MXPA06010916A - Novedoso metodo de proteccion neurologica mediante inhibicion farmacologica de proteina quinasa activada por amp. - Google Patents
Novedoso metodo de proteccion neurologica mediante inhibicion farmacologica de proteina quinasa activada por amp.Info
- Publication number
- MXPA06010916A MXPA06010916A MXPA06010916A MXPA06010916A MXPA06010916A MX PA06010916 A MXPA06010916 A MX PA06010916A MX PA06010916 A MXPA06010916 A MX PA06010916A MX PA06010916 A MXPA06010916 A MX PA06010916A MX PA06010916 A MXPA06010916 A MX PA06010916A
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- Prior art keywords
- ampk
- ischemic
- pampk
- compound
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
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- A61K31/365—Lactones
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K39/00—Medicinal preparations containing antigens or antibodies
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Toxicology (AREA)
- Molecular Biology (AREA)
- Immunology (AREA)
- Microbiology (AREA)
- Mycology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US55600004P | 2004-03-24 | 2004-03-24 | |
| PCT/US2005/009797 WO2005092068A2 (en) | 2004-03-24 | 2005-03-23 | Novel method of neuroprotection by pharmacological inhibition of amp-activated protein kinase |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA06010916A true MXPA06010916A (es) | 2007-07-25 |
Family
ID=35056772
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA06010916A MXPA06010916A (es) | 2004-03-24 | 2005-03-23 | Novedoso metodo de proteccion neurologica mediante inhibicion farmacologica de proteina quinasa activada por amp. |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US8293791B2 (https=) |
| EP (1) | EP1734973A4 (https=) |
| JP (1) | JP2008504228A (https=) |
| KR (2) | KR20070085093A (https=) |
| CN (1) | CN101132802A (https=) |
| AU (1) | AU2005226731A1 (https=) |
| BR (1) | BRPI0509085A (https=) |
| CA (1) | CA2560843A1 (https=) |
| IL (1) | IL178242A0 (https=) |
| MX (1) | MXPA06010916A (https=) |
| WO (1) | WO2005092068A2 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0509085A (pt) | 2004-03-24 | 2007-08-21 | Fasgen Llc | processo de neuroproteção através da inibição farmacológica da proteìna quinase ativada por amp |
| KR101152607B1 (ko) | 2005-12-20 | 2012-06-05 | 에스케이케미칼주식회사 | ６-[４-(２-피페리딘-1-일-에톡시)-페닐]-３-피리딘-４-일-피라졸로[１,５-ａ]피리미딘의 제조방법 |
| US7741350B1 (en) * | 2009-01-28 | 2010-06-22 | Cara Therapeutics, Inc. | Bicyclic pyrazolo-heterocycles |
| WO2010088050A2 (en) | 2009-01-28 | 2010-08-05 | Cara Therapeutics, Inc. | Bicyclic pyrazolo-heterocycles |
| HK1221119A1 (zh) | 2013-03-28 | 2017-05-26 | The Trustees Of Columbia University In The City Of New York | 用omega-3甘油酯再灌注促进对用於移植的供体器官的保护 |
| KR101532211B1 (ko) * | 2014-04-30 | 2015-06-30 | 세종대학교산학협력단 | Ampk 억제기능에 기반한 뇌졸중 치료용 약학적 조성물 및 방법 |
| CN119868551B (zh) * | 2024-11-28 | 2026-04-14 | 四川大学华西医院 | F-box蛋白48的抑制剂的新用途和治疗缺血性脑血管病的药物 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9602080D0 (en) * | 1996-02-02 | 1996-04-03 | Pfizer Ltd | Pharmaceutical compounds |
| US5981575A (en) * | 1996-11-15 | 1999-11-09 | Johns Hopkins University, The | Inhibition of fatty acid synthase as a means to reduce adipocyte mass |
| CO5180581A1 (es) | 1999-09-30 | 2002-07-30 | Pfizer Prod Inc | Compuestos para el tratamiento de la isquemia ciones farmaceuticas que los contienen para el tratamiento de la isquemia |
| US6423705B1 (en) * | 2001-01-25 | 2002-07-23 | Pfizer Inc. | Combination therapy |
| IL147696A0 (en) * | 2001-01-25 | 2002-08-14 | Pfizer Prod Inc | Combination therapy |
| BRPI0509085A (pt) | 2004-03-24 | 2007-08-21 | Fasgen Llc | processo de neuroproteção através da inibição farmacológica da proteìna quinase ativada por amp |
-
2005
- 2005-03-23 BR BRPI0509085-7A patent/BRPI0509085A/pt not_active IP Right Cessation
- 2005-03-23 AU AU2005226731A patent/AU2005226731A1/en not_active Abandoned
- 2005-03-23 US US10/593,710 patent/US8293791B2/en not_active Expired - Fee Related
- 2005-03-23 WO PCT/US2005/009797 patent/WO2005092068A2/en not_active Ceased
- 2005-03-23 CN CNA2005800127675A patent/CN101132802A/zh active Pending
- 2005-03-23 MX MXPA06010916A patent/MXPA06010916A/es not_active Application Discontinuation
- 2005-03-23 KR KR1020067022076A patent/KR20070085093A/ko not_active Ceased
- 2005-03-23 KR KR1020127016911A patent/KR101283416B1/ko not_active Expired - Fee Related
- 2005-03-23 EP EP05732234A patent/EP1734973A4/en not_active Withdrawn
- 2005-03-23 JP JP2007505165A patent/JP2008504228A/ja active Pending
- 2005-03-23 CA CA002560843A patent/CA2560843A1/en not_active Abandoned
-
2006
- 2006-09-21 IL IL178242A patent/IL178242A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR101283416B1 (ko) | 2013-07-08 |
| KR20120078756A (ko) | 2012-07-10 |
| US8293791B2 (en) | 2012-10-23 |
| IL178242A0 (en) | 2007-03-08 |
| EP1734973A2 (en) | 2006-12-27 |
| US20090137665A1 (en) | 2009-05-28 |
| WO2005092068A2 (en) | 2005-10-06 |
| KR20070085093A (ko) | 2007-08-27 |
| AU2005226731A1 (en) | 2005-10-06 |
| EP1734973A4 (en) | 2010-08-04 |
| WO2005092068A3 (en) | 2007-09-20 |
| BRPI0509085A (pt) | 2007-08-21 |
| CN101132802A (zh) | 2008-02-27 |
| JP2008504228A (ja) | 2008-02-14 |
| CA2560843A1 (en) | 2005-10-06 |
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