MX9304266A - Quinolinas y naftiridinas de 3-carboxaldehido sustituidas. - Google Patents

Quinolinas y naftiridinas de 3-carboxaldehido sustituidas.

Info

Publication number
MX9304266A
MX9304266A MX9304266A MX9304266A MX9304266A MX 9304266 A MX9304266 A MX 9304266A MX 9304266 A MX9304266 A MX 9304266A MX 9304266 A MX9304266 A MX 9304266A MX 9304266 A MX9304266 A MX 9304266A
Authority
MX
Mexico
Prior art keywords
naftiridines
carboxaldehido
quinolins
substituted
prodrugs
Prior art date
Application number
MX9304266A
Other languages
English (en)
Inventor
Martin R Jefson
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MX9304266A publication Critical patent/MX9304266A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Esta invención se refiere a profármacos de quinolina y naftiridina que tienen un grupo 3-carboxaldehído, a composiciones antibacterianas que contienen dichos profármacos y a un método para tratar infecciones bacterianas administrando dichos profármacos.
MX9304266A 1992-07-15 1993-07-14 Quinolinas y naftiridinas de 3-carboxaldehido sustituidas. MX9304266A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/914,188 US5235054A (en) 1992-07-15 1992-07-15 3-carboxaldehyde substituted quinolines and naphthyridines

Publications (1)

Publication Number Publication Date
MX9304266A true MX9304266A (es) 1994-01-31

Family

ID=25434020

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9304266A MX9304266A (es) 1992-07-15 1993-07-14 Quinolinas y naftiridinas de 3-carboxaldehido sustituidas.

Country Status (20)

Country Link
US (1) US5235054A (es)
EP (1) EP0650488A1 (es)
JP (1) JPH07504684A (es)
KR (1) KR950702561A (es)
CN (1) CN1083053A (es)
AU (1) AU669958B2 (es)
BR (1) BR9306733A (es)
CA (1) CA2140135A1 (es)
CZ (1) CZ280603B6 (es)
FI (1) FI933203A (es)
HU (1) HUT68745A (es)
IL (1) IL106264A0 (es)
MX (1) MX9304266A (es)
NO (1) NO950142L (es)
NZ (1) NZ252847A (es)
PL (1) PL307135A1 (es)
RU (1) RU2097379C1 (es)
SK (1) SK4695A3 (es)
WO (1) WO1994002480A1 (es)
ZA (1) ZA935076B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5378694A (en) * 1990-09-07 1995-01-03 Schering Corporation Acyl and alkoxy substituted quinolines
EP0868183B1 (en) * 1995-12-21 2002-01-30 Pfizer Inc. Injectable quinolone formulations
JO3077B1 (ar) * 2005-07-28 2017-03-15 Janssen Pharmaceutica Nv مشتقات كوينولين مضادة للبكتيريا
EP2429991B1 (en) 2009-05-15 2014-09-10 Redx Pharma Limited Redox drug derivatives
WO2020184578A1 (ja) * 2019-03-11 2020-09-17 小胞体ストレス研究所株式会社 新規なeIF2αのリン酸化促進剤

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2509728A1 (fr) * 1981-07-17 1983-01-21 Roussel Uclaf Nouveaux derives de la quinoleine, leurs sels, procede de preparation, application a titre de medicaments et compositions les renfermant
IN166416B (es) * 1985-09-18 1990-05-05 Pfizer
JP2777661B2 (ja) * 1988-10-20 1998-07-23 大塚製薬株式会社 ベンゾヘテロ環化合物

Also Published As

Publication number Publication date
PL307135A1 (en) 1995-05-02
KR950702561A (ko) 1995-07-29
HUT68745A (en) 1995-07-28
NZ252847A (en) 1996-07-26
WO1994002480A1 (en) 1994-02-03
FI933203A0 (fi) 1993-07-14
NO950142D0 (no) 1995-01-13
AU669958B2 (en) 1996-06-27
NO950142L (no) 1995-01-13
SK4695A3 (en) 1995-07-11
US5235054A (en) 1993-08-10
RU2097379C1 (ru) 1997-11-27
CZ10195A3 (en) 1995-09-13
CA2140135A1 (en) 1994-02-03
FI933203A (fi) 1994-01-16
HU9302018D0 (en) 1993-10-28
ZA935076B (en) 1995-01-16
IL106264A0 (en) 1993-11-15
EP0650488A1 (en) 1995-05-03
RU95105159A (ru) 1997-02-10
JPH07504684A (ja) 1995-05-25
CN1083053A (zh) 1994-03-02
BR9306733A (pt) 1999-01-12
AU5574694A (en) 1994-02-14
CZ280603B6 (cs) 1996-03-13

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Legal Events

Date Code Title Description
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