MX2020012523A - Proceso para producir 4-aminoindanos sustituidos. - Google Patents

Proceso para producir 4-aminoindanos sustituidos.

Info

Publication number
MX2020012523A
MX2020012523A MX2020012523A MX2020012523A MX2020012523A MX 2020012523 A MX2020012523 A MX 2020012523A MX 2020012523 A MX2020012523 A MX 2020012523A MX 2020012523 A MX2020012523 A MX 2020012523A MX 2020012523 A MX2020012523 A MX 2020012523A
Authority
MX
Mexico
Prior art keywords
producing
present
aminoindanes
substituted
inden
Prior art date
Application number
MX2020012523A
Other languages
English (en)
Inventor
Mark James Ford
Florian Erver
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of MX2020012523A publication Critical patent/MX2020012523A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C11/00—Aliphatic unsaturated hydrocarbons
    • C07C11/02—Alkenes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/04—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups
    • C07C209/06—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms
    • C07C209/10—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms with formation of amino groups bound to carbon atoms of six-membered aromatic rings or from amines having nitrogen atoms bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/54—Preparation of compounds containing amino groups bound to a carbon skeleton by rearrangement reactions
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/68—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/44—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring
    • C07C211/45—Monoamines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/44—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring
    • C07C211/45—Monoamines
    • C07C211/48—N-alkylated amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/57—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton
    • C07C211/60—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton containing a ring other than a six-membered aromatic ring forming part of at least one of the condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/16—Systems containing only non-condensed rings with a six-membered ring the ring being unsaturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pyridine Compounds (AREA)

Abstract

La presente invención se refiere principalmente a un proceso para producir ciertas 2-alilanilinas sustituidas de la fórmula (I) anteriormente definida y su uso en un proceso para producir derivados de 4-aminoindano sustituidos de fórmula (V) anteriormente definida. La presente invención se refiere además a un proceso para producir indanilo carboxamidas fungicidas. En particular, la presente invención se refiere a un proceso para producir 2-(difluorometil)-N-(1,1-dimetil-3-propil-2,3-dihidro-1H- inden-4-il)nicotinamida y/o 3- (difluorometil)-N-[(R)-2,3-dihidro- 1,1,3-trimetil-1H-inden-4-il]-1-metilpirazol-4-carboxamida.
MX2020012523A 2018-05-23 2019-05-21 Proceso para producir 4-aminoindanos sustituidos. MX2020012523A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18173859 2018-05-23
EP18173856 2018-05-23
PCT/EP2019/063063 WO2019224181A1 (en) 2018-05-23 2019-05-21 Process for producing substituted 4-aminoindanes

Publications (1)

Publication Number Publication Date
MX2020012523A true MX2020012523A (es) 2021-02-16

Family

ID=66625989

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2020012523A MX2020012523A (es) 2018-05-23 2019-05-21 Proceso para producir 4-aminoindanos sustituidos.

Country Status (9)

Country Link
US (1) US20210363106A1 (es)
JP (1) JP2021524854A (es)
KR (1) KR20210011382A (es)
CN (1) CN112119061A (es)
BR (1) BR112020023624A2 (es)
IL (1) IL278815A (es)
MX (1) MX2020012523A (es)
TW (1) TW202016074A (es)
WO (1) WO2019224181A1 (es)

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT649888A (es) * 1960-03-02
ES2011602T3 (es) 1986-08-12 1994-07-16 Mitsubishi Chem Ind Derivados de piridinacarboxamida y su uso como fungicidas.
US5093347A (en) 1991-01-28 1992-03-03 Monsanto Company 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use
EP0654464A1 (en) 1993-10-22 1995-05-24 Shell Internationale Researchmaatschappij B.V. Processes for the preparation of pesticides and intermediates
US5521317A (en) 1993-10-22 1996-05-28 American Cyanamid Co. Processes for the preparation of pesticides and intermediates
JP3675112B2 (ja) 1997-06-23 2005-07-27 富士写真フイルム株式会社 画像読取装置及び情報処理装置
JP2009545565A (ja) 2006-08-01 2009-12-24 ノシーラ ソシエダー アノニマ 認知性、神経変性性、または神経性の疾患または障害の治療のためのｎ−フェニル−プレニルアミン誘導体
ITMI20090488A1 (it) 2009-03-27 2010-09-28 Isagro Ricerca Srl Composti benzammidici ad elevata attivita' fungicida e relativo uso
US9375004B2 (en) 2010-11-15 2016-06-28 Bayer Intellectual Property Gmbh 5-halogenopyrazolecarboxamides
IT1403275B1 (it) 2010-12-20 2013-10-17 Isagro Ricerca Srl Indanilanilidi ad elevata attività fungicida e loro composizioni fitosanitarie
JP6240666B2 (ja) 2012-05-09 2017-11-29 バイエル・クロップサイエンス・アクチェンゲゼルシャフト ピラゾールインダニルカルボキサミド類
US9249104B2 (en) 2012-05-09 2016-02-02 Bayer Cropscience Ag Pyrazole indanyl carboxamides
EP2935213B1 (en) 2012-12-19 2019-05-22 Bayer CropScience Aktiengesellschaft Difluoromethyl-nicotinic-indanyl carboxamides as fungicides
BR112015015097B1 (pt) 2012-12-27 2021-02-17 Sumitomo Chemical Company, Limited método para produção de composto de amina purificada
AR101820A1 (es) * 2014-06-25 2017-01-18 Bayer Cropscience Ag Difluorometil-indanil-carboxamidas nicotínicas
TW201738200A (zh) * 2016-02-03 2017-11-01 拜耳作物科學股份有限公司 製備經取代的４－胺基茚烷衍生物之方法
US10640454B2 (en) 2016-04-15 2020-05-05 Stichting I-F Product Collaboration Processes for preparation of 4-aminoindane compounds and related aminoindane amides

Also Published As

Publication number Publication date
TW202016074A (zh) 2020-05-01
KR20210011382A (ko) 2021-02-01
JP2021524854A (ja) 2021-09-16
IL278815A (en) 2021-01-31
CN112119061A (zh) 2020-12-22
BR112020023624A2 (pt) 2021-02-17
US20210363106A1 (en) 2021-11-25
WO2019224181A1 (en) 2019-11-28

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