MX17107A - Procedimiento para la preparacion de tiazolo-(1,5)-benzodiazepinas y producto obtenido - Google Patents
Procedimiento para la preparacion de tiazolo-(1,5)-benzodiazepinas y producto obtenidoInfo
- Publication number
- MX17107A MX17107A MX1710789A MX1710789A MX17107A MX 17107 A MX17107 A MX 17107A MX 1710789 A MX1710789 A MX 1710789A MX 1710789 A MX1710789 A MX 1710789A MX 17107 A MX17107 A MX 17107A
- Authority
- MX
- Mexico
- Prior art keywords
- tiazolo
- benzodiazepines
- procedure
- preparation
- product obtained
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Neurology (AREA)
- Public Health (AREA)
- Psychiatry (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB888819059A GB8819059D0 (en) | 1988-08-11 | 1988-08-11 | Benzodiazepine compounds & their use as pharmaceuticals |
Publications (1)
Publication Number | Publication Date |
---|---|
MX17107A true MX17107A (es) | 1993-08-01 |
Family
ID=10641942
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX1710789A MX17107A (es) | 1988-08-11 | 1989-08-08 | Procedimiento para la preparacion de tiazolo-(1,5)-benzodiazepinas y producto obtenido |
Country Status (22)
Country | Link |
---|---|
US (2) | US4977150A (es) |
EP (1) | EP0354781B1 (es) |
JP (1) | JP2779219B2 (es) |
KR (1) | KR0138527B1 (es) |
CN (1) | CN1025857C (es) |
AR (1) | AR246972A1 (es) |
AT (1) | ATE113600T1 (es) |
AU (1) | AU625067B2 (es) |
CA (1) | CA1318669C (es) |
DE (1) | DE68919154T2 (es) |
DK (1) | DK393489A (es) |
ES (1) | ES2062012T3 (es) |
GB (1) | GB8819059D0 (es) |
HU (1) | HU202239B (es) |
IE (1) | IE64598B1 (es) |
IL (1) | IL91246A (es) |
MX (1) | MX17107A (es) |
NZ (1) | NZ230251A (es) |
PH (1) | PH27010A (es) |
PT (1) | PT91401B (es) |
RU (1) | RU2002752C1 (es) |
ZA (1) | ZA896039B (es) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE1004596A4 (fr) * | 1990-09-26 | 1992-12-22 | Therabel Res S A N V | Derives de methylpiperazinoazepine, leur preparation et leur utilisation. |
US5627178A (en) | 1991-04-23 | 1997-05-06 | Lilly Industries Limited | 2-methyl-thieno-benzodiazepine |
US5393752A (en) * | 1992-05-26 | 1995-02-28 | Therabel Research S.A./N.V. | Methylpiperazinoazepine compounds, preparation and use thereof |
US6034078A (en) * | 1992-05-29 | 2000-03-07 | Eli Lilly And Company Limited | Thienobenzodiazepine compounds |
US6617321B2 (en) * | 1997-09-30 | 2003-09-09 | Eli Lilly And Company | 2-methyl-thieno-benzodiazepine formulation |
DE60318030T2 (de) | 2002-03-28 | 2008-04-10 | Eli Lilly And Co., Indianapolis | Piperazine-substituierte aryl-benzodiazepine und ihre verwendung als dopaminrezeptor-antagonisten zur behandlung von psychosen |
PT1546134E (pt) * | 2002-08-05 | 2007-08-10 | Lilly Co Eli | ''arilbenzodiazepinas substituídas com piperazina'' |
CA2536107A1 (en) * | 2003-09-09 | 2005-03-24 | Eli Lilly And Company | Substituted piperazines of azepines, oxazepines, and thiazepines |
EP1838716B1 (en) * | 2005-01-05 | 2011-06-01 | Eli Lilly And Company | Olanzapine pamoate dihydrate |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH468400A (de) * | 1965-12-23 | 1969-02-15 | Sandoz Ag | Verfahren zur Herstellung neuer Thieno(2,3-b)(1,5)benzothiazepin-4-on-Verbindungen |
US3539573A (en) * | 1967-03-22 | 1970-11-10 | Jean Schmutz | 11-basic substituted dibenzodiazepines and dibenzothiazepines |
US3758479A (en) * | 1967-03-22 | 1973-09-11 | Sandoz Ag | Nitro and sulphamoyl substituted dibenzodiazepines |
GB1292410A (en) * | 1970-05-13 | 1972-10-11 | Yoshitomi Pharmaceutical | Thienobenzothiazepine derivatives |
CH554362A (de) * | 1970-07-30 | 1974-09-30 | Spofa Vereinigte Pharma Werke | Verfahren zur herstellung von neuen estern tricyklischer piperazinoalkanole. |
US3897446A (en) * | 1973-09-04 | 1975-07-29 | Upjohn Co | 6-Phenylthiazolo{8 3,2-a{9 {8 1,4{9 benzodiazepin-1-(2H)-ones, and processes |
SU629879A3 (ru) * | 1974-11-26 | 1978-10-25 | Лилли Индастриз Лимитед, (Фирма) | Способ получени тиено(1,5) бензодиазепинов или их солей |
US4115568A (en) * | 1974-11-26 | 1978-09-19 | Lilly Industries Limited | Thieno[3,2-b]-[1,5]benzodiazepines |
US3951981A (en) * | 1975-02-24 | 1976-04-20 | American Cyanamid Company | Substituted benzodiazepines and method of use |
US4404137A (en) * | 1979-10-16 | 1983-09-13 | Lilly Industries Limited | Pyrazolo [3,4-b][1,5]benzodiazepine compounds |
US4431589A (en) * | 1980-12-11 | 1984-02-14 | Lilly House | Benzodiazepine compounds and their use as pharmaceuticals |
-
1988
- 1988-08-11 GB GB888819059A patent/GB8819059D0/en active Pending
-
1989
- 1989-08-04 US US07/390,029 patent/US4977150A/en not_active Expired - Lifetime
- 1989-08-07 PH PH39061A patent/PH27010A/en unknown
- 1989-08-07 AU AU39399/89A patent/AU625067B2/en not_active Ceased
- 1989-08-08 CA CA000607760A patent/CA1318669C/en not_active Expired - Fee Related
- 1989-08-08 NZ NZ230251A patent/NZ230251A/en unknown
- 1989-08-08 MX MX1710789A patent/MX17107A/es unknown
- 1989-08-08 PT PT91401A patent/PT91401B/pt active IP Right Grant
- 1989-08-08 IL IL9124689A patent/IL91246A/en not_active IP Right Cessation
- 1989-08-08 ZA ZA896039A patent/ZA896039B/xx unknown
- 1989-08-09 ES ES89308099T patent/ES2062012T3/es not_active Expired - Lifetime
- 1989-08-09 AT AT89308099T patent/ATE113600T1/de not_active IP Right Cessation
- 1989-08-09 EP EP89308099A patent/EP0354781B1/en not_active Expired - Lifetime
- 1989-08-09 DE DE68919154T patent/DE68919154T2/de not_active Expired - Fee Related
- 1989-08-10 DK DK393489A patent/DK393489A/da not_active Application Discontinuation
- 1989-08-10 AR AR89314625A patent/AR246972A1/es active
- 1989-08-10 CN CN89105557A patent/CN1025857C/zh not_active Expired - Fee Related
- 1989-08-10 JP JP1207770A patent/JP2779219B2/ja not_active Expired - Lifetime
- 1989-08-10 IE IE257689A patent/IE64598B1/en not_active IP Right Cessation
- 1989-08-10 HU HU894101A patent/HU202239B/hu not_active IP Right Cessation
- 1989-08-10 KR KR1019890011365A patent/KR0138527B1/ko not_active IP Right Cessation
- 1989-08-10 RU SU894614830A patent/RU2002752C1/ru active
-
1990
- 1990-08-02 US US07/562,055 patent/US5051516A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
CA1318669C (en) | 1993-06-01 |
IL91246A0 (en) | 1990-03-19 |
JPH02104591A (ja) | 1990-04-17 |
US4977150A (en) | 1990-12-11 |
IE892576L (en) | 1990-02-11 |
EP0354781B1 (en) | 1994-11-02 |
PT91401B (pt) | 1995-05-04 |
KR0138527B1 (ko) | 1998-05-15 |
ATE113600T1 (de) | 1994-11-15 |
EP0354781A3 (en) | 1991-04-03 |
AR246972A1 (es) | 1994-10-31 |
DE68919154T2 (de) | 1995-03-09 |
HU202239B (en) | 1991-02-28 |
IL91246A (en) | 1994-01-25 |
JP2779219B2 (ja) | 1998-07-23 |
CN1025857C (zh) | 1994-09-07 |
RU2002752C1 (ru) | 1993-11-15 |
IE64598B1 (en) | 1995-08-23 |
AU3939989A (en) | 1990-02-15 |
HUT53109A (en) | 1990-09-28 |
PT91401A (pt) | 1990-03-08 |
DK393489A (da) | 1990-02-12 |
DE68919154D1 (de) | 1994-12-08 |
PH27010A (en) | 1993-02-01 |
ES2062012T3 (es) | 1994-12-16 |
AU625067B2 (en) | 1992-07-02 |
ZA896039B (en) | 1991-04-24 |
EP0354781A2 (en) | 1990-02-14 |
DK393489D0 (da) | 1989-08-10 |
US5051516A (en) | 1991-09-24 |
GB8819059D0 (en) | 1988-09-14 |
CN1040798A (zh) | 1990-03-28 |
NZ230251A (en) | 1992-05-26 |
KR900003179A (ko) | 1990-03-23 |
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