MX17107A - Procedimiento para la preparacion de tiazolo-(1,5)-benzodiazepinas y producto obtenido - Google Patents

Procedimiento para la preparacion de tiazolo-(1,5)-benzodiazepinas y producto obtenido

Info

Publication number
MX17107A
MX17107A MX1710789A MX1710789A MX17107A MX 17107 A MX17107 A MX 17107A MX 1710789 A MX1710789 A MX 1710789A MX 1710789 A MX1710789 A MX 1710789A MX 17107 A MX17107 A MX 17107A
Authority
MX
Mexico
Prior art keywords
tiazolo
benzodiazepines
procedure
preparation
product obtained
Prior art date
Application number
MX1710789A
Other languages
English (en)
Inventor
Jiban Kumar Chakrabarti
Original Assignee
Lilly Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd
Publication of MX17107A publication Critical patent/MX17107A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
MX1710789A 1988-08-11 1989-08-08 Procedimiento para la preparacion de tiazolo-(1,5)-benzodiazepinas y producto obtenido MX17107A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB888819059A GB8819059D0 (en) 1988-08-11 1988-08-11 Benzodiazepine compounds & their use as pharmaceuticals

Publications (1)

Publication Number Publication Date
MX17107A true MX17107A (es) 1993-08-01

Family

ID=10641942

Family Applications (1)

Application Number Title Priority Date Filing Date
MX1710789A MX17107A (es) 1988-08-11 1989-08-08 Procedimiento para la preparacion de tiazolo-(1,5)-benzodiazepinas y producto obtenido

Country Status (22)

Country Link
US (2) US4977150A (es)
EP (1) EP0354781B1 (es)
JP (1) JP2779219B2 (es)
KR (1) KR0138527B1 (es)
CN (1) CN1025857C (es)
AR (1) AR246972A1 (es)
AT (1) ATE113600T1 (es)
AU (1) AU625067B2 (es)
CA (1) CA1318669C (es)
DE (1) DE68919154T2 (es)
DK (1) DK393489A (es)
ES (1) ES2062012T3 (es)
GB (1) GB8819059D0 (es)
HU (1) HU202239B (es)
IE (1) IE64598B1 (es)
IL (1) IL91246A (es)
MX (1) MX17107A (es)
NZ (1) NZ230251A (es)
PH (1) PH27010A (es)
PT (1) PT91401B (es)
RU (1) RU2002752C1 (es)
ZA (1) ZA896039B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE1004596A4 (fr) * 1990-09-26 1992-12-22 Therabel Res S A N V Derives de methylpiperazinoazepine, leur preparation et leur utilisation.
US5627178A (en) 1991-04-23 1997-05-06 Lilly Industries Limited 2-methyl-thieno-benzodiazepine
US5393752A (en) * 1992-05-26 1995-02-28 Therabel Research S.A./N.V. Methylpiperazinoazepine compounds, preparation and use thereof
US6034078A (en) * 1992-05-29 2000-03-07 Eli Lilly And Company Limited Thienobenzodiazepine compounds
US6617321B2 (en) * 1997-09-30 2003-09-09 Eli Lilly And Company 2-methyl-thieno-benzodiazepine formulation
DE60318030T2 (de) 2002-03-28 2008-04-10 Eli Lilly And Co., Indianapolis Piperazine-substituierte aryl-benzodiazepine und ihre verwendung als dopaminrezeptor-antagonisten zur behandlung von psychosen
PT1546134E (pt) * 2002-08-05 2007-08-10 Lilly Co Eli ''arilbenzodiazepinas substituídas com piperazina''
CA2536107A1 (en) * 2003-09-09 2005-03-24 Eli Lilly And Company Substituted piperazines of azepines, oxazepines, and thiazepines
EP1838716B1 (en) * 2005-01-05 2011-06-01 Eli Lilly And Company Olanzapine pamoate dihydrate

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH468400A (de) * 1965-12-23 1969-02-15 Sandoz Ag Verfahren zur Herstellung neuer Thieno(2,3-b)(1,5)benzothiazepin-4-on-Verbindungen
US3539573A (en) * 1967-03-22 1970-11-10 Jean Schmutz 11-basic substituted dibenzodiazepines and dibenzothiazepines
US3758479A (en) * 1967-03-22 1973-09-11 Sandoz Ag Nitro and sulphamoyl substituted dibenzodiazepines
GB1292410A (en) * 1970-05-13 1972-10-11 Yoshitomi Pharmaceutical Thienobenzothiazepine derivatives
CH554362A (de) * 1970-07-30 1974-09-30 Spofa Vereinigte Pharma Werke Verfahren zur herstellung von neuen estern tricyklischer piperazinoalkanole.
US3897446A (en) * 1973-09-04 1975-07-29 Upjohn Co 6-Phenylthiazolo{8 3,2-a{9 {8 1,4{9 benzodiazepin-1-(2H)-ones, and processes
SU629879A3 (ru) * 1974-11-26 1978-10-25 Лилли Индастриз Лимитед, (Фирма) Способ получени тиено(1,5) бензодиазепинов или их солей
US4115568A (en) * 1974-11-26 1978-09-19 Lilly Industries Limited Thieno[3,2-b]-[1,5]benzodiazepines
US3951981A (en) * 1975-02-24 1976-04-20 American Cyanamid Company Substituted benzodiazepines and method of use
US4404137A (en) * 1979-10-16 1983-09-13 Lilly Industries Limited Pyrazolo [3,4-b][1,5]benzodiazepine compounds
US4431589A (en) * 1980-12-11 1984-02-14 Lilly House Benzodiazepine compounds and their use as pharmaceuticals

Also Published As

Publication number Publication date
CA1318669C (en) 1993-06-01
IL91246A0 (en) 1990-03-19
JPH02104591A (ja) 1990-04-17
US4977150A (en) 1990-12-11
IE892576L (en) 1990-02-11
EP0354781B1 (en) 1994-11-02
PT91401B (pt) 1995-05-04
KR0138527B1 (ko) 1998-05-15
ATE113600T1 (de) 1994-11-15
EP0354781A3 (en) 1991-04-03
AR246972A1 (es) 1994-10-31
DE68919154T2 (de) 1995-03-09
HU202239B (en) 1991-02-28
IL91246A (en) 1994-01-25
JP2779219B2 (ja) 1998-07-23
CN1025857C (zh) 1994-09-07
RU2002752C1 (ru) 1993-11-15
IE64598B1 (en) 1995-08-23
AU3939989A (en) 1990-02-15
HUT53109A (en) 1990-09-28
PT91401A (pt) 1990-03-08
DK393489A (da) 1990-02-12
DE68919154D1 (de) 1994-12-08
PH27010A (en) 1993-02-01
ES2062012T3 (es) 1994-12-16
AU625067B2 (en) 1992-07-02
ZA896039B (en) 1991-04-24
EP0354781A2 (en) 1990-02-14
DK393489D0 (da) 1989-08-10
US5051516A (en) 1991-09-24
GB8819059D0 (en) 1988-09-14
CN1040798A (zh) 1990-03-28
NZ230251A (en) 1992-05-26
KR900003179A (ko) 1990-03-23

Similar Documents

Publication Publication Date Title
MX13836A (es) Procedimiento para producir derivados de 5'-deoxi-5-fluorocitidina y producto obtenido,
MX12168A (es) Procedimiento para la preparacion de derivados de benzopirano y producto obtenido
MX22877A (es) Procedimiento para la preparacion de pirimidas, producto obtenido y composicion farmaceutica que lo incluye
MX5220A (es) Procedimiento para la produccion de derivados de dicloroanilina y producto obtenido
MX17169A (es) Proceso para la preparacion de derivados de triazol y producto obtenido
MX14331A (es) Procedimiento para preparar derivados de adenosinaprocedimiento para preparar derivados de adenosina y producto obtenido y producto obtenido
MX174238B (es) Procedimiento para la preparacion de derivados de pirimidina y producto obtenido
ES553096A0 (es) Procedimiento para la preparacion de un producto alimenticio gelificado
MX2954A (es) Procedimiento para preparar isoxazoles y producto obtenido.
MX14910A (es) 2',3' -dideoxi-2',2'-difluoronucleosidos y procedimiento para su preparacion.
MX14411A (es) Procedimiento para producir 1,2-dioxetanos e intermediarios de los mismos y producto obtenido.
BR8903877A (pt) Processo para preparacao de diorganopolissiloxano linear,produto obtido e utilizacao deste produto
MX14310A (es) Procedimiento para la preparacion de nuevos agentes antiarritmicos, producto obtenido y preparacion farmaceutica que lo incluye.
MX9260A (es) Procedimiento de preparacion de nuevos derivados de 1-bencenosulfonil-2-oxo-5-alcoxipirrolidina y producto obtenido
MX11493A (es) Procedimiento para la preparacion de derivados de pirimidina y producto obtenido.
FI894546A (fi) Menetelmä uusien 2'-halogeenimetylideeni-, 2'-etenylideeni- ja 2'-etynyyliadenosiinijohdannaisten valmistamiseksi
MX17107A (es) Procedimiento para la preparacion de tiazolo-(1,5)-benzodiazepinas y producto obtenido
MX21871A (es) Procedimiento para la preparacion de oxadiazolil fenoxialquilisoxazoles y compuestos resultantes
MX9173A (es) Procedimiento para la preparacion de compuestos anionicos ciclo-diilidicos y producto obtenido.
MX12881A (es) Procedimiento para la preparacion de acidos 4-oxo-3-quinolincarboxilicos y producto obtenido
NO903347D0 (no) Fremgangsmaate for fremstilling av 14,17alfa-ethano- og ethanooestratriener.
MX14990A (es) Procedimiento para la preparacion de derivados de estilbeno y producto obtenido.
MX10085A (es) Procedimiento para la preparacion de 4-arilcarbonil-1-((4-morfolinil)-alquilo-inferior)-1h-indoles y producto obtenido.
MX14871A (es) Procedimiento para la preparacion de pirroles substituidos y producto obtenido.
MX9517A (es) Procedimiento para la preparacion de cetonas triciclicas y producto obtenido