MX9704079A - Liberacion de farmacos antiinflamatorios no esteroides empleando uan goam hidrocoloide en polvo que se obtiene de plantas superiores. - Google Patents

Liberacion de farmacos antiinflamatorios no esteroides empleando uan goam hidrocoloide en polvo que se obtiene de plantas superiores.

Info

Publication number
MX9704079A
MX9704079A MX9704079A MX9704079A MX9704079A MX 9704079 A MX9704079 A MX 9704079A MX 9704079 A MX9704079 A MX 9704079A MX 9704079 A MX9704079 A MX 9704079A MX 9704079 A MX9704079 A MX 9704079A
Authority
MX
Mexico
Prior art keywords
nsaid
composition
higher plants
hydrocolloid gum
gum obtainable
Prior art date
Application number
MX9704079A
Other languages
English (en)
Inventor
Eric H Kuhrts
David R Friend
Karen Yu
Jagdish Parasrampuria
Original Assignee
Cibus Pharmaceutical Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cibus Pharmaceutical Inc filed Critical Cibus Pharmaceutical Inc
Publication of MX9704079A publication Critical patent/MX9704079A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/60Salicylic acid; Derivatives thereof
    • A61K31/612Salicylic acid; Derivatives thereof having the hydroxy group in position 2 esterified, e.g. salicylsulfuric acid
    • A61K31/616Salicylic acid; Derivatives thereof having the hydroxy group in position 2 esterified, e.g. salicylsulfuric acid by carboxylic acids, e.g. acetylsalicylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Medicines Containing Plant Substances (AREA)

Abstract

Una composicion farmacéutica de suministracion oral para reducir el efecto de irritacion gástrica de un AINE en el tracto GI superior de un mamífero. La composicion incluye (a) una cantidad protectora de la mucosa de una goma hidrocoloide farmacéuticamente aceptable obtenible a partir de plantas superiores, (b) una cantidad mejoradora de dispersion de otro excipiente y (c) una cantidad terapéuticamente efectiva de un ATNE. Se describe también un procedimiento para preparar la composicion y un método para reducir el efecto de irritacion gástrica del AINE al administrar la composicion. Asimismo, se describe una composicion particularmente util para preparar una suspension acuosa.
MX9704079A 1994-12-01 1995-11-30 Liberacion de farmacos antiinflamatorios no esteroides empleando uan goam hidrocoloide en polvo que se obtiene de plantas superiores. MX9704079A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US34760194A 1994-12-01 1994-12-01
PCT/US1995/015599 WO1996016639A1 (en) 1994-12-01 1995-11-30 Nsaid delivery employing a powdered hydrocolloid gum obtainable from higher plants

Publications (1)

Publication Number Publication Date
MX9704079A true MX9704079A (es) 1997-12-31

Family

ID=23364417

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9704079A MX9704079A (es) 1994-12-01 1995-11-30 Liberacion de farmacos antiinflamatorios no esteroides empleando uan goam hidrocoloide en polvo que se obtiene de plantas superiores.

Country Status (8)

Country Link
EP (1) EP0804169A4 (es)
JP (1) JPH10509982A (es)
AU (1) AU690417B2 (es)
CA (1) CA2205442C (es)
FI (1) FI972305A0 (es)
MX (1) MX9704079A (es)
NO (1) NO972485L (es)
WO (1) WO1996016639A1 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5811388A (en) * 1995-06-07 1998-09-22 Cibus Pharmaceutical, Inc. Delivery of drugs to the lower GI tract
IL123505A (en) * 1996-07-08 2004-12-15 Penwest Pharmaceuticals Compan Sustained release matrix for high-dose insoluble drugs
US5955107A (en) * 1997-12-12 1999-09-21 Fmc Corporation Pharmaceutical suspension tablet compositions
US6106862A (en) * 1998-08-13 2000-08-22 Andrx Corporation Once daily analgesic tablet
RS50104B (sr) * 1998-08-21 2009-01-22 Novartis Ag., Nova oralna formulacija za 5-th4 agoniste ili antagoniste
SE0003125D0 (sv) * 2000-09-05 2000-09-05 Astrazeneca Ab Modified polymers

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1327938A (en) * 1969-12-17 1973-08-22 Sucrest Corp Composition for use in forming tablets
DE2130545A1 (de) * 1971-06-19 1972-12-21 Merck Patent Gmbh Pharmazeutischer Formkoerper
WO1986006627A1 (en) * 1985-05-15 1986-11-20 Riker Laboratories, Inc. Sustained release theophylline compositions and processes
US5096714A (en) * 1988-06-28 1992-03-17 Hauser-Kuhrts, Inc. Prolonged release drug tablet formulations
US5292534A (en) * 1992-03-25 1994-03-08 Valentine Enterprises, Inc. Sustained release composition and method utilizing xanthan gum and an active ingredient
CA2152795C (en) * 1992-12-30 1999-02-16 Victor Louis King Readily available konjac glucomannan sustained release excipient

Also Published As

Publication number Publication date
NO972485D0 (no) 1997-05-30
JPH10509982A (ja) 1998-09-29
EP0804169A4 (en) 1998-08-19
CA2205442A1 (en) 1996-06-06
FI972305A (fi) 1997-05-30
EP0804169A1 (en) 1997-11-05
FI972305A0 (fi) 1997-05-30
AU4595196A (en) 1996-06-19
WO1996016639A1 (en) 1996-06-06
AU690417B2 (en) 1998-04-23
CA2205442C (en) 2003-01-21
NO972485L (no) 1997-07-31

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