MX9206563A - Utilizacion de derivados de anfotericina b como inhibidores de proteasas. - Google Patents

Utilizacion de derivados de anfotericina b como inhibidores de proteasas.

Info

Publication number
MX9206563A
MX9206563A MX9206563A MX9206563A MX9206563A MX 9206563 A MX9206563 A MX 9206563A MX 9206563 A MX9206563 A MX 9206563A MX 9206563 A MX9206563 A MX 9206563A MX 9206563 A MX9206563 A MX 9206563A
Authority
MX
Mexico
Prior art keywords
amphotericin
derivatives
protease inhibitors
pathogens
multiplication
Prior art date
Application number
MX9206563A
Other languages
English (en)
Inventor
Michel Seman
Original Assignee
Mayoly Spindler Lab
Michel Seman
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mayoly Spindler Lab, Michel Seman filed Critical Mayoly Spindler Lab
Publication of MX9206563A publication Critical patent/MX9206563A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)

Abstract

Nueva utilización de la anfotericina b, o de un derivado de la misma, como inhibidor de proteasas. Aplicación para obtener medicamentos inhibidores de la multiplicación de agentes patógenos, en particular el VIH.
MX9206563A 1991-11-14 1992-11-13 Utilizacion de derivados de anfotericina b como inhibidores de proteasas. MX9206563A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9113999A FR2683723B1 (fr) 1991-11-14 1991-11-14 Nouveaux medicaments antiviraux actifs sur le virus vih.

Publications (1)

Publication Number Publication Date
MX9206563A true MX9206563A (es) 1993-11-01

Family

ID=9418894

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9206563A MX9206563A (es) 1991-11-14 1992-11-13 Utilizacion de derivados de anfotericina b como inhibidores de proteasas.

Country Status (10)

Country Link
US (1) US5514662A (es)
EP (1) EP0542630A3 (es)
JP (1) JPH06504295A (es)
KR (1) KR930702994A (es)
AU (1) AU669143B2 (es)
CA (1) CA2099490A1 (es)
FR (1) FR2683723B1 (es)
MX (1) MX9206563A (es)
TW (1) TW225991B (es)
WO (1) WO1993009791A2 (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1993018006A1 (en) 1992-03-11 1993-09-16 Narhex Limited Amine derivatives of oxo- and hydroxy-substitued hydrocarbons
US6071895A (en) 1992-03-11 2000-06-06 Narhex Limited Polar-substituted hydrocarbons
ATE253050T1 (de) 1992-03-11 2003-11-15 Narhex Ltd Aminderivate von oxo- und hydroxy- substituierten kohlenwasserstoffen
US5888992A (en) 1992-03-11 1999-03-30 Narhex Limited Polar substituted hydrocarbons
US6869925B1 (en) 1992-09-09 2005-03-22 Amgen Inc. Inhibition of retrovirus infection
IL110898A0 (en) * 1993-09-10 1994-11-28 Narhex Australia Pty Ltd Polar-substituted hydrocarbons
US6017880A (en) * 1994-03-09 2000-01-25 Amgen Inc. Inhibition of retrovirus infection
GB2290708A (en) * 1994-06-28 1996-01-10 Georgi Stankov Pharmaceutical uses of polyene macrolides
GB2290707A (en) * 1994-06-28 1996-01-10 Georgi Stankov Pharmaceutical uses of Amphotericin B
US6413537B1 (en) 2000-03-10 2002-07-02 Wisconsin Alumni Research Foundation Nystatin formulation having reduced toxicity
JP2003327536A (ja) * 2002-03-07 2003-11-19 Kitasato Inst:The ヒト免疫不全症候群ウイルスの感染、増殖抑制剤
US20060194814A1 (en) * 2003-06-02 2006-08-31 Vassilios Papadopoulos Benzamide compounds
WO2005112922A2 (en) * 2004-04-22 2005-12-01 Samaritan Pharmaceuticals Benzamide compounds
EP3156410A4 (en) 2014-06-12 2018-01-03 Shionogi & Co., Ltd. Polyene macrolide derivative

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8829592D0 (en) * 1988-12-19 1989-02-08 Beecham Group Plc Novel compounds
EP0350164A3 (en) * 1988-06-13 1991-07-24 Beecham Group Plc Amphotericin derivatives
GB8829593D0 (en) * 1988-12-19 1989-02-08 Beecham Group Plc Novel compounds
US5175172A (en) * 1988-12-19 1992-12-29 Francois Dietlin Method of alleviating AIDS symptoms and compositions therefor
FR2654339B1 (fr) * 1989-11-14 1994-10-28 Mayoly Spindler Laboratoires Nouveaux derives solubles et non toxiques des macrolides polyeniques basiques, leur preparation et leurs applications.
EP0431870A1 (en) * 1989-12-08 1991-06-12 Beecham Group p.l.c. Amphotericin B derivatives
EP0431874A1 (en) * 1989-12-08 1991-06-12 Beecham Group p.l.c. Novel compounds
US5185366A (en) * 1990-07-31 1993-02-09 Ohio State University Research Foundation Method for treatment and prevention of diseases caused by enveloped viruses, including herpes simplex virus types 1 and 2 diseases, using 3,4-dihydroxy-2H-benzopyran-2H-one
US5120718A (en) * 1991-06-13 1992-06-09 Abbott Laboratories Candida acid protease inhibiting compounds
WO1993003737A1 (en) * 1991-08-14 1993-03-04 Liposome Technology, Inc. Hiv-treatment method with low-toxicity amphotericin b

Also Published As

Publication number Publication date
KR930702994A (ko) 1993-11-29
WO1993009791A3 (fr) 1993-06-24
AU3162893A (en) 1993-06-15
WO1993009791A2 (fr) 1993-05-27
CA2099490A1 (fr) 1993-05-15
FR2683723B1 (fr) 1995-05-19
AU669143B2 (en) 1996-05-30
TW225991B (es) 1994-07-01
EP0542630A2 (fr) 1993-05-19
FR2683723A1 (fr) 1993-05-21
JPH06504295A (ja) 1994-05-19
US5514662A (en) 1996-05-07
EP0542630A3 (en) 1993-08-04

Similar Documents

Publication Publication Date Title
MX9206563A (es) Utilizacion de derivados de anfotericina b como inhibidores de proteasas.
AR005703A1 (es) Oxazolidinonas sustituidas, procedimiento para su preparacion, uso de las mismas para preparar medicamentos y medicamentos que las contienen
ES2053778T3 (es) Procedimiento para la obtencion de derivados del tiazol.
ES2054860T5 (es) Derivados de 9-halogeno-(z)-prostaglandinas, procedimiento para su preparacion y su utilizacion como medicamentos.
PA8468401A1 (es) Compuestos para el tratamiento de la isquemia
PA8493401A1 (es) Uso de inhibidores de cyp2d6 en terapias de combinacion
DE69322390T2 (de) Absorbierder artikel mit slipseiten umgreifenden schutzelementen
AR021535A1 (es) Formas de dosificacion de liberacion controlada que comprenden zolpidem o sales del mismo
FI941222A (fi) Ei-peptidyyli-tyyppisiä integriini-inhibiittoreita, jotka ovat spesifisiä GPIIbIIIa-reseptorin suhteen
DK0815856T3 (da) Retrovirale proteaseinhibitorer
ES2083668T5 (es) Combinaciones antiviricas que contienen analogos de nucleosido.
MX9307821A (es) Nueva clase de inhibidores de proteasa aspartilo.
ES2089687T3 (es) 4-fenil-piridonas y 4-fenil-2-alcoxipiridinas sustituidas como inhibidores de la hmg-coa-reductasa.
PA8586801A1 (es) Inhibidores de hiv-integrasa, composiciones farmaceuticas y metodos para su uso
ES2043665T3 (es) 6,11-dihidro-11-(4-piperidiliden)-5h-benzo-(5,6)-ciclohepta-(1,2-b)-piridinas y composiciones y metodos de uso.
MX9300399A (es) Derivados heterotriciclicos.
AR013411A1 (es) Composicion de aplicacion para tratamientos antivirales y afecciones micosicas y/o bacterianas y utilizacion de dichas composiciones.
ES2125356T3 (es) Empleo de leflunomida para la inhibicion de interleuquina 8.
DE59102350D1 (de) Lichtschutz.
AR021463A1 (es) Antibiotico de piridona con perfil de seguridad mejorado
UY27394A1 (es) Pedidos con actividad anti- angiogéna.
AR008236A1 (es) Forma cristalina anhidra del clorhidrato de acido r(-)-n-(4,4-di(3- metiltien-2-il)but-3-enil)-nipecotico, una composicion farmaceutica y el uso de dicha sal cristalina para la preparacion de una composicion farmaceutica
ES2097023T3 (es) Derivados del acido succinoilamino-hidroxietilamino-sulfamico utiles como inhibidores de proteasas retrovirales.
MX9206365A (es) Tetrahidrobenzotienopiridinas,proceso para su preparacion y composicion farmaceutica que las contiene
ES2188797T3 (es) Sales de n-(4-oxo-2-(1h-tetrazoil-5-il)-4h-1 benzopran-8-il)-4-(4-fenilbutoxi)benzamida.

Legal Events

Date Code Title Description
FA Abandonment or withdrawal