NL189297B - PROCESS FOR PREPARING A PHARMACEUTICAL PREPARATION WITH ANTIBIOTIC ACTION AND PROCESS FOR PREPARING A THIENAMYCIN DERIVATIVE. - Google Patents
PROCESS FOR PREPARING A PHARMACEUTICAL PREPARATION WITH ANTIBIOTIC ACTION AND PROCESS FOR PREPARING A THIENAMYCIN DERIVATIVE.Info
- Publication number
- NL189297B NL189297B NLAANVRAGE7612939,A NL7612939A NL189297B NL 189297 B NL189297 B NL 189297B NL 7612939 A NL7612939 A NL 7612939A NL 189297 B NL189297 B NL 189297B
- Authority
- NL
- Netherlands
- Prior art keywords
- preparing
- pharmaceutical preparation
- antibiotic action
- thienamycin derivative
- thienamycin
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title 2
- WKDDRNSBRWANNC-ATRFCDNQSA-N Thienamycin Chemical class C1C(SCCN)=C(C(O)=O)N2C(=O)[C@H]([C@H](O)C)[C@H]21 WKDDRNSBRWANNC-ATRFCDNQSA-N 0.000 title 1
- 230000003115 biocidal effect Effects 0.000 title 1
- 239000000825 pharmaceutical preparation Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
- C07D477/10—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D477/12—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
- C07D477/16—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hetero atoms or carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 3
- C07D477/20—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/10—Compounds having one or more C—Si linkages containing nitrogen having a Si-N linkage
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US63429675A | 1975-11-21 | 1975-11-21 | |
US67626176A | 1976-04-12 | 1976-04-12 | |
US73365476A | 1976-10-18 | 1976-10-18 |
Publications (3)
Publication Number | Publication Date |
---|---|
NL7612939A NL7612939A (en) | 1977-05-24 |
NL189297B true NL189297B (en) | 1992-10-01 |
NL189297C NL189297C (en) | 1993-03-01 |
Family
ID=27417545
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NLAANVRAGE7612939,A NL189297C (en) | 1975-11-21 | 1976-11-19 | PROCESS FOR PREPARING A PHARMACEUTICAL PREPARATION WITH ANTIBIOTIC ACTION AND PROCESS FOR PREPARING A THIENAMYCIN DERIVATIVE. |
Country Status (27)
Country | Link |
---|---|
AT (1) | AT358168B (en) |
AU (1) | AU512383B2 (en) |
BG (1) | BG34037A3 (en) |
CA (1) | CA1083577A (en) |
CH (2) | CH632510A5 (en) |
DD (1) | DD127742A5 (en) |
DE (1) | DE2652679A1 (en) |
DK (1) | DK157401C (en) |
EG (1) | EG12261A (en) |
ES (1) | ES453501A1 (en) |
FI (1) | FI62306C (en) |
FR (1) | FR2332012A1 (en) |
GB (1) | GB1570990A (en) |
GR (1) | GR62072B (en) |
HK (1) | HK29683A (en) |
HU (1) | HU180865B (en) |
IE (1) | IE44433B1 (en) |
IL (1) | IL50911A (en) |
KE (1) | KE3286A (en) |
NL (1) | NL189297C (en) |
NO (1) | NO153298C (en) |
NZ (1) | NZ182630A (en) |
PH (1) | PH16714A (en) |
PL (1) | PL110937B1 (en) |
PT (1) | PT65865B (en) |
SE (1) | SE427841B (en) |
SG (1) | SG10983G (en) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1593524A (en) * | 1976-11-19 | 1981-07-15 | Merck & Co Inc | 1-carba-2-penem-3-carboxylic acids |
SE436569B (en) * | 1977-05-05 | 1985-01-07 | Merck & Co Inc | ANALOGY PROCEDURE FOR THE PREPARATION OF TIENAMYCIN DERIVATIVES |
US4232030A (en) * | 1977-09-15 | 1980-11-04 | Merck & Co., Inc. | Substituted N-methylene derivatives of thienamycin sulfoxide and sulfone |
DK153486C (en) * | 1978-07-03 | 1988-11-28 | Merck & Co Inc | ANALOGY PROCEDURE FOR THE PREPARATION OF CRYSTALLINIC N-FORMIMIDOYL-THIENAMYCINE MONOHYDRATE |
EP0044170A1 (en) * | 1980-07-11 | 1982-01-20 | Beecham Group Plc | Beta-lactam antibiotics, their preparation and use |
WO1992004054A1 (en) * | 1990-08-30 | 1992-03-19 | STATE OF OREGON, acting by and through THE OREGON STATE BOARD OF HIGHER EDUCATION, acting for and on behalf of THE OREGON HEALTH SCIENCES UNIVERSITY, PORTLAND, OREGON, and THE UNIVERSITY OF OREGON, EUGENE, OREGON, Johnson Hall, University of Oregon | Substituted amidines having high binding to the sigma receptor and the use thereof |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1004670A (en) * | 1963-04-23 | 1965-09-15 | Beecham Res Lab | Penicillins |
GB1348984A (en) * | 1970-06-16 | 1974-03-27 | Merck & Co Inc | Antibiotics and processes for their production |
US3950357A (en) * | 1974-11-25 | 1976-04-13 | Merck & Co., Inc. | Antibiotics |
-
1976
- 1976-11-15 AU AU19647/76A patent/AU512383B2/en not_active Expired
- 1976-11-15 NZ NZ182630A patent/NZ182630A/en unknown
- 1976-11-15 IL IL50911A patent/IL50911A/en unknown
- 1976-11-18 FI FI763308A patent/FI62306C/en not_active IP Right Cessation
- 1976-11-18 IE IE2542/76A patent/IE44433B1/en not_active IP Right Cessation
- 1976-11-18 PH PH19142A patent/PH16714A/en unknown
- 1976-11-19 CH CH1462376A patent/CH632510A5/en not_active IP Right Cessation
- 1976-11-19 SE SE7612963A patent/SE427841B/en not_active IP Right Cessation
- 1976-11-19 CA CA266,186A patent/CA1083577A/en not_active Expired
- 1976-11-19 DD DD7600195868A patent/DD127742A5/en unknown
- 1976-11-19 NO NO763958A patent/NO153298C/en unknown
- 1976-11-19 GB GB48240/76A patent/GB1570990A/en not_active Expired
- 1976-11-19 BG BG7634723A patent/BG34037A3/en unknown
- 1976-11-19 HU HU76ME2032A patent/HU180865B/en unknown
- 1976-11-19 DK DK523576A patent/DK157401C/en not_active IP Right Cessation
- 1976-11-19 NL NLAANVRAGE7612939,A patent/NL189297C/en not_active IP Right Cessation
- 1976-11-19 AT AT863476A patent/AT358168B/en active Protection Beyond IP Right Term
- 1976-11-19 DE DE19762652679 patent/DE2652679A1/en active Granted
- 1976-11-19 ES ES453501A patent/ES453501A1/en not_active Expired
- 1976-11-19 PT PT65865A patent/PT65865B/en unknown
- 1976-11-19 FR FR7634882A patent/FR2332012A1/en active Granted
- 1976-11-20 PL PL1976193809A patent/PL110937B1/en not_active IP Right Cessation
- 1976-11-20 GR GR52223A patent/GR62072B/en unknown
- 1976-11-21 EG EG76723A patent/EG12261A/en active
-
1980
- 1980-09-26 CH CH725580A patent/CH633800A5/en not_active IP Right Cessation
-
1983
- 1983-03-14 SG SG109/83A patent/SG10983G/en unknown
- 1983-04-08 KE KE3286A patent/KE3286A/en unknown
- 1983-08-18 HK HK296/83A patent/HK29683A/en unknown
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Legal Events
Date | Code | Title | Description |
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BA | A request for search or an international-type search has been filed | ||
BB | A search report has been drawn up | ||
BC | A request for examination has been filed | ||
A85 | Still pending on 85-01-01 | ||
V4 | Discontinued because of reaching the maximum lifetime of a patent |
Free format text: 961119 |