MX2011006022A - Una sal tris de 8-cloro-3-pentil-3,7-dihidro-1h-purina-2,6-diona de formula (a), sus formulaciones farmaceuticas y usos de la misma, y el procedimiento para preparar la misma. - Google Patents
Una sal tris de 8-cloro-3-pentil-3,7-dihidro-1h-purina-2,6-diona de formula (a), sus formulaciones farmaceuticas y usos de la misma, y el procedimiento para preparar la misma.Info
- Publication number
- MX2011006022A MX2011006022A MX2011006022A MX2011006022A MX2011006022A MX 2011006022 A MX2011006022 A MX 2011006022A MX 2011006022 A MX2011006022 A MX 2011006022A MX 2011006022 A MX2011006022 A MX 2011006022A MX 2011006022 A MX2011006022 A MX 2011006022A
- Authority
- MX
- Mexico
- Prior art keywords
- compound
- formula
- treatment
- dyslipidemia
- purine
- Prior art date
Links
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- A61K31/52—Purines, e.g. adenine
- A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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Landscapes
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Applications Claiming Priority (2)
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| US12059608P | 2008-12-08 | 2008-12-08 | |
| PCT/US2009/066941 WO2010068581A1 (en) | 2008-12-08 | 2009-12-07 | Novel compounds |
Publications (1)
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| MX2011006022A true MX2011006022A (es) | 2011-06-28 |
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| CN101863888B (zh) * | 2004-02-14 | 2012-07-18 | 葛兰素史密斯克莱有限责任公司 | 具有hm74a受体活性的药物 |
| HRP20100725T1 (hr) | 2005-08-10 | 2011-01-31 | Glaxosmithkline Llc | Derivati ksantina kao selektivni agonisti hm74a |
| JP2015510947A (ja) * | 2012-03-22 | 2015-04-13 | トランステック・ファーマ，エルエルシー | 小分子ｇｌｐ１ｒアゴニストのトリス（ヒドロキシメチル）アミノメタン塩ならびにその医薬組成物および使用 |
| AU2024229006A1 (en) | 2023-02-27 | 2025-09-18 | Shanton Pharma Pte. Ltd. | Crystal form of 8-chloro-3-pentyl-3,7-dihydro-1h-purin-2,6-dione compound and preparation method therefor |
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| US3657327A (en) * | 1970-06-01 | 1972-04-18 | Upjohn Co | Prostaglandin salts of tris(hydroxymethyl)aminomethane |
| US4647585A (en) | 1984-11-08 | 1987-03-03 | E. R. Squibb & Sons, Inc. | Bicycloheptane substituted ethers |
| JP2003534238A (ja) * | 1999-12-15 | 2003-11-18 | スミスクライン・ビーチャム・コーポレイション | シス−４−シアノ−４−［３−（シクロペンチルオキシ）−４−メトキシフェニル］シクロヘキサン−１−カルボン酸の塩。 |
| US20030013905A1 (en) | 2002-06-10 | 2003-01-16 | Huang Guishu Kris | Salts of cis-4-cyano-4[3(cyclopentyloxy)-4-methoxyphenyl]cyclohexane-1-carboxylic acid |
| CN101863888B (zh) * | 2004-02-14 | 2012-07-18 | 葛兰素史密斯克莱有限责任公司 | 具有hm74a受体活性的药物 |
| GB0423568D0 (en) * | 2004-10-22 | 2004-11-24 | Smithkline Beecham Corp | Novel compounds |
| US20090209561A1 (en) | 2004-10-22 | 2009-08-20 | Richard Jonathan Daniel Hatley | Xanthine Derivatives with HM74A Receptor Activity |
| HRP20100725T1 (hr) | 2005-08-10 | 2011-01-31 | Glaxosmithkline Llc | Derivati ksantina kao selektivni agonisti hm74a |
| GB0516464D0 (en) * | 2005-08-10 | 2005-09-14 | Smithkline Beecham Corp | Novel compounds |
-
2009
- 2009-12-07 ES ES09832421.3T patent/ES2527354T3/es active Active
- 2009-12-07 CA CA2746316A patent/CA2746316C/en not_active Expired - Fee Related
- 2009-12-07 EP EP09832421.3A patent/EP2370440B1/en active Active
- 2009-12-07 JP JP2011539772A patent/JP5666464B2/ja not_active Expired - Fee Related
- 2009-12-07 WO PCT/US2009/066941 patent/WO2010068581A1/en not_active Ceased
- 2009-12-07 MX MX2011006022A patent/MX2011006022A/es active IP Right Grant
- 2009-12-07 BR BRPI0922134-4A patent/BRPI0922134A2/pt not_active Application Discontinuation
- 2009-12-07 US US13/133,486 patent/US9163024B2/en not_active Expired - Fee Related
- 2009-12-07 EA EA201170783A patent/EA020037B1/ru not_active IP Right Cessation
- 2009-12-07 RS RS20150086A patent/RS53777B1/sr unknown
- 2009-12-07 PT PT98324213T patent/PT2370440E/pt unknown
- 2009-12-07 HR HRP20150026AT patent/HRP20150026T1/hr unknown
- 2009-12-07 PL PL09832421T patent/PL2370440T3/pl unknown
- 2009-12-07 DK DK09832421.3T patent/DK2370440T3/en active
- 2009-12-07 SI SI200931113T patent/SI2370440T1/sl unknown
- 2009-12-07 CN CN200980148973.7A patent/CN102245606B/zh not_active Expired - Fee Related
- 2009-12-07 KR KR1020117012975A patent/KR101743783B1/ko not_active Expired - Fee Related
- 2009-12-07 AU AU2009324811A patent/AU2009324811B2/en not_active Ceased
-
2011
- 2011-05-10 ZA ZA2011/03397A patent/ZA201103397B/en unknown
- 2011-05-19 IL IL213032A patent/IL213032A/en not_active IP Right Cessation
-
2014
- 2014-12-16 CY CY20141101047T patent/CY1116032T1/el unknown
-
2015
- 2015-01-16 SM SM201500012T patent/SMT201500012B/xx unknown
- 2015-08-31 US US14/840,549 patent/US20150366870A1/en not_active Abandoned
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2016
- 2016-10-11 US US15/289,996 patent/US20170027945A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP2370440B1 (en) | 2014-11-12 |
| AU2009324811A1 (en) | 2011-06-23 |
| AU2009324811B2 (en) | 2013-01-24 |
| US20170027945A1 (en) | 2017-02-02 |
| SMT201500012B (it) | 2015-05-03 |
| HRP20150026T1 (hr) | 2015-02-13 |
| JP5666464B2 (ja) | 2015-02-12 |
| BRPI0922134A2 (pt) | 2015-08-18 |
| WO2010068581A1 (en) | 2010-06-17 |
| CA2746316C (en) | 2017-01-03 |
| US20150366870A1 (en) | 2015-12-24 |
| SI2370440T1 (sl) | 2015-02-27 |
| PT2370440E (pt) | 2015-01-14 |
| KR20110097816A (ko) | 2011-08-31 |
| ES2527354T3 (es) | 2015-01-22 |
| IL213032A (en) | 2015-02-26 |
| EA020037B1 (ru) | 2014-08-29 |
| CA2746316A1 (en) | 2010-06-17 |
| CY1116032T1 (el) | 2017-01-25 |
| RS53777B1 (sr) | 2015-06-30 |
| EP2370440A1 (en) | 2011-10-05 |
| CN102245606A (zh) | 2011-11-16 |
| IL213032A0 (en) | 2011-07-31 |
| US9163024B2 (en) | 2015-10-20 |
| JP2012511028A (ja) | 2012-05-17 |
| KR101743783B1 (ko) | 2017-06-05 |
| EA201170783A1 (ru) | 2011-12-30 |
| DK2370440T3 (en) | 2014-12-08 |
| EP2370440A4 (en) | 2012-05-30 |
| PL2370440T3 (pl) | 2015-05-29 |
| CN102245606B (zh) | 2014-08-20 |
| ZA201103397B (en) | 2012-01-25 |
| US20110251218A1 (en) | 2011-10-13 |
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