 1973-11-09 1974-10-22 Novel 2,6-disubstituted phenyl-aminoguanidine compounds
IE2173/74A IE40409B1 (en) 1973-11-09 1974-10-22 Novel 2,6-dusubstituted phenyl-aminoguanidine compounds
GB45874/74A GB1487852A (en) 1973-11-09 1974-10-23 2,6-disubstituted phenyl-aminoguanidine compounds
US05/517,554 US3972932A (en) 1973-11-09 1974-10-24 Novel 2,6-disubstituted phenyl-aminoguanidine compounds
CH1484974A CH616656A5 (esLanguage) 1973-11-09 1974-11-06
HU74AO00000394A HU171856B (hu) 1973-11-09 1974-11-06 Sposob poluchenija novykh 2,6-dvykhzamehhjonnykh v fenile proizvodnykh fenil-amino-guanidina
DE19742452691 DE2452691A1 (de) 1973-11-09 1974-11-06 2,6-disubstituierte phenylaminoguanidinverbindungen
DK579774AA DK138791B (da) 1973-11-09 1974-11-06 Analogifremgangsmåde til fremstilling af 2,6-disubstituerede fenylaminoguanidinforbindelser.
FI3243/74A FI62064C (fi) 1973-11-09 1974-11-07 Foerfarande foer framstaellning av nya 2,6-disubstituerade fenylaminoguanidinfoereningar vilka aer anvaendbara saosom blodtrycknedsaettande laekemedel
JP12882574A JPS5546389B2 (esLanguage) 1973-11-09 1974-11-08
BE150356A BE822019A (fr) 1973-11-09 1974-11-08 Nouveaux derives de phenyl(2
FR7437192A FR2250521B1 (esLanguage) 1973-11-09 1974-11-08
SE7414045A SE420720B (sv) 1973-11-09 1974-11-08 Forfarande for framstellning av 2,6-disubstuerade fenylaminoguanidinforeningar
CA213,351A CA1032962A (en) 1973-11-09 1974-11-08 2,6-disubstituted phenyl-aminoguanidine compounds
ES431775A ES431775A1 (es) 1973-11-09 1974-11-08 Procedimiento para la preparacion de derivados de 1-fenil-2-aminoguanidina.
US05/653,318 US4101675A (en) 1973-11-09 1976-01-29 Novel 2,6-di-substituted phenyl-aminoquanidine containing compositions and methods of using same and pharmaceutical compositions containing the same and therapeutic method

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
NL7315350A NL7315350A (nl) 1973-11-09 1973-11-09 Nieuwe aminoguanidine verbindingen.

Publications (1)

Publication Number Publication Date
NL7315350A true NL7315350A (nl) 1975-05-13

Family

ID=19819967

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7315350A NL7315350A (nl) 1973-11-09 1973-11-09 Nieuwe aminoguanidine verbindingen.

Country Status (17)

Country Link
US (1) US3972932A (esLanguage)
JP (1) JPS5546389B2 (esLanguage)
AR (1) AR205358A1 (esLanguage)
BE (1) BE822019A (esLanguage)
CA (1) CA1032962A (esLanguage)
CH (1) CH616656A5 (esLanguage)
DE (1) DE2452691A1 (esLanguage)
DK (1) DK138791B (esLanguage)
ES (1) ES431775A1 (esLanguage)
FI (1) FI62064C (esLanguage)
FR (1) FR2250521B1 (esLanguage)
GB (1) GB1487852A (esLanguage)
HU (1) HU171856B (esLanguage)
IE (1) IE40409B1 (esLanguage)
NL (1) NL7315350A (esLanguage)
SE (1) SE420720B (esLanguage)
ZA (1) ZA746701B (esLanguage)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4141992A (en) * 1975-08-22 1979-02-27 American Cyanamid Company Cycloalkylcarboxyamidines and halobenzamidines as anti-amebic agents
US4113776A (en) * 1976-04-15 1978-09-12 Hoffmann-La Roche Inc. 1-(2-Aminoethyl)-3-(2,6-dihalophenyl)guanidines
HU190639B (en) * 1983-12-12 1986-09-29 Gyogyszerkutato Intezet Kv,Hu Process for production of new aminoguanidin derivatives
ZA857153B (en) * 1984-09-19 1986-05-28 Ciba Geigy Ag Substituted carbodiimides
ATE59633T1 (de) * 1984-09-19 1991-01-15 Ciba Geigy Ag Substituierte carbodiimide.
JP3298875B2 (ja) 1990-03-02 2002-07-08 オレゴン州 三置換―および四置換グアニジン類およびそれらの興奮性アミノ酸アンタゴニストとしての用途
US5262568A (en) * 1990-03-02 1993-11-16 State Of Oregon Tri- and tetra-substituted guanidines and their use as excitatory amino acid antagonists
US5847006A (en) * 1991-02-08 1998-12-08 Cambridge Neuroscience, Inc. Therapeutic guanidines
DE69230220T2 (de) * 1991-02-08 2000-06-21 Cambridge Neuroscience Research, Inc. Substituierte guanidine und derivate hiervon als modulatoren der freisetzung von neurotransmittern und neue methode zur identifizierung von inhibitoren der neurotransmitter-freisetzung
US5741661A (en) * 1991-02-08 1998-04-21 Cambridge Neuroscience, Inc. Substituted guanidines and derivatives thereof as modulators of neurotransmitter release and novel methodology for identifying neurotransmitter release blockers
KR20030097618A (ko) * 1993-05-27 2003-12-31 캠브리지 뉴로사이언스, 인코포레이티드 치료용 치환 구아니딘류
EP0739200A4 (en) * 1993-11-23 1997-12-17 Cambridge Neuroscience Inc SUBSTITUTED GUANIDINES FOR THERAPEUTIC USE
US7351743B1 (en) 1994-02-03 2008-04-01 Wyeth Therapeutic guanidines
US6787569B1 (en) 1994-02-03 2004-09-07 Cambridge Neuroscience, Inc. Therapeutic guanidines
US6143791A (en) * 1994-02-03 2000-11-07 Cambridge Neuroscience, Inc. Therapeutic guanidines
KR100423272B1 (ko) 1994-02-03 2004-09-01 캠브리지 뉴로사이언스, 인코포레이티드 신경전달물질의방출을조절하는화합물,이의약학적으로허용가능한염및이를포함하는약학조성물
JP4564786B2 (ja) * 2004-06-07 2010-10-20 株式会社日本ファインケム 1−置換―1―アミノグアニジン又はその塩、及びこれらの製造方法
JP4739695B2 (ja) * 2004-06-07 2011-08-03 株式会社日本ファインケム 5−アミノ―1―置換―1,2,4―トリアゾールの製造方法、及び該製造方法で得られるトリアゾール誘導体

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB800869A (en) * 1955-09-28 1958-09-03 Ici Ltd Substituted amino-guanidines
NL7011683A (esLanguage) * 1970-08-07 1972-02-09

Also Published As

Publication number Publication date
DK579774A (esLanguage) 1975-07-07
SE420720B (sv) 1981-10-26
FI62064B (fi) 1982-07-30
IE40409L (en) 1975-05-09
SE7414045L (esLanguage) 1975-05-12
CH616656A5 (esLanguage) 1980-04-15
JPS5546389B2 (esLanguage) 1980-11-22
AR205358A1 (es) 1976-04-30
US3972932A (en) 1976-08-03
IE40409B1 (en) 1979-05-23
CA1032962A (en) 1978-06-13
GB1487852A (en) 1977-10-05
FR2250521B1 (esLanguage) 1979-03-16
ZA746701B (en) 1975-11-26
DK138791C (esLanguage) 1979-04-09
HU171856B (hu) 1978-04-28
JPS5077328A (esLanguage) 1975-06-24
FR2250521A1 (esLanguage) 1975-06-06
ES431775A1 (es) 1976-12-16
FI324374A7 (esLanguage) 1975-05-10
DE2452691A1 (de) 1975-05-15
FI62064C (fi) 1982-11-10
DK138791B (da) 1978-10-30
BE822019A (fr) 1975-05-09

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Legal Events

Date Code Title Description
BC A request for examination has been filed
BV The patent application has lapsed