MX2022006500A - Terapia de combinacion que involucra compuestos macrociclicos de diarilo. - Google Patents
Terapia de combinacion que involucra compuestos macrociclicos de diarilo.Info
- Publication number
- MX2022006500A MX2022006500A MX2022006500A MX2022006500A MX2022006500A MX 2022006500 A MX2022006500 A MX 2022006500A MX 2022006500 A MX2022006500 A MX 2022006500A MX 2022006500 A MX2022006500 A MX 2022006500A MX 2022006500 A MX2022006500 A MX 2022006500A
- Authority
- MX
- Mexico
- Prior art keywords
- combination therapy
- macrocyclic compounds
- therapy involving
- diaryl
- diaryl macrocyclic
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente divulgación se refiere a los métodos y las composiciones utilizados para el tratamiento de cáncer con el macrociclo de diarilo en combinación con un inhibidor KRAS, tal como un inhibidor de KRAS G12C.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201962941026P | 2019-11-27 | 2019-11-27 | |
US202062981822P | 2020-02-26 | 2020-02-26 | |
US202063005681P | 2020-04-06 | 2020-04-06 | |
PCT/US2020/062390 WO2021108682A1 (en) | 2019-11-27 | 2020-11-25 | Combination therapy involving diaryl macrocyclic compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2022006500A true MX2022006500A (es) | 2022-07-04 |
Family
ID=76129920
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2022006500A MX2022006500A (es) | 2019-11-27 | 2020-11-25 | Terapia de combinacion que involucra compuestos macrociclicos de diarilo. |
Country Status (12)
Country | Link |
---|---|
US (2) | US11654145B2 (es) |
EP (1) | EP4065125A4 (es) |
JP (1) | JP2023505056A (es) |
KR (1) | KR20220133866A (es) |
CN (1) | CN114901286B (es) |
AU (1) | AU2020391222A1 (es) |
BR (1) | BR112022010278A2 (es) |
CA (1) | CA3162632A1 (es) |
IL (1) | IL293206A (es) |
MX (1) | MX2022006500A (es) |
TW (1) | TW202133855A (es) |
WO (1) | WO2021108682A1 (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA3168648A1 (en) * | 2020-01-31 | 2021-08-05 | Verastem, Inc. | Combination therapy for treating abnormal cell growth |
BR112023018734A2 (pt) * | 2021-03-17 | 2023-10-24 | Amgen Inc | Regimes de dosagem de sotorasib |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2011060328A1 (en) * | 2009-11-13 | 2011-05-19 | Infinity Pharmaceuticals, Inc. | Compositions, kits, and methods for identification, assessment, prevention, and therapy of cancer |
ES2735729T3 (es) | 2014-01-24 | 2019-12-20 | Turning Point Therapeutics Inc | Macrociclos de diarilo como moduladores de proteínas cinasas |
JO3556B1 (ar) | 2014-09-18 | 2020-07-05 | Araxes Pharma Llc | علاجات مدمجة لمعالجة السرطان |
US10316044B2 (en) * | 2015-07-02 | 2019-06-11 | Tp Therapeutics, Inc. | Chiral diaryl macrocycles as modulators of protein kinases |
BR112018000297A2 (pt) * | 2015-07-06 | 2018-09-04 | Tp Therapeutics Inc | polimorfo de macrociclo de diarila |
BR112018008357A2 (pt) * | 2015-10-26 | 2018-11-27 | Array Biopharma Inc | mutações de ponto em câncer resistente a inibidor de trk e métodos relacionados às mesmas |
TWI808958B (zh) * | 2017-01-25 | 2023-07-21 | 美商特普醫葯公司 | 涉及二芳基巨環化合物之組合療法 |
US20190134056A1 (en) * | 2017-03-10 | 2019-05-09 | The Trustees Of The Stevens Institute Of Technolog | K-ras mutations and antagonists |
JOP20190272A1 (ar) | 2017-05-22 | 2019-11-21 | Amgen Inc | مثبطات kras g12c وطرق لاستخدامها |
HUE061599T2 (hu) | 2017-11-15 | 2023-07-28 | Mirati Therapeutics Inc | KRas G12C inhibotorok |
US10647715B2 (en) | 2017-11-15 | 2020-05-12 | Mirati Therapeutics, Inc. | KRas G12C inhibitors |
JP7060694B2 (ja) * | 2018-01-18 | 2022-04-26 | アレイ バイオファーマ インコーポレイテッド | Retキナーゼ阻害剤としての置換ピロロ[2,3-d]ピリミジン化合物 |
JP2022500381A (ja) * | 2018-09-10 | 2022-01-04 | ミラティ セラピューティクス, インコーポレイテッド | 組み合わせ療法 |
CN110256421A (zh) * | 2019-06-26 | 2019-09-20 | 微境生物医药科技(上海)有限公司 | Kras-g12c抑制剂 |
CA3163095A1 (en) * | 2019-11-27 | 2021-06-03 | Turning Point Therapeutics, Inc. | Combination therapy involving diaryl macrocyclic compounds |
WO2021148581A1 (en) * | 2020-01-22 | 2021-07-29 | Onxeo | Novel dbait molecule and its use |
-
2020
- 2020-11-25 CN CN202080089330.6A patent/CN114901286B/zh active Active
- 2020-11-25 KR KR1020227021852A patent/KR20220133866A/ko unknown
- 2020-11-25 TW TW109141454A patent/TW202133855A/zh unknown
- 2020-11-25 CA CA3162632A patent/CA3162632A1/en active Pending
- 2020-11-25 BR BR112022010278A patent/BR112022010278A2/pt unknown
- 2020-11-25 WO PCT/US2020/062390 patent/WO2021108682A1/en unknown
- 2020-11-25 MX MX2022006500A patent/MX2022006500A/es unknown
- 2020-11-25 AU AU2020391222A patent/AU2020391222A1/en active Pending
- 2020-11-25 EP EP20894516.2A patent/EP4065125A4/en active Pending
- 2020-11-25 IL IL293206A patent/IL293206A/en unknown
- 2020-11-25 US US17/104,752 patent/US11654145B2/en active Active
- 2020-11-25 JP JP2022531006A patent/JP2023505056A/ja active Pending
-
2023
- 2023-04-24 US US18/138,644 patent/US20240033266A1/en active Pending
Also Published As
Publication number | Publication date |
---|---|
EP4065125A1 (en) | 2022-10-05 |
US20240033266A1 (en) | 2024-02-01 |
AU2020391222A1 (en) | 2022-06-30 |
CA3162632A1 (en) | 2021-06-03 |
TW202133855A (zh) | 2021-09-16 |
CN114901286B (zh) | 2024-05-10 |
JP2023505056A (ja) | 2023-02-08 |
IL293206A (en) | 2022-07-01 |
WO2021108682A1 (en) | 2021-06-03 |
US20210220364A1 (en) | 2021-07-22 |
EP4065125A4 (en) | 2024-01-03 |
US11654145B2 (en) | 2023-05-23 |
CN114901286A (zh) | 2022-08-12 |
KR20220133866A (ko) | 2022-10-05 |
BR112022010278A2 (pt) | 2022-10-04 |
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