MX394784B - Composiciones farmacéuticas de un inhibidor de tirosina cinasa de bruton. - Google Patents

Composiciones farmacéuticas de un inhibidor de tirosina cinasa de bruton.

Info

Publication number
MX394784B
MX394784B MX2017011270A MX2017011270A MX394784B MX 394784 B MX394784 B MX 394784B MX 2017011270 A MX2017011270 A MX 2017011270A MX 2017011270 A MX2017011270 A MX 2017011270A MX 394784 B MX394784 B MX 394784B
Authority
MX
Mexico
Prior art keywords
tyrosine kinase
pharmaceutical compositions
kinase inhibitor
conditions
bruton tyrosine
Prior art date
Application number
MX2017011270A
Other languages
English (en)
Spanish (es)
Other versions
MX2017011270A (es
Inventor
Ching Wah Chong
Harisha Atluri
Heow Tan
Robert Kuehl
Original Assignee
Pharmacyclics Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=56848552&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX394784(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Llc filed Critical Pharmacyclics Llc
Publication of MX2017011270A publication Critical patent/MX2017011270A/es
Publication of MX394784B publication Critical patent/MX394784B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Inorganic Chemistry (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
MX2017011270A 2015-03-03 2016-03-02 Composiciones farmacéuticas de un inhibidor de tirosina cinasa de bruton. MX394784B (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562127717P 2015-03-03 2015-03-03
US201562193518P 2015-07-16 2015-07-16
PCT/US2016/020467 WO2016141068A1 (en) 2015-03-03 2016-03-02 Pharmaceutical formulations of bruton's tyrosine kinase inhibtor

Publications (2)

Publication Number Publication Date
MX2017011270A MX2017011270A (es) 2018-01-12
MX394784B true MX394784B (es) 2025-03-24

Family

ID=56848552

Family Applications (5)

Application Number Title Priority Date Filing Date
MX2017011270A MX394784B (es) 2015-03-03 2016-03-02 Composiciones farmacéuticas de un inhibidor de tirosina cinasa de bruton.
MX2021015408A MX2021015408A (es) 2015-03-03 2017-09-04 Composiciones farmaceuticas de un inhibidor de tirosina cinasa de bruton.
MX2021015370A MX2021015370A (es) 2015-03-03 2017-09-04 Composiciones farmaceuticas de un inhibidor de tirosina cinasa de bruton.
MX2021015405A MX2021015405A (es) 2015-03-03 2017-09-04 Composiciones farmaceuticas de un inhibidor de tirosina cinasa de bruton.
MX2021015368A MX2021015368A (es) 2015-03-03 2017-09-04 Composiciones farmaceuticas de un inhibidor de tirosina cinasa de bruton.

Family Applications After (4)

Application Number Title Priority Date Filing Date
MX2021015408A MX2021015408A (es) 2015-03-03 2017-09-04 Composiciones farmaceuticas de un inhibidor de tirosina cinasa de bruton.
MX2021015370A MX2021015370A (es) 2015-03-03 2017-09-04 Composiciones farmaceuticas de un inhibidor de tirosina cinasa de bruton.
MX2021015405A MX2021015405A (es) 2015-03-03 2017-09-04 Composiciones farmaceuticas de un inhibidor de tirosina cinasa de bruton.
MX2021015368A MX2021015368A (es) 2015-03-03 2017-09-04 Composiciones farmaceuticas de un inhibidor de tirosina cinasa de bruton.

Country Status (28)

Country Link
US (9) US9655857B2 (OSRAM)
EP (2) EP4338738A3 (OSRAM)
JP (3) JP7149076B2 (OSRAM)
KR (2) KR20250016514A (OSRAM)
CN (1) CN107427498A (OSRAM)
AU (4) AU2016226279B2 (OSRAM)
BR (2) BR122023020985A2 (OSRAM)
CA (3) CA2976695C (OSRAM)
DK (1) DK3265084T3 (OSRAM)
ES (1) ES2971597T3 (OSRAM)
FI (1) FI3265084T3 (OSRAM)
HR (1) HRP20240231T1 (OSRAM)
HU (1) HUE065703T2 (OSRAM)
IL (3) IL315294A (OSRAM)
LT (1) LT3265084T (OSRAM)
MD (1) MD3265084T2 (OSRAM)
MX (5) MX394784B (OSRAM)
NZ (1) NZ734446A (OSRAM)
PL (1) PL3265084T3 (OSRAM)
PT (1) PT3265084T (OSRAM)
RS (1) RS65234B1 (OSRAM)
RU (1) RU2017133990A (OSRAM)
SG (2) SG11201707122QA (OSRAM)
SI (1) SI3265084T1 (OSRAM)
SM (1) SMT202400074T1 (OSRAM)
TW (5) TWI733027B (OSRAM)
WO (1) WO2016141068A1 (OSRAM)
ZA (1) ZA201907661B (OSRAM)

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KR20250151610A (ko) 2012-06-04 2025-10-21 파마싸이클릭스 엘엘씨 브루톤 타이로신 키나아제 저해제의 결정 형태
BR112015001690A2 (pt) 2012-07-24 2017-11-07 Pharmacyclics Inc mutações associadas com a resistência a inibidores da tirosina quinase de bruton (btk)
CA2928721C (en) * 2013-10-25 2020-12-22 Pharmacyclics Llc Use of ibrutinib for treating and preventing chronic graft versus host disease
PH12020552048A1 (en) * 2013-12-02 2022-05-11 Pharmacyclics Llc Methods of treating and preventing alloantibody driven chronic graft versus host disease
CA2955747A1 (en) * 2014-08-07 2016-02-11 Pharmacyclics Llc Novel formulations of a bruton's tyrosine kinase inhibitor
IL315294A (en) * 2015-03-03 2024-10-01 Pharmacyclics Llc Pharmaceutical formulations of bruton's tyrosine kinase inhibitor
KR20170129804A (ko) 2015-03-20 2017-11-27 더 트러스티스 오브 더 유니버시티 오브 펜실바니아 Cd40 리간드를 어쥬번트로서 갖는 백신
DK3892302T3 (da) * 2015-04-06 2023-11-13 Janssen Pharmaceutica Nv Sammensætninger indeholdende ibrutinib
MX2018008771A (es) * 2016-01-19 2018-11-09 Janssen Pharmaceutica Nv Formulaciones/composiciones que comprenden un inhibidor de btk.
WO2018065504A1 (en) 2016-10-06 2018-04-12 Janssen Pharmaceutica Nv Processes and intermediates for preparing a btk inhibitor
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US20210228479A1 (en) * 2020-01-29 2021-07-29 Farmakeio Nutraceuticals Llc Steroidal compositions and method of making and use
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