MX9803556A - Derivados de aminoacidos, medicamentos que contienen tales compuestos y metodos para producirlos. - Google Patents

Derivados de aminoacidos, medicamentos que contienen tales compuestos y metodos para producirlos.

Info

Publication number
MX9803556A
MX9803556A MX9803556A MX9803556A MX9803556A MX 9803556 A MX9803556 A MX 9803556A MX 9803556 A MX9803556 A MX 9803556A MX 9803556 A MX9803556 A MX 9803556A MX 9803556 A MX9803556 A MX 9803556A
Authority
MX
Mexico
Prior art keywords
compounds
producing
amino acid
methods
acid derivatives
Prior art date
Application number
MX9803556A
Other languages
English (en)
Other versions
MXPA98003556A (es
Inventor
Wolfhard Engel
Wolfgang Eberlein
Klaus Rudolf
Henri Doods
Heike-Andrea Wieland
Klaus-Dieter Willim
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of MX9803556A publication Critical patent/MX9803556A/es
Publication of MXPA98003556A publication Critical patent/MXPA98003556A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/18—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to carbon atoms of six-membered aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/20—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylguanidines
    • C07C279/24—Y being a hetero atom
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
    • G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
    • G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
    • G01N33/58—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving labelled substances
    • G01N33/60—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving labelled substances involving radioactive labelled substances
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
    • G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
    • G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
    • G01N33/68—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving proteins, peptides or amino acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

Abstract

La invencion se relaciona con derivados de aminoácidos nuevos de formula general (Ver Formula) en la que R, U, V, Y, n, m y R1 a R3 se definen de conformidad con la reivindicacion 1, sus tautomeros, diastereomeros, enantiomeros, mezclas de los mismos y sales de los mismos, particularmente las sales Fisiologicamente aceptables de los mismos con ácidos o bases inorgánicas u orgánicas, los cuales tienen propiedades farmacologicas valiosas, particularmente propiedades antagonistas selectivas de NPY, composiciones farmacéuticas que contienen estos compuestos, el uso de los mismos y procesos para prepararlos.
MXPA/A/1998/003556A 1995-11-30 1998-05-06 Derivados de aminoacidos, medicamentos que contienen tales compuestos y metodos para producirlos MXPA98003556A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19544685.2 1995-11-30
DE19544685A DE19544685A1 (de) 1995-11-30 1995-11-30 Aminosäurederivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung

Publications (2)

Publication Number Publication Date
MX9803556A true MX9803556A (es) 1998-09-30
MXPA98003556A MXPA98003556A (es) 1998-11-16

Family

ID=

Also Published As

Publication number Publication date
DE19544685A1 (de) 1997-06-05
US5962530A (en) 1999-10-05
JP2000501090A (ja) 2000-02-02
CA2235937A1 (en) 1997-06-05
EP0865425A1 (de) 1998-09-23
WO1997019913A1 (de) 1997-06-05

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