NL7308483A - - Google Patents

Info

Publication number
NL7308483A
NL7308483A NL7308483A NL7308483A NL7308483A NL 7308483 A NL7308483 A NL 7308483A NL 7308483 A NL7308483 A NL 7308483A NL 7308483 A NL7308483 A NL 7308483A NL 7308483 A NL7308483 A NL 7308483A
Authority
NL
Netherlands
Application number
NL7308483A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of NL7308483A publication Critical patent/NL7308483A/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Steroid Compounds (AREA)
NL7308483A 1972-06-19 1973-06-19 NL7308483A (cg-RX-API-DMAC10.html)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2229695A DE2229695A1 (de) 1972-06-19 1972-06-19 2-(heteroaryl-methyl)-5,9 beta-dialkyl6,7-benzomorphane, deren saeureadditionssalze sowie verfahren zu deren herstellung

Publications (1)

Publication Number Publication Date
NL7308483A true NL7308483A (cg-RX-API-DMAC10.html) 1973-12-21

Family

ID=5848060

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7308483A NL7308483A (cg-RX-API-DMAC10.html) 1972-06-19 1973-06-19

Country Status (13)

Country Link
US (1) US3931194A (cg-RX-API-DMAC10.html)
JP (1) JPS5711908B2 (cg-RX-API-DMAC10.html)
AT (6) AT328627B (cg-RX-API-DMAC10.html)
BE (1) BE801079A (cg-RX-API-DMAC10.html)
CH (9) CH582698A5 (cg-RX-API-DMAC10.html)
DE (1) DE2229695A1 (cg-RX-API-DMAC10.html)
DK (1) DK136904C (cg-RX-API-DMAC10.html)
ES (8) ES416037A1 (cg-RX-API-DMAC10.html)
FR (1) FR2189056B1 (cg-RX-API-DMAC10.html)
GB (1) GB1433817A (cg-RX-API-DMAC10.html)
NL (1) NL7308483A (cg-RX-API-DMAC10.html)
NO (1) NO137694C (cg-RX-API-DMAC10.html)
SE (1) SE405121B (cg-RX-API-DMAC10.html)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2437610A1 (de) * 1974-08-05 1976-02-26 Boehringer Sohn Ingelheim Neue 5,9-beta-disubstituierte 2-tetrahydrofurfuryl-6,7-benzomorphane, deren saeureadditionssalze, ihre verwendung als arzneimittel und verfahren zu deren herstellung
GB1575009A (en) * 1976-06-21 1980-09-17 Acf Chemiefarma Nv 6,7-benzomorphan derivatives
JPS63177704A (ja) * 1987-01-16 1988-07-21 松山株式会社 農作業機連結装置
AR067673A1 (es) 2007-07-26 2009-10-21 Vitae Pharmaceuticals Inc Derivados de 1,3 oxazinan - 2 - ona como inhibidores ciclicos de la 11 beta -hidroxiesteroide deshidrogenasa 1. composiciones farmaceuticas.
AR069545A1 (es) * 2007-11-16 2010-02-03 Boehringer Ingelheim Pharma Derivados de aril y heteroarilcarbonilo de benzomorfanos y estructuras relacionadas, composiciones farmaceuticas que contienen dichos compuestos, obtencion de las mismas, su uso en el tratamiento de enfermedades mediadas por la inhibicion de la enzima 11beta-hidroxiesteroide deshidrogenasa (hsd) 1 y
US8440658B2 (en) 2007-12-11 2013-05-14 Vitae Pharmaceuticals, Inc. Cyclic urea inhibitors of 11β-hydroxysteroid dehydrogenase 1
TW200934490A (en) 2008-01-07 2009-08-16 Vitae Pharmaceuticals Inc Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1
JP5490020B2 (ja) 2008-01-24 2014-05-14 ヴァイティー ファーマシューティカルズ,インコーポレイテッド 11β−ヒドロキシステロイドデヒドロゲナーゼ1の環状カルバゼート及びセミカルバジドインヒビター
EP2245014B1 (en) * 2008-02-12 2011-11-02 Boehringer Ingelheim International GmbH Urea derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use
WO2009102460A2 (en) 2008-02-15 2009-08-20 Vitae Pharmaceuticals, Inc. Inhibitors of 11beta-hydroxysteroid dehydrogenase 1
WO2009134392A1 (en) 2008-05-01 2009-11-05 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
WO2009134387A1 (en) 2008-05-01 2009-11-05 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
MX2010011935A (es) 2008-05-01 2011-05-19 Vitae Pharmaceuticals Inc Inhibidores ciclicos de 11 beta-hidroxiesteroide deshidrogenasa 1.
JP5711115B2 (ja) 2008-05-13 2015-04-30 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ベンゾモルファン及び関連骨格のアリサイクリックカルボン酸誘導体、そのような化合物を含有する医薬及びその使用
NZ590495A (en) 2008-07-25 2012-10-26 Vitae Pharmaceuticals Inc Dihydropyridin-phenyl-3-oxazinan-2-ones as inhibitors of 11beta-hydroxysteroid dehydrogenase 1
EP2324017B1 (en) 2008-07-25 2014-12-31 Boehringer Ingelheim International GmbH INHIBITORS OF 11beta-HYDROXYSTEROID DEHYDROGENASE 1
UA109255C2 (ru) 2009-04-30 2015-08-10 Берінгер Інгельхайм Інтернешнл Гмбх Циклические ингибиторы 11бета-гидроксистероиддегидрогеназы 1
EP2440537A1 (en) 2009-06-11 2012-04-18 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1 based on the 1,3 -oxazinan- 2 -one structure
TWI531571B (zh) * 2009-11-06 2016-05-01 維它藥物公司 六氫茚并吡啶及八氫苯并喹啉之芳基-及雜芳基羰基衍生物
WO2011159760A1 (en) 2010-06-16 2011-12-22 Vitae Pharmaceuticals, Inc. Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use
TWI537258B (zh) 2010-11-05 2016-06-11 百靈佳殷格翰國際股份有限公司 六氫茚并吡啶及八氫苯并喹啉之芳基-及雜環芳基羰基衍生物
EP2744783A1 (en) 2011-08-17 2014-06-25 Boehringer Ingelheim International GmbH Indenopyridine derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE582575A (cg-RX-API-DMAC10.html) * 1958-09-22
FR1281227A (fr) * 1958-09-22 1962-01-12 Smith Kline French Lab Perfectionnements apportés aux procédés pour la préparation de dérivés d'aralcoylbenzomorphane
CS166803B2 (cg-RX-API-DMAC10.html) * 1971-02-08 1976-03-29 Boehringer Sohn Ingelheim
SE392895B (sv) * 1971-08-24 1977-04-25 Sumitomo Chemical Co Forfarande for framstellning av bensomorfanderivat och deras salter

Also Published As

Publication number Publication date
AT325218B (de) 1975-10-10
US3931194A (en) 1976-01-06
FR2189056A1 (cg-RX-API-DMAC10.html) 1974-01-25
CH583229A5 (cg-RX-API-DMAC10.html) 1976-12-31
ATA489874A (de) 1975-07-15
AT329200B (de) 1976-04-26
ES416037A1 (es) 1976-02-16
CH583227A5 (cg-RX-API-DMAC10.html) 1976-12-31
CH589649A5 (cg-RX-API-DMAC10.html) 1977-07-15
AU5704673A (en) 1974-12-19
AT328629B (de) 1976-03-25
CH583230A5 (cg-RX-API-DMAC10.html) 1976-12-31
JPS5711908B2 (cg-RX-API-DMAC10.html) 1982-03-08
ES431513A1 (es) 1976-11-01
ES431510A1 (es) 1976-11-01
ES431516A1 (es) 1976-11-16
AT328628B (de) 1976-03-25
CH589648A5 (cg-RX-API-DMAC10.html) 1977-07-15
ES431514A1 (es) 1976-11-01
SE405121B (sv) 1978-11-20
ES431515A1 (es) 1976-11-01
ATA489474A (de) 1975-06-15
JPS4961170A (cg-RX-API-DMAC10.html) 1974-06-13
ES431511A1 (es) 1976-11-01
ES431512A1 (es) 1976-11-01
CH583228A5 (cg-RX-API-DMAC10.html) 1976-12-31
DE2229695A1 (de) 1974-01-31
AT328627B (de) 1976-03-25
CH583231A5 (cg-RX-API-DMAC10.html) 1976-12-31
GB1433817A (en) 1976-04-28
BE801079A (fr) 1973-12-18
NO137694C (no) 1978-04-05
FR2189056B1 (cg-RX-API-DMAC10.html) 1976-10-22
AT329199B (de) 1976-04-26
CH582698A5 (cg-RX-API-DMAC10.html) 1976-12-15
ATA489974A (de) 1975-07-15
CH582697A5 (cg-RX-API-DMAC10.html) 1976-12-15
NO137694B (no) 1977-12-27
ATA490074A (de) 1975-06-15
DK136904C (da) 1978-06-26
DK136904B (da) 1977-12-12
ATA489774A (de) 1975-06-15

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Legal Events

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BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BV The patent application has lapsed