NL7302669A - - Google Patents

Info

Publication number
NL7302669A
NL7302669A NL7302669A NL7302669A NL7302669A NL 7302669 A NL7302669 A NL 7302669A NL 7302669 A NL7302669 A NL 7302669A NL 7302669 A NL7302669 A NL 7302669A NL 7302669 A NL7302669 A NL 7302669A
Authority
NL
Netherlands
Application number
NL7302669A
Other versions
NL179729C (nl
NL179729B (nl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of NL7302669A publication Critical patent/NL7302669A/xx
Publication of NL179729B publication Critical patent/NL179729B/xx
Application granted granted Critical
Publication of NL179729C publication Critical patent/NL179729C/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NLAANVRAGE7302669,A 1972-02-29 1973-02-26 Werkwijze ter bereiding van farmaceutische preparaten op basis van 1h-indazool-3-carbonzuurderivaten alsmede werkwijze ter bereiding van deze 1h-indazool-3-carbonzuurderivaten. NL179729C (nl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT48628/72A IT1052111B (it) 1972-02-29 1972-02-29 Acidi i benzil i h indazol 3 carbossilici sostituiti e loro derivati

Publications (3)

Publication Number Publication Date
NL7302669A true NL7302669A (de) 1973-08-31
NL179729B NL179729B (nl) 1986-06-02
NL179729C NL179729C (nl) 1986-11-03

Family

ID=11267725

Family Applications (1)

Application Number Title Priority Date Filing Date
NLAANVRAGE7302669,A NL179729C (nl) 1972-02-29 1973-02-26 Werkwijze ter bereiding van farmaceutische preparaten op basis van 1h-indazool-3-carbonzuurderivaten alsmede werkwijze ter bereiding van deze 1h-indazool-3-carbonzuurderivaten.

Country Status (9)

Country Link
US (1) US3895026A (de)
CA (1) CA994347A (de)
DE (1) DE2310031C3 (de)
FR (1) FR2181773B1 (de)
GB (1) GB1381422A (de)
HU (1) HU165172B (de)
IN (1) IN139264B (de)
IT (1) IT1052111B (de)
NL (1) NL179729C (de)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1050741B (it) * 1975-12-01 1981-03-20 Acraf Utilizzazione degli acidi i benzil ih indazol 3 carbossilici sostituiti e loro derivati nel campo della contraccezione femminile
US5229408A (en) * 1988-07-15 1993-07-20 Ici Pharma 4-carbamoyl-1,2-dihydro-3H-indazol-3-one derivatives
US5914405A (en) * 1997-10-07 1999-06-22 Eli Lilly And Company Process for preparing 3-substituted indazoles
US6001865A (en) * 1999-05-04 1999-12-14 Angelini Pharmaceuticals Inc. 3-substituted 1-benzyl-1H-indazole derivatives as antifertility agents
KR100424341B1 (ko) * 2001-10-23 2004-03-24 하나제약 주식회사 1-메틸인다졸-3-카르복실산의 제조방법
JP2006515885A (ja) * 2003-01-17 2006-06-08 スレッシュオールド ファーマシューティカルズ, インコーポレイテッド 癌の処置のための併用療法
MXPA05007572A (es) * 2003-01-17 2005-11-17 Threshold Pharmaceuticals Inc Tratamiento de hiperplasia prostatica benigna.
TW200602324A (en) * 2004-03-24 2006-01-16 Janssen Pharmaceutica Nv Tetrahydro-indazole cannabinoid modulators cross reference to related applications
WO2005120498A2 (en) * 2004-06-03 2005-12-22 Threshold Pharmaceuticals, Inc. Method for synthesis of lonidamine and related indazole derivatives
WO2006010077A2 (en) * 2004-07-08 2006-01-26 Threshold Pharmaceuticals, Inc. Prodrugs of lonidamine and lonidamine analogs
US7514463B2 (en) * 2004-08-20 2009-04-07 University Of Kansas Lonidamine analogues and their use in male contraception and cancer treatment
CN101759644B (zh) * 2005-08-17 2011-11-02 杭州民生药业有限公司 氯尼达明的结晶形式iii、其制备方法和含有所述结晶形式iii的组合物
CN101735151B (zh) * 2005-08-17 2012-07-04 杭州民生药业有限公司 氯尼达明的结晶形式i、其制备方法和含有所述结晶形式i的组合物
CN104011027A (zh) * 2009-07-06 2014-08-27 堪萨斯大学 氯尼达明类似物于生育力调节上的用途
AU2016277126A1 (en) 2015-06-12 2017-12-14 Vettore, LLC MCT4 inhibitors for treating disease
BR112019011825A2 (pt) 2016-12-12 2019-10-22 Vettore Llc composto, enantiômero isolado, composição farmacêutica, método para inibir a atividade do transportador de monocarboxilato mct4, ou um mutante do mesmo, em uma amostra biológica, método para inibir a atividade do transportador de monocarboxilato mct4, ou um mutante do mesmo, em relação ao transportador de monocarboxilato mct1, ou um mutante do mesmo, em um paciente, método para tratar um distúrbio mediado por transportador de monocarboxilato mct4 em um sujeito que necessite do mesmo, uso de um composto e método para obter um efeito em um paciente

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3007938A (en) * 1959-04-17 1961-11-07 Sterling Drug Inc 1-(3-indazolecarbonyl)-hydrazines and their preparation
US3145215A (en) * 1961-12-19 1964-08-18 Sterling Drug Inc Indazole derivatives
IL28032A (en) * 1966-08-29 1971-08-25 Acraf Indazol-3-yl-oxyalkanoic acids and process for the preparation thereof
US3567721A (en) * 1968-11-29 1971-03-02 Geigy Chem Corp Indazolecarboxylic acids and derivatives thereof
DE1948793A1 (de) * 1969-09-26 1971-04-01 Rhein Chemie Rheinau Gmbh Verfahren zur Herstellung von 4,5,6,7-Tetrahydroindazolen

Also Published As

Publication number Publication date
NL179729C (nl) 1986-11-03
IN139264B (de) 1976-05-29
FR2181773B1 (de) 1975-12-26
IT1052111B (it) 1981-06-20
FR2181773A1 (de) 1973-12-07
DE2310031A1 (de) 1973-09-20
CA994347A (en) 1976-08-03
US3895026A (en) 1975-07-15
NL179729B (nl) 1986-06-02
GB1381422A (en) 1975-01-22
DE2310031B2 (de) 1979-11-15
DE2310031C3 (de) 1980-07-31
HU165172B (de) 1974-07-27

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Legal Events

Date Code Title Description
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
A85 Still pending on 85-01-01
V4 Discontinued because of reaching the maximum lifetime of a patent