ME00293B - Sastavi estrogen-ciklodekstrin kompleksa - Google Patents

Sastavi estrogen-ciklodekstrin kompleksa

Info

Publication number
ME00293B
ME00293B MEP-2008-381A MEP2008381A ME00293B ME 00293 B ME00293 B ME 00293B ME P2008381 A MEP2008381 A ME P2008381A ME 00293 B ME00293 B ME 00293B
Authority
ME
Montenegro
Prior art keywords
estrogen
cyclodextrin
composition
compositions
ethinyl estradiol
Prior art date
Application number
MEP-2008-381A
Other languages
English (en)
Inventor
Thomas Backensfeld
Wolfgang Heil
Ralph Lipp
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP00610135A external-priority patent/EP1216713A1/en
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of ME00293B publication Critical patent/ME00293B/me

Links

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Obezbeđeni su farmaceutski sastavi koji obuhvataju niske doze osetljivih kompleksa između estrogena i ciklodekstrina sa poboljšanom stabilnošću. U specifičnoj realizaciji sastav obuhvata kompleks između etinil estradiola i ?-ciklodekstrin u granulatnom preparatu a u još jednoj realizaciji sastav obuhvata limitiranu količinu polivinilpirolidona pošto je za ovaj inertni punilac pronađeno da degradira etinil estradiol. Dalje, obezbeđen je postupak za poboljšanje stabilnosti estrogena u sastavu i za proizvodnju takvog stabilnog sastava. U osnovi, granulatni preparat je proizveden uz pažljivu kontrolu relativne vlažnosti.
MEP-2008-381A 2000-12-20 2001-12-20 Sastavi estrogen-ciklodekstrin kompleksa ME00293B (me)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00610135A EP1216713A1 (en) 2000-12-20 2000-12-20 Compositions of estrogen-cyclodextrin complexes
PCT/IB2001/002605 WO2002049675A1 (en) 2000-12-20 2001-12-20 Compositions of estrogen-cyclodextrin complexes

Publications (1)

Publication Number Publication Date
ME00293B true ME00293B (me) 2011-05-10

Family

ID=37516219

Family Applications (1)

Application Number Title Priority Date Filing Date
MEP-2008-381A ME00293B (me) 2000-12-20 2001-12-20 Sastavi estrogen-ciklodekstrin kompleksa

Country Status (7)

Country Link
CN (1) CN101116666B (me)
AR (1) AR032205A1 (me)
ME (1) ME00293B (me)
PE (1) PE20020709A1 (me)
UA (1) UA77626C2 (me)
UY (1) UY27088A1 (me)
ZA (1) ZA200305532B (me)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102512688A (zh) * 2011-12-29 2012-06-27 上海新华联制药有限公司 尼尔雌醇-β-环糊精包合物及制剂和制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4727064A (en) * 1984-04-25 1988-02-23 The United States Of America As Represented By The Department Of Health And Human Services Pharmaceutical preparations containing cyclodextrin derivatives
NL8801670A (nl) * 1988-07-01 1990-02-01 Walter Adrianus Josephus Johan Farmaceutisch preparaat.
US5324718A (en) * 1992-07-14 1994-06-28 Thorsteinn Loftsson Cyclodextrin/drug complexation
DE19848303A1 (de) * 1998-10-14 2000-04-20 Schering Ag Kombination aus Gestagenen und Zuckern

Also Published As

Publication number Publication date
CN101116666A (zh) 2008-02-06
ZA200305532B (en) 2006-06-28
PE20020709A1 (es) 2002-08-23
UY27088A1 (es) 2002-07-31
AR032205A1 (es) 2003-10-29
UA77626C2 (en) 2006-12-15
CN101116666B (zh) 2014-01-08

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