MXPA04003346A - Formulacion de dosis oral de disolucion instantanea. - Google Patents

Formulacion de dosis oral de disolucion instantanea.

Info

Publication number
MXPA04003346A
MXPA04003346A MXPA04003346A MXPA04003346A MXPA04003346A MX PA04003346 A MXPA04003346 A MX PA04003346A MX PA04003346 A MXPA04003346 A MX PA04003346A MX PA04003346 A MXPA04003346 A MX PA04003346A MX PA04003346 A MXPA04003346 A MX PA04003346A
Authority
MX
Mexico
Prior art keywords
granules
sodium
oral dosage
dosage forms
dosage formulation
Prior art date
Application number
MXPA04003346A
Other languages
English (en)
Inventor
Desai Divyakant
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Priority claimed from PCT/US2001/031530 external-priority patent/WO2003030868A1/en
Publication of MXPA04003346A publication Critical patent/MXPA04003346A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Zoology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Seasonings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se proporcionan granulos para la produccion de formas de dosis orales farmaceuticas de disolucion instantanea mejoradas. Ademas de uno o mas medicamentos, los granulos estan compuestos de una combinacion de excipientes que consiste en un superdesintegrante (de dos o mas agentes seleccionados del grupo que consiste en crospovidona, croscarmelosa de sodio, glicolato de almidon de sodio, hidroxipropilcelulosa de baja sustitucion o almidon pregelatinizado), un agente dispersante, un agente de distribucion y un aglutinante, y tambien puede incluir otros ingredientes convencionales tales como los agentes edulcorantes y saborizantes. Los presentes granulos son adecuados porque son estables y pueden prepararse sin la ayuda de solventes y sin la necesidad de ambientes o manejo especiales. Las formas de dosis, especialmente tabletas, preparadas de los mismos en equipo convencional se desintegran en la boca en menos de aproximadamente cinco segundos.
MXPA04003346A 2001-10-09 2001-10-09 Formulacion de dosis oral de disolucion instantanea. MXPA04003346A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2001/031530 WO2003030868A1 (en) 2001-10-09 2001-10-09 Flashmelt oral dosage formulation

Publications (1)

Publication Number Publication Date
MXPA04003346A true MXPA04003346A (es) 2004-09-28

Family

ID=32505152

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA04003346A MXPA04003346A (es) 2001-10-09 2001-10-09 Formulacion de dosis oral de disolucion instantanea.

Country Status (13)

Country Link
EP (1) EP1441698B1 (es)
JP (1) JP2005507397A (es)
KR (1) KR20040045499A (es)
CN (1) CN100490810C (es)
BR (1) BR0117147A (es)
CA (1) CA2462886C (es)
HR (1) HRP20040322A2 (es)
HU (1) HUP0500638A3 (es)
IL (1) IL161143A0 (es)
IS (1) IS7208A (es)
MX (1) MXPA04003346A (es)
NO (1) NO340570B1 (es)
RS (1) RS55392B1 (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5279487B2 (ja) * 2005-05-18 2013-09-04 エムペックス・ファーマシューティカルズ・インコーポレーテッド エアロゾル化フルオロキノロンおよびその使用
KR100780553B1 (ko) * 2005-08-18 2007-11-29 한올제약주식회사 메트포르민 서방정 및 그의 제조방법
CN101322709B (zh) * 2007-06-12 2011-03-02 成都康弘药业集团股份有限公司 一种含有阿立哌唑的药物组合物及其制备方法
WO2010106936A1 (ja) * 2009-03-16 2010-09-23 ニプロ株式会社 口腔内崩壊錠
WO2011049122A1 (ja) * 2009-10-21 2011-04-28 第一三共株式会社 プラバスタチンナトリウム口腔内速崩壊錠及びその製造方法
HU1000278D0 (en) * 2010-05-28 2010-07-28 Egis Gyogyszergyar Nyilvanosan Novel pharmaceutical use uf silicic acid
CN102397552B (zh) * 2010-09-10 2016-06-08 广州自远生物科技有限公司 一种含喹诺酮类的药物复合制剂及其制备方法和应用
JP2012121850A (ja) * 2010-12-09 2012-06-28 Otsuka Pharmaceut Co Ltd アリピプラゾールの経口速溶性組成物
CN102357086A (zh) * 2011-11-01 2012-02-22 上海理工大学 一种头孢丙烯口腔崩解片
KR101285008B1 (ko) * 2012-04-18 2013-07-10 제일약품주식회사 저용량 엔테카비어의 경구투여 제제의 제조방법
CN102670533B (zh) * 2012-05-17 2017-06-16 浙江华海药业股份有限公司 稳定的阿立哌唑口腔崩解片及其制备方法
CN104138382B (zh) * 2014-08-14 2015-08-12 广州一品红制药有限公司 一种含盐酸左氧氟沙星的组合物
JP6558530B2 (ja) * 2015-04-20 2019-08-14 高田製薬株式会社 アリピプラゾール医薬品製剤
JP2015172084A (ja) * 2015-07-06 2015-10-01 大塚製薬株式会社 アリピプラゾールの経口速溶性組成物
CN106913548A (zh) * 2015-12-28 2017-07-04 药源药物化学(上海)有限公司 一种阿立哌唑口崩片及其制备方法
JP6572257B2 (ja) * 2017-05-16 2019-09-04 大塚製薬株式会社 アリピプラゾールの経口速溶性組成物
KR101808513B1 (ko) 2017-06-22 2018-01-18 임철수 한대의본체로 다수가 사용하는 컴퓨터장치 및 그 운영방법

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5994348A (en) * 1995-06-07 1999-11-30 Sanofi Pharmaceutical compositions containing irbesartan
EP0918456A1 (en) * 1996-07-23 1999-06-02 Fmc Corporation Disintegrant composition for dispersible solids
CA2311734C (en) * 2000-04-12 2011-03-08 Bristol-Myers Squibb Company Flash-melt oral dosage formulation

Also Published As

Publication number Publication date
CN100490810C (zh) 2009-05-27
NO20041383L (no) 2004-06-01
KR20040045499A (ko) 2004-06-01
RS55392B1 (sr) 2017-03-31
BR0117147A (pt) 2006-05-09
HUP0500638A3 (en) 2008-04-28
IL161143A0 (en) 2004-08-31
EP1441698A1 (en) 2004-08-04
CA2462886A1 (en) 2003-04-17
NO340570B1 (no) 2017-05-15
CN1561200A (zh) 2005-01-05
HUP0500638A2 (en) 2007-02-28
HRP20040322A2 (en) 2004-12-31
EP1441698A4 (en) 2008-08-13
IS7208A (is) 2004-04-06
CA2462886C (en) 2013-07-30
EP1441698B1 (en) 2018-05-02
JP2005507397A (ja) 2005-03-17

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