MX2013010009A - Metodo de radiofluoracion. - Google Patents
Metodo de radiofluoracion.Info
- Publication number
- MX2013010009A MX2013010009A MX2013010009A MX2013010009A MX2013010009A MX 2013010009 A MX2013010009 A MX 2013010009A MX 2013010009 A MX2013010009 A MX 2013010009A MX 2013010009 A MX2013010009 A MX 2013010009A MX 2013010009 A MX2013010009 A MX 2013010009A
- Authority
- MX
- Mexico
- Prior art keywords
- sup
- labelled
- present
- compound
- radiofluorination method
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
- C07B59/002—Heterocyclic compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
- C07D295/135—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención proporciona un método novedoso para obtener un compuesto 18F-marcado, en donde dicho compuesto comprende un anillo piridilo 18F-marcado. El método de la invención es ventajoso sobre los métodos de la técnica anterior ya que proporciona estos compuestos en rendimientos radioquímicos más altos que los que han sido posibles con métodos previos. También, la presente invención proporciona un sintón 18F-marcado útil en el método de la invención.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201161447724P | 2011-03-01 | 2011-03-01 | |
GBGB1103455.0A GB201103455D0 (en) | 2011-03-01 | 2011-03-01 | Radiofluorination method |
PCT/EP2012/053547 WO2012117069A1 (en) | 2011-03-01 | 2012-03-01 | Radiofluorination method |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2013010009A true MX2013010009A (es) | 2013-11-20 |
Family
ID=43904348
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2013010009A MX2013010009A (es) | 2011-03-01 | 2012-03-01 | Metodo de radiofluoracion. |
Country Status (12)
Country | Link |
---|---|
US (1) | US20130338361A1 (es) |
EP (1) | EP2681177A1 (es) |
JP (1) | JP2014514254A (es) |
KR (1) | KR20140007412A (es) |
CN (1) | CN103384654A (es) |
AU (1) | AU2012222344A1 (es) |
BR (1) | BR112013021249A2 (es) |
CA (1) | CA2828500A1 (es) |
GB (1) | GB201103455D0 (es) |
MX (1) | MX2013010009A (es) |
RU (1) | RU2013138232A (es) |
WO (1) | WO2012117069A1 (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB201409536D0 (en) * | 2014-05-29 | 2014-07-16 | Univ The Durham | Chemically modifying peptides |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5630962A (en) * | 1990-12-19 | 1997-05-20 | Hoechst Aktiengesellschaft | 2-Fluoropyridines, their preparation and their use in liquid crystal mixtures |
-
2011
- 2011-03-01 GB GBGB1103455.0A patent/GB201103455D0/en not_active Ceased
-
2012
- 2012-03-01 RU RU2013138232/04A patent/RU2013138232A/ru not_active Application Discontinuation
- 2012-03-01 CN CN201280010915XA patent/CN103384654A/zh active Pending
- 2012-03-01 WO PCT/EP2012/053547 patent/WO2012117069A1/en active Application Filing
- 2012-03-01 CA CA2828500A patent/CA2828500A1/en not_active Abandoned
- 2012-03-01 AU AU2012222344A patent/AU2012222344A1/en not_active Abandoned
- 2012-03-01 JP JP2013555877A patent/JP2014514254A/ja active Pending
- 2012-03-01 EP EP12707289.0A patent/EP2681177A1/en not_active Withdrawn
- 2012-03-01 MX MX2013010009A patent/MX2013010009A/es not_active Application Discontinuation
- 2012-03-01 KR KR1020137022752A patent/KR20140007412A/ko not_active Application Discontinuation
- 2012-03-01 US US14/001,952 patent/US20130338361A1/en not_active Abandoned
- 2012-03-01 BR BR112013021249A patent/BR112013021249A2/pt not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CA2828500A1 (en) | 2012-09-07 |
JP2014514254A (ja) | 2014-06-19 |
CN103384654A (zh) | 2013-11-06 |
WO2012117069A1 (en) | 2012-09-07 |
EP2681177A1 (en) | 2014-01-08 |
US20130338361A1 (en) | 2013-12-19 |
AU2012222344A1 (en) | 2013-08-15 |
RU2013138232A (ru) | 2015-04-10 |
BR112013021249A2 (pt) | 2019-09-24 |
GB201103455D0 (en) | 2011-04-13 |
KR20140007412A (ko) | 2014-01-17 |
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Legal Events
Date | Code | Title | Description |
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FA | Abandonment or withdrawal |