MX2022002718A - Compuestos inhibidores de rip1 y metodos para preparar y usar los mismos. - Google Patents

Compuestos inhibidores de rip1 y metodos para preparar y usar los mismos.

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Publication number
MX2022002718A
MX2022002718A MX2022002718A MX2022002718A MX2022002718A MX 2022002718 A MX2022002718 A MX 2022002718A MX 2022002718 A MX2022002718 A MX 2022002718A MX 2022002718 A MX2022002718 A MX 2022002718A MX 2022002718 A MX2022002718 A MX 2022002718A
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Mexico
Prior art keywords
inhibitory compounds
rip1
making
methods
same
Prior art date
Application number
MX2022002718A
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English (en)
Inventor
Somasekhar Bhamidipati
Vanessa Taylor
Original Assignee
Rigel Pharmaceuticals Inc
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Filing date
Publication date
Application filed by Rigel Pharmaceuticals Inc filed Critical Rigel Pharmaceuticals Inc
Publication of MX2022002718A publication Critical patent/MX2022002718A/es

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Abstract

En la presente descripción se describen compuestos inhibidores de cinasas, tales como compuestos inhibidores de la proteína cinasa 1 que interactúa con el receptor (RIP1), así como también composiciones farmacéuticas y combinaciones que comprenden tales compuestos inhibidores. Los compuestos, composiciones farmacéuticas y/o combinaciones descritas pueden usarse para tratar o prevenir una enfermedad o afección asociada a cinasas, particularmente una enfermedad o afección asociada a RIP1.
MX2022002718A 2019-09-06 2020-09-04 Compuestos inhibidores de rip1 y metodos para preparar y usar los mismos. MX2022002718A (es)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201962897223P 2019-09-06 2019-09-06
US201962932404P 2019-11-07 2019-11-07
US202063001016P 2020-03-27 2020-03-27
US202063004301P 2020-04-02 2020-04-02
US202063004290P 2020-04-02 2020-04-02
US202063004319P 2020-04-02 2020-04-02
PCT/US2020/049451 WO2021046382A1 (en) 2019-09-06 2020-09-04 Rip1 inhibitory compounds and methods for making and using the same

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MX2022002718A true MX2022002718A (es) 2022-08-10

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Application Number Title Priority Date Filing Date
MX2022002737A MX2022002737A (es) 2019-09-06 2020-09-04 Compuestos inhibidores de rip1 y metodos para hacer y utilizar los mismos.
MX2022002719A MX2022002719A (es) 2019-09-06 2020-09-04 Inhibidores heterociclicos de la quinasa rip1.
MX2022002718A MX2022002718A (es) 2019-09-06 2020-09-04 Compuestos inhibidores de rip1 y metodos para preparar y usar los mismos.

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MX2022002737A MX2022002737A (es) 2019-09-06 2020-09-04 Compuestos inhibidores de rip1 y metodos para hacer y utilizar los mismos.
MX2022002719A MX2022002719A (es) 2019-09-06 2020-09-04 Inhibidores heterociclicos de la quinasa rip1.

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US (6) US11479543B2 (es)
EP (3) EP4025568A1 (es)
JP (4) JP7376218B2 (es)
KR (3) KR20220042204A (es)
CN (3) CN114761398A (es)
AU (3) AU2020343681B2 (es)
BR (3) BR112022002580A2 (es)
CA (3) CA3149963A1 (es)
CO (1) CO2022002630A2 (es)
DO (1) DOP2022000051A (es)
EC (1) ECSP22016571A (es)
IL (3) IL290780A (es)
JO (1) JOP20220062A1 (es)
MX (3) MX2022002737A (es)
PE (1) PE20221628A1 (es)
TW (3) TW202122389A (es)
WO (3) WO2021046407A1 (es)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY192762A (en) * 2015-07-02 2022-09-07 Hoffmann La Roche Bicyclic lactams and methods of use thereof
WO2019213447A1 (en) 2018-05-03 2019-11-07 Rigel Pharmaceuticals, Inc. Rip1 inhibitory compounds and methods for making and using the same
MD3788045T2 (ro) 2018-05-03 2023-09-30 Rigel Pharmaceuticals Inc Compuși inhibitori ai RIP1 și procedee de obţinere și utilizare a acestora
CA3149963A1 (en) 2019-09-06 2021-03-11 Simon Shaw Heterocyclic rip1 kinase inhibitors
JOP20220056A1 (ar) 2019-09-06 2023-01-30 Rigel Pharmaceuticals Inc مركبات rip1 تثبيطية وطرق عملها واستخدامها
TW202132307A (zh) * 2019-11-07 2021-09-01 美商雷傑製藥公司 雜環ｒｉｐ１抑制性化合物
AU2021225921A1 (en) * 2020-02-28 2022-09-22 Board Of Regents, The University Of Texas System Inhibitors of Receptor Interacting Protein Kinase I for the treatment of disease
AR121717A1 (es) 2020-04-02 2022-06-29 Rigel Pharmaceuticals Inc Inhibidores de rip1k
AR122703A1 (es) 2020-07-01 2022-09-28 Rigel Pharmaceuticals Inc Inhibidores de rip1k
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