MX2020007092A - Metodos de uso de inhibidores ehmt2 para tratar o prevenir transtornos sanguineos. - Google Patents

Metodos de uso de inhibidores ehmt2 para tratar o prevenir transtornos sanguineos.

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Publication number
MX2020007092A
MX2020007092A MX2020007092A MX2020007092A MX2020007092A MX 2020007092 A MX2020007092 A MX 2020007092A MX 2020007092 A MX2020007092 A MX 2020007092A MX 2020007092 A MX2020007092 A MX 2020007092A MX 2020007092 A MX2020007092 A MX 2020007092A
Authority
MX
Mexico
Prior art keywords
treating
methods
blood disorders
preventing blood
ehmt2
Prior art date
Application number
MX2020007092A
Other languages
English (en)
Inventor
Elayne Penebre
Veronica Gibaja
Maria Alejandra Raimondi
Original Assignee
Epizyme Inc
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Filing date
Publication date
Application filed by Epizyme Inc filed Critical Epizyme Inc
Publication of MX2020007092A publication Critical patent/MX2020007092A/es

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    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
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Abstract

La presente divulgación se refiere a un método para prevenir o tratar un trastorno sanguineo (por ejemplo, enfermedad de células falciformes) mediante la administración de un compuesto inhibidor de EHMT2 desvelado en este documento o una composición farmacéutica del mismo a sujetos que lo necesitan. La presente divulgación también se refiere al uso de tales compuestos en investigación u otros fines no terapéuticos.
MX2020007092A 2017-10-18 2018-10-18 Metodos de uso de inhibidores ehmt2 para tratar o prevenir transtornos sanguineos. MX2020007092A (es)

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PCT/US2018/056530 WO2019079607A1 (en) 2017-10-18 2018-10-18 METHODS OF USING EHMT2 INHIBITORS IN THE TREATMENT OR PREVENTION OF BLOOD DISORDERS

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