MX2018012439A - Composiciones y metodos para el tratamiento de enfermedades de la mucosa nasal y paranasal con agonistas del receptor de acetilcolina de tipo nicotinico. - Google Patents

Composiciones y metodos para el tratamiento de enfermedades de la mucosa nasal y paranasal con agonistas del receptor de acetilcolina de tipo nicotinico.

Info

Publication number
MX2018012439A
MX2018012439A MX2018012439A MX2018012439A MX2018012439A MX 2018012439 A MX2018012439 A MX 2018012439A MX 2018012439 A MX2018012439 A MX 2018012439A MX 2018012439 A MX2018012439 A MX 2018012439A MX 2018012439 A MX2018012439 A MX 2018012439A
Authority
MX
Mexico
Prior art keywords
methods
acetylcholine receptor
nicotinic acetylcholine
compositions
receptor agonists
Prior art date
Application number
MX2018012439A
Other languages
English (en)
Inventor
Solis Herrera Arturo
Original Assignee
Solis Herrera Arturo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from AU2016901359A external-priority patent/AU2016901359A0/en
Application filed by Solis Herrera Arturo filed Critical Solis Herrera Arturo
Publication of MX2018012439A publication Critical patent/MX2018012439A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/465Nicotine; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/60Salicylic acid; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0043Nose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/12Aerosols; Foams
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12Carboxylic acids; Salts or anhydrides thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61NELECTROTHERAPY; MAGNETOTHERAPY; RADIATION THERAPY; ULTRASOUND THERAPY
    • A61N5/00Radiation therapy
    • A61N5/06Radiation therapy using light
    • A61N5/0601Apparatus for use inside the body
    • A61N5/0603Apparatus for use inside the body for treatment of body cavities
    • A61N2005/0607Nose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61NELECTROTHERAPY; MAGNETOTHERAPY; RADIATION THERAPY; ULTRASOUND THERAPY
    • A61N5/00Radiation therapy
    • A61N5/06Radiation therapy using light
    • A61N5/0601Apparatus for use inside the body
    • A61N5/0603Apparatus for use inside the body for treatment of body cavities

Abstract

Se describen metodos de tratamiento y prevencion de condiciones de una membrana mucosa nasal o paranasal; los metodos incluyen administrar una composicion farmaceutica que incluye un agonista del receptor de acetilcolina de tipo nicotinico (nAChR), tal como (S)-(1-metil-2-pirrolidinil)-piridina, o una sal, analogo, precursor, o derivado farmaceuticamente aceptable del mismo; los metodos se pueden usar para tratar una amplia variedad de condiciones de la membrana mucosa nasal o paranasal, tal como congestion nasal y sangrados nasales.
MX2018012439A 2016-04-12 2017-04-12 Composiciones y metodos para el tratamiento de enfermedades de la mucosa nasal y paranasal con agonistas del receptor de acetilcolina de tipo nicotinico. MX2018012439A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AU2016901359A AU2016901359A0 (en) 2016-04-12 Application of Nicotine Compounds to Nasal Membranes
PCT/IB2017/000764 WO2017178897A2 (en) 2016-04-12 2017-04-12 Compositions and methods for treating paranasal mucosa diseases with nicotinic acetylcholine receptor agonists

Publications (1)

Publication Number Publication Date
MX2018012439A true MX2018012439A (es) 2019-02-21

Family

ID=60042487

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2018012439A MX2018012439A (es) 2016-04-12 2017-04-12 Composiciones y metodos para el tratamiento de enfermedades de la mucosa nasal y paranasal con agonistas del receptor de acetilcolina de tipo nicotinico.

Country Status (13)

Country Link
US (1) US10639300B2 (es)
EP (1) EP3442583B1 (es)
JP (1) JP6770091B2 (es)
KR (1) KR102199560B1 (es)
CN (1) CN109069649A (es)
AU (1) AU2017250514B2 (es)
BR (2) BR122023020807A2 (es)
CA (1) CA3014725C (es)
HK (1) HK1258883A1 (es)
MX (1) MX2018012439A (es)
NZ (1) NZ744942A (es)
RU (1) RU2718061C1 (es)
WO (1) WO2017178897A2 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11096932B2 (en) * 2016-09-29 2021-08-24 The Uab Research Foundation Methods and compositions for increasing mucus clearance

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8301659D0 (en) 1983-01-21 1983-02-23 Leo Ab Smoking substitutes
GB9310412D0 (en) 1993-05-20 1993-07-07 Danbiosyst Uk Nasal nicotine system
MA23588A1 (fr) * 1994-06-23 1995-12-31 Procter & Gamble Traitement du besoin en nicotine et/ou du syndrome de manque lie au tabagisme
US6277855B1 (en) 2000-04-21 2001-08-21 Inspire Pharmaceuticals, Inc. Method of treating dry eye disease with nicotinic acetylcholine receptor agonists
US6596740B2 (en) * 2000-10-24 2003-07-22 Richard L. Jones Nicotine mucosal spray
HU224941B1 (en) 2001-08-10 2006-04-28 Bgi Innovacios Kft Phototerapy apparatus
US20040254146A1 (en) * 2002-05-21 2004-12-16 Nastech Pharmaceutical Company Inc. Carboxylate salts of galantamine and their pharmaceutical use
CN1735414A (zh) 2002-12-06 2006-02-15 北岸长岛犹太人研究学院 用α7受体结合类胆碱激动剂抑制炎症
PL1663168T3 (pl) 2003-09-08 2009-07-31 Mcneil Ab Preparaty nikotyny i ich zastosowanie
CN101001843B (zh) 2004-07-15 2014-08-27 拉瓦尔大学 用于治疗炎性疾病的烟碱受体激动剂
CN101437515B (zh) 2006-05-08 2016-04-20 阿图罗·索利斯埃雷拉 烟碱、其类似物、其前体或其衍生物用于通过以预防形式或治疗形式参与的α-MSH改善治疗各种病理过程的应用
WO2008062453A2 (en) * 2006-09-25 2008-05-29 Nikki Nikhilesh Singh Composition containing nicotine base aromatic oils and alkyl salicylate for the delivery of nicotine base in vapour form
CL2008003507A1 (es) 2007-11-26 2009-11-27 Neuroderm Ltd Composicion farmaceutica que comprende nicotina y un inhibidor de la desensibilizacion del receptor de acetilcolina nicotinico (nachr) opipramol; kit farmaceutico; dispositivo medico; y uso para tratar una enfermedad o trastorno del sistema nervioso central o periferico.
US9744375B2 (en) * 2010-08-05 2017-08-29 Allergia, Inc. Apparatus and methods for controlling and applying flash lamp radiation
WO2015084544A1 (en) 2013-12-05 2015-06-11 Ploom, Inc. Nicotine liquid formulations for aerosol devices and methods thereof
CN104706556A (zh) 2015-03-31 2015-06-17 苏州维泰生物技术有限公司 抗过敏组合物及其在化妆品中的应用

Also Published As

Publication number Publication date
AU2017250514B2 (en) 2019-12-19
RU2718061C1 (ru) 2020-03-30
AU2017250514A1 (en) 2018-08-23
EP3442583B1 (en) 2024-04-10
EP3442583A4 (en) 2019-12-25
JP2019511520A (ja) 2019-04-25
CN109069649A (zh) 2018-12-21
BR112018067718A2 (pt) 2019-01-08
WO2017178897A2 (en) 2017-10-19
US20190111038A1 (en) 2019-04-18
JP6770091B2 (ja) 2020-10-14
CA3014725C (en) 2020-09-22
HK1258883A1 (zh) 2019-11-22
CA3014725A1 (en) 2017-10-19
BR122023020807A2 (pt) 2023-12-12
NZ744942A (en) 2020-08-28
WO2017178897A3 (en) 2017-11-23
EP3442583A2 (en) 2019-02-20
US10639300B2 (en) 2020-05-05
KR20180108821A (ko) 2018-10-04
KR102199560B1 (ko) 2021-01-07

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