MXPA02001473A - Azaindoles que tienen afinidad con el receptor de serotonina. - Google Patents
Azaindoles que tienen afinidad con el receptor de serotonina.Info
- Publication number
- MXPA02001473A MXPA02001473A MXPA02001473A MXPA02001473A MXPA02001473A MX PA02001473 A MXPA02001473 A MX PA02001473A MX PA02001473 A MXPA02001473 A MX PA02001473A MX PA02001473 A MXPA02001473 A MX PA02001473A MX PA02001473 A MXPA02001473 A MX PA02001473A
- Authority
- MX
- Mexico
- Prior art keywords
- group
- formula
- azaindoles
- double bond
- serotonin receptor
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US14834399P | 1999-08-12 | 1999-08-12 | |
PCT/IB2000/001122 WO2001012629A1 (en) | 1999-08-12 | 2000-08-14 | Azaindoles having serotonin receptor affinity |
Publications (1)
Publication Number | Publication Date |
---|---|
MXPA02001473A true MXPA02001473A (es) | 2003-07-21 |
Family
ID=22525363
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MXPA02001473A MXPA02001473A (es) | 1999-08-12 | 2000-08-14 | Azaindoles que tienen afinidad con el receptor de serotonina. |
Country Status (10)
Country | Link |
---|---|
EP (1) | EP1204662B1 (es) |
JP (1) | JP4969004B2 (es) |
AT (1) | ATE268330T1 (es) |
AU (1) | AU779832B2 (es) |
CA (1) | CA2382247C (es) |
DE (1) | DE60011269T2 (es) |
DK (1) | DK1204662T3 (es) |
ES (1) | ES2222219T3 (es) |
MX (1) | MXPA02001473A (es) |
WO (1) | WO2001012629A1 (es) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10030037A1 (de) | 2000-06-17 | 2001-12-20 | Mann & Hummel Filter | Zylindrische Filterpatrone mit Stützrohr |
ITRM20010356A1 (it) | 2001-06-21 | 2002-12-23 | Sigma Tau Ind Farmaceuti | "5-alogeno derivati della triptamina utili come ligandi del recettore5-ht6 e/o 5-ht7 della serotonina. |
CA2470863C (en) * | 2001-12-20 | 2012-05-15 | Wyeth | Indolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands |
TW200301251A (en) | 2001-12-20 | 2003-07-01 | Wyeth Corp | Azaindolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands |
GB0202679D0 (en) * | 2002-02-05 | 2002-03-20 | Glaxo Group Ltd | Novel compounds |
AU2003226724A1 (en) * | 2002-03-27 | 2003-10-08 | Glaxo Group Limited | Quinoline and aza-indole derivatives and their use as 5-ht6 ligands |
UA78999C2 (en) * | 2002-06-04 | 2007-05-10 | Wyeth Corp | 1-(aminoalkyl)-3-sulfonylazaindoles as ligands of 5-hydroxytryptamine-6 |
EP1897876A3 (en) | 2002-06-20 | 2009-03-18 | Biovitrum AB (publ) | Compounds useful for the treatment of obesity, type II diabetes and CNS disorders |
TW200403243A (en) | 2002-07-18 | 2004-03-01 | Wyeth Corp | 1-Heterocyclylalkyl-3-sulfonylazaindole or-azaindazole derivatives as 5-hydroxytryptamine-6 ligands |
EP1592772A2 (en) * | 2003-01-31 | 2005-11-09 | Pfizer Products Incorporated | 5ht7 antagonists and inverse agonists |
BRPI0407493A (pt) * | 2003-02-14 | 2006-02-14 | Wyeth Corp | derivados heterociclil-3-sulfinilazaindol ou -azaindazol como ligantes de 5-hidroxitriptamina-6 |
BRPI0412809A (pt) * | 2003-07-23 | 2006-09-26 | Wyeth Corp | compostos de sulfonildihidrobenzimidazolona como ligantes a 5-hidróxitriptamina-6 |
ES2222828B1 (es) | 2003-07-30 | 2006-04-16 | Laboratorios Del Dr. Esteve, S.A. | Derivados de 1-sulfonilindoles, su preparacion y su aplicacion como medicamentos. |
US7696229B2 (en) | 2006-02-17 | 2010-04-13 | Memory Pharmaceuticals Corporation | Compounds having 5-HT6 receptor affinity |
ES2398299T3 (es) * | 2006-07-03 | 2013-03-15 | Proximagen Ltd. | Indoles como moduladores de 5-HT6 |
JP2014515368A (ja) * | 2011-05-26 | 2014-06-30 | 第一三共株式会社 | プロテインキナーゼ阻害剤としての複素環化合物 |
JP6454346B2 (ja) | 2013-12-20 | 2019-01-16 | サンシャイン・レイク・ファーマ・カンパニー・リミテッドSunshine Lake Pharma Co.,Ltd. | 芳香族複素環式化合物及び医薬におけるその応用 |
CA2953004C (en) | 2014-07-08 | 2023-02-21 | Sunshine Lake Pharma Co., Ltd. | Aromatic heterocyclic derivatives and pharmaceutical applications thereof |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PL310443A1 (en) * | 1993-03-01 | 1995-12-11 | Merck Sharp & Dohme | Derivatives of pyrolo-pyridine |
US5846982A (en) * | 1996-06-14 | 1998-12-08 | Eli Lilly And Company | Inhibition of serotonin reuptake |
EP0875513A1 (en) * | 1997-04-14 | 1998-11-04 | Eli Lilly And Company | Substituted heteroaromatic 5-HT 1F agonists |
US5905084A (en) * | 1997-11-14 | 1999-05-18 | Eli Lilly And Company | 5-HTIF -agonists effective in treating migraine |
US6562809B1 (en) * | 1998-09-18 | 2003-05-13 | Nps Allelix Corp. | 3-bicycloindole compounds |
-
2000
- 2000-08-14 WO PCT/IB2000/001122 patent/WO2001012629A1/en active IP Right Grant
- 2000-08-14 MX MXPA02001473A patent/MXPA02001473A/es active IP Right Grant
- 2000-08-14 ES ES00949846T patent/ES2222219T3/es not_active Expired - Lifetime
- 2000-08-14 AU AU63103/00A patent/AU779832B2/en not_active Ceased
- 2000-08-14 DE DE60011269T patent/DE60011269T2/de not_active Expired - Lifetime
- 2000-08-14 AT AT00949846T patent/ATE268330T1/de active
- 2000-08-14 CA CA2382247A patent/CA2382247C/en not_active Expired - Fee Related
- 2000-08-14 JP JP2001517527A patent/JP4969004B2/ja not_active Expired - Fee Related
- 2000-08-14 DK DK00949846T patent/DK1204662T3/da active
- 2000-08-14 EP EP00949846A patent/EP1204662B1/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
JP2003507380A (ja) | 2003-02-25 |
AU779832B2 (en) | 2005-02-10 |
ATE268330T1 (de) | 2004-06-15 |
DE60011269T2 (de) | 2005-06-23 |
DK1204662T3 (da) | 2004-10-04 |
DE60011269D1 (de) | 2004-07-08 |
WO2001012629A1 (en) | 2001-02-22 |
EP1204662B1 (en) | 2004-06-02 |
CA2382247A1 (en) | 2001-02-22 |
JP4969004B2 (ja) | 2012-07-04 |
ES2222219T3 (es) | 2005-02-01 |
EP1204662A1 (en) | 2002-05-15 |
AU6310300A (en) | 2001-03-13 |
CA2382247C (en) | 2010-09-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant or registration | ||
GB | Transfer or rights | ||
HC | Change of company name or juridical status |