MX2010002642A - Proceso para la elaboracion de intermediarios monobactamicos puenteados. - Google Patents
Proceso para la elaboracion de intermediarios monobactamicos puenteados.Info
- Publication number
- MX2010002642A MX2010002642A MX2010002642A MX2010002642A MX2010002642A MX 2010002642 A MX2010002642 A MX 2010002642A MX 2010002642 A MX2010002642 A MX 2010002642A MX 2010002642 A MX2010002642 A MX 2010002642A MX 2010002642 A MX2010002642 A MX 2010002642A
- Authority
- MX
- Mexico
- Prior art keywords
- sub
- unsubstituted
- formula
- substituted
- group
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/40—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings
- C07C271/42—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/54—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Un proceso para elaborar un compuesto de Fórmula (I) el cual tiene conformación cis y en donde R1 representa un grupo 1-fenil-alquiloC1-C4 o 1-naftil-alquiloC1-C4, en donde la porción fenilo o naftilo de R1 es no sustituida o sustituida con uno o más grupos alcoxi C1-C4 y los átomos de carbono en la posición 2-, 3- y/o 4- de la parte alquilo de R1 son, independientemente de la porción fenilo o naftilo de R1 e independientemente uno del otro, no sustituidos o sustituidos con alcoxi C1-C4 y/o sililoxi o, preferiblemente, son no sustituidos o sustituidos con un grupo alcoxi C1-C4 y/o grupo sililoxi por átomo de carbono, y R2 representa un grupo alquilo C1-C6 o un grupo bencilo no sustituido o sustituido, en el proceso un compuesto de Fórmula (II) en donde R3 representa un grupo alquilo C1-C6 o un grupo bencilo no sustituido o sustituido, y R1 y R2 tienen el mismo significado que en la fórmula (I); es tratado con una base a una temperatura de 0° C o menor en un solvente líquido aprótico durante un período de tiempo suficiente para obtener el compuesto de la fórmula (I).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP07116603 | 2007-09-17 | ||
PCT/EP2008/062258 WO2009037229A1 (en) | 2007-09-17 | 2008-09-15 | Process for the manufacture of bridged monobactam intermediates |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2010002642A true MX2010002642A (es) | 2010-03-26 |
Family
ID=39027525
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2010002642A MX2010002642A (es) | 2007-09-17 | 2008-09-15 | Proceso para la elaboracion de intermediarios monobactamicos puenteados. |
Country Status (17)
Country | Link |
---|---|
US (2) | US8450477B2 (es) |
EP (1) | EP2197881B1 (es) |
JP (1) | JP5551072B2 (es) |
KR (1) | KR101421774B1 (es) |
CN (1) | CN101801974B (es) |
AU (1) | AU2008300616B2 (es) |
BR (1) | BRPI0816909A2 (es) |
CA (1) | CA2698441C (es) |
CY (1) | CY1114147T1 (es) |
DK (1) | DK2197881T3 (es) |
ES (1) | ES2419255T3 (es) |
HK (1) | HK1142900A1 (es) |
MX (1) | MX2010002642A (es) |
PL (1) | PL2197881T3 (es) |
PT (1) | PT2197881E (es) |
WO (1) | WO2009037229A1 (es) |
ZA (1) | ZA201001694B (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20160221992A1 (en) | 2013-05-16 | 2016-08-04 | Universite De Strasbourg | Dendritic compounds including a chelating, fluorochrome or recognition agent, compositions including same and uses thereof |
CN103554112B (zh) * | 2013-11-07 | 2016-04-13 | 中国科学院昆明植物研究所 | 顺式稠环的β-内酰胺化合物的合成方法 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1262128A (en) * | 1981-08-27 | 1989-10-03 | Christian N. Hubschwerlen | .beta.-lactams |
ZA826089B (en) * | 1981-08-27 | 1983-07-27 | Hoffmann La Roche | Beta-lactams |
DK0508234T3 (da) * | 1991-04-11 | 1996-10-28 | Hoffmann La Roche | Beta-lactamer |
CA2143519A1 (en) * | 1994-03-11 | 1995-09-12 | Markus Bohringer | Beta-lactams |
TW358097B (en) * | 1996-05-24 | 1999-05-11 | Hoffmann La Roche | Beta-lactams and their process and pharmaceutical compositions |
RS52068B (en) * | 2005-12-07 | 2012-06-30 | Basilea Pharmaceutica Ag. | USEFUL MANOBACTAM ANTIBIOTICS |
-
2008
- 2008-09-15 PL PL08804217T patent/PL2197881T3/pl unknown
- 2008-09-15 EP EP08804217.1A patent/EP2197881B1/en active Active
- 2008-09-15 MX MX2010002642A patent/MX2010002642A/es active IP Right Grant
- 2008-09-15 US US12/676,580 patent/US8450477B2/en not_active Expired - Fee Related
- 2008-09-15 PT PT88042171T patent/PT2197881E/pt unknown
- 2008-09-15 AU AU2008300616A patent/AU2008300616B2/en not_active Ceased
- 2008-09-15 WO PCT/EP2008/062258 patent/WO2009037229A1/en active Application Filing
- 2008-09-15 CA CA2698441A patent/CA2698441C/en not_active Expired - Fee Related
- 2008-09-15 DK DK08804217.1T patent/DK2197881T3/da active
- 2008-09-15 ES ES08804217T patent/ES2419255T3/es active Active
- 2008-09-15 CN CN200880107296XA patent/CN101801974B/zh not_active Expired - Fee Related
- 2008-09-15 KR KR1020107006295A patent/KR101421774B1/ko not_active IP Right Cessation
- 2008-09-15 BR BRPI0816909 patent/BRPI0816909A2/pt not_active IP Right Cessation
- 2008-09-15 JP JP2010525315A patent/JP5551072B2/ja not_active Expired - Fee Related
-
2010
- 2010-03-09 ZA ZA201001694A patent/ZA201001694B/xx unknown
- 2010-09-30 HK HK10109377.2A patent/HK1142900A1/xx not_active IP Right Cessation
-
2013
- 2013-04-26 US US13/871,338 patent/US8877961B2/en not_active Expired - Fee Related
- 2013-07-15 CY CY20131100597T patent/CY1114147T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
BRPI0816909A2 (pt) | 2015-03-17 |
ES2419255T3 (es) | 2013-08-20 |
PT2197881E (pt) | 2013-06-28 |
AU2008300616B2 (en) | 2013-02-14 |
ZA201001694B (en) | 2010-10-27 |
EP2197881B1 (en) | 2013-04-17 |
CA2698441A1 (en) | 2009-03-26 |
HK1142900A1 (en) | 2010-12-17 |
KR20100074157A (ko) | 2010-07-01 |
PL2197881T3 (pl) | 2013-09-30 |
KR101421774B1 (ko) | 2014-07-30 |
CA2698441C (en) | 2012-04-03 |
CN101801974A (zh) | 2010-08-11 |
DK2197881T3 (da) | 2013-06-24 |
US20110178291A1 (en) | 2011-07-21 |
JP2010539211A (ja) | 2010-12-16 |
US8450477B2 (en) | 2013-05-28 |
CN101801974B (zh) | 2013-08-28 |
CY1114147T1 (el) | 2016-07-27 |
EP2197881A1 (en) | 2010-06-23 |
US8877961B2 (en) | 2014-11-04 |
AU2008300616A1 (en) | 2009-03-26 |
US20130274503A1 (en) | 2013-10-17 |
WO2009037229A1 (en) | 2009-03-26 |
JP5551072B2 (ja) | 2014-07-16 |
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Legal Events
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FG | Grant or registration |