MX9704079A - Liberacion de farmacos antiinflamatorios no esteroides empleando uan goam hidrocoloide en polvo que se obtiene de plantas superiores. - Google Patents

Liberacion de farmacos antiinflamatorios no esteroides empleando uan goam hidrocoloide en polvo que se obtiene de plantas superiores.

Info

Publication number
MX9704079A
MX9704079A MX9704079A MX9704079A MX9704079A MX 9704079 A MX9704079 A MX 9704079A MX 9704079 A MX9704079 A MX 9704079A MX 9704079 A MX9704079 A MX 9704079A MX 9704079 A MX9704079 A MX 9704079A
Authority
MX
Mexico
Prior art keywords
composition
goam
hydrocoloid
uan
release
Prior art date
Application number
MX9704079A
Other languages
English (en)
Inventor
Eric H Kuhrts
David R Friend
Karen Yu
Jagdish Parasrampuria
Original Assignee
Cibus Pharmaceutical Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cibus Pharmaceutical Inc filed Critical Cibus Pharmaceutical Inc
Publication of MX9704079A publication Critical patent/MX9704079A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/60Salicylic acid; Derivatives thereof
    • A61K31/612Salicylic acid; Derivatives thereof having the hydroxy group in position 2 esterified, e.g. salicylsulfuric acid
    • A61K31/616Salicylic acid; Derivatives thereof having the hydroxy group in position 2 esterified, e.g. salicylsulfuric acid by carboxylic acids, e.g. acetylsalicylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)

Abstract

Una composicion farmacéutica de suministracion oral para reducir el efecto de irritacion gástrica de un AINE en el tracto GI superior de un mamífero. La composicion incluye (a) una cantidad protectora de la mucosa de una goma hidrocoloide farmacéuticamente aceptable obtenible a partir de plantas superiores, (b) una cantidad mejoradora de dispersion de otro excipiente y (c) una cantidad terapéuticamente efectiva de un ATNE. Se describe también un procedimiento para preparar la composicion y un método para reducir el efecto de irritacion gástrica del AINE al administrar la composicion. Asimismo, se describe una composicion particularmente util para preparar una suspension acuosa.
MX9704079A 1994-12-01 1995-11-30 Liberacion de farmacos antiinflamatorios no esteroides empleando uan goam hidrocoloide en polvo que se obtiene de plantas superiores. MX9704079A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US34760194A 1994-12-01 1994-12-01
PCT/US1995/015599 WO1996016639A1 (en) 1994-12-01 1995-11-30 Nsaid delivery employing a powdered hydrocolloid gum obtainable from higher plants

Publications (1)

Publication Number Publication Date
MX9704079A true MX9704079A (es) 1997-12-31

Family

ID=23364417

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9704079A MX9704079A (es) 1994-12-01 1995-11-30 Liberacion de farmacos antiinflamatorios no esteroides empleando uan goam hidrocoloide en polvo que se obtiene de plantas superiores.

Country Status (8)

Country Link
EP (1) EP0804169A4 (es)
JP (1) JPH10509982A (es)
AU (1) AU690417B2 (es)
CA (1) CA2205442C (es)
FI (1) FI972305A0 (es)
MX (1) MX9704079A (es)
NO (1) NO972485L (es)
WO (1) WO1996016639A1 (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5811388A (en) * 1995-06-07 1998-09-22 Cibus Pharmaceutical, Inc. Delivery of drugs to the lower GI tract
JP3148256B2 (ja) * 1996-07-08 2001-03-19 エドワード メンデル カンパニー.,インコーポレーテッド 高用量難溶性薬物用持続放出マトリックス
US5955107A (en) * 1997-12-12 1999-09-21 Fmc Corporation Pharmaceutical suspension tablet compositions
US6106862A (en) * 1998-08-13 2000-08-22 Andrx Corporation Once daily analgesic tablet
RU2260424C9 (ru) * 1998-08-21 2006-05-20 Новартис Аг Новая композиция для перорального введения
ES2257869T3 (es) * 1998-08-21 2006-08-01 Novartis Ag Nueva formulacion oral para agonistas o antagonistas de 5-ht4.
SE0003125D0 (sv) * 2000-09-05 2000-09-05 Astrazeneca Ab Modified polymers
CN114901267A (zh) * 2019-12-05 2022-08-12 旗舰创业创新五公司 酰化活性剂及其用于治疗代谢障碍和非酒精性脂肪肝病的方法
JP7782842B2 (ja) * 2022-06-02 2025-12-09 株式会社パウレック 速崩壊性圧縮成形物の製造方法および速崩壊性圧縮成形物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1327938A (en) * 1969-12-17 1973-08-22 Sucrest Corp Composition for use in forming tablets
DE2130545A1 (de) * 1971-06-19 1972-12-21 Merck Patent Gmbh Pharmazeutischer Formkoerper
EP0222883A1 (en) * 1985-05-15 1987-05-27 Riker Laboratories, Inc. Sustained release theophylline compositions and processes
US5096714A (en) * 1988-06-28 1992-03-17 Hauser-Kuhrts, Inc. Prolonged release drug tablet formulations
US5292534A (en) * 1992-03-25 1994-03-08 Valentine Enterprises, Inc. Sustained release composition and method utilizing xanthan gum and an active ingredient
EP0676967A4 (en) * 1992-12-30 1996-10-02 Fmc Corp RELEASED, EXTENDED, EASY TO PRODUCE EXCIPIENT, BASED ON KONJAC GLUCOMANNANE.

Also Published As

Publication number Publication date
NO972485D0 (no) 1997-05-30
CA2205442A1 (en) 1996-06-06
AU4595196A (en) 1996-06-19
FI972305A7 (fi) 1997-05-30
NO972485L (no) 1997-07-31
EP0804169A1 (en) 1997-11-05
FI972305L (fi) 1997-05-30
CA2205442C (en) 2003-01-21
WO1996016639A1 (en) 1996-06-06
FI972305A0 (fi) 1997-05-30
AU690417B2 (en) 1998-04-23
EP0804169A4 (en) 1998-08-19
JPH10509982A (ja) 1998-09-29

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