MD3771F1 - Inhibitori ai enzimei 17Beta-HSD, stimulatoare a multiplicarii celulelor cancerului prostatei - Google Patents

Inhibitori ai enzimei 17Beta-HSD, stimulatoare a multiplicarii celulelor cancerului prostatei Download PDF

Info

Publication number
MD3771F1
MD3771F1 MDA20080118A MD20080118A MD3771F1 MD 3771 F1 MD3771 F1 MD 3771F1 MD A20080118 A MDA20080118 A MD A20080118A MD 20080118 A MD20080118 A MD 20080118A MD 3771 F1 MD3771 F1 MD 3771F1
Authority
MD
Moldova
Prior art keywords
prostate cancer
inhibitors
17beta
stimulator
cancer cell
Prior art date
Application number
MDA20080118A
Other languages
English (en)
Other versions
MD3771G2 (ro
Inventor
Aurelian Gulea
Donald Poirier
Jenny Roy
Victor Tapcov
Original Assignee
Universitatea De Stat Din Moldova
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Universitatea De Stat Din Moldova filed Critical Universitatea De Stat Din Moldova
Priority to MDA20080118A priority Critical patent/MD3771G2/ro
Publication of MD3771F1 publication Critical patent/MD3771F1/ro
Publication of MD3771G2 publication Critical patent/MD3771G2/ro

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Inventia se refera la chimie, si anume la compusii organici din clasa tiosemicarbazonelor, care pot fi utilizati pentru tratamentul cancerului prostatei. Esenta inventiei consta in utilizarea 4-feniltiosemicarbazonelor aldehidelor salicilice si 2-hidroxi-1-naftoice in calitate de inhibitori ai enzimei 17b-HSD (hidroxisteroid dehidrogenaza), stimulatoare a multiplicarii celulelor cancerului prostatei.
MDA20080118A 2008-04-30 2008-04-30 Inhibitori ai enzimei 17β-HSD, stimulatoare a multiplicării celulelor cancerului prostatei MD3771G2 (ro)

Priority Applications (1)

Application Number Priority Date Filing Date Title
MDA20080118A MD3771G2 (ro) 2008-04-30 2008-04-30 Inhibitori ai enzimei 17β-HSD, stimulatoare a multiplicării celulelor cancerului prostatei

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
MDA20080118A MD3771G2 (ro) 2008-04-30 2008-04-30 Inhibitori ai enzimei 17β-HSD, stimulatoare a multiplicării celulelor cancerului prostatei

Publications (2)

Publication Number Publication Date
MD3771F1 true MD3771F1 (ro) 2008-12-31
MD3771G2 MD3771G2 (ro) 2009-07-31

Family

ID=40255075

Family Applications (1)

Application Number Title Priority Date Filing Date
MDA20080118A MD3771G2 (ro) 2008-04-30 2008-04-30 Inhibitori ai enzimei 17β-HSD, stimulatoare a multiplicării celulelor cancerului prostatei

Country Status (1)

Country Link
MD (1) MD3771G2 (ro)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MD3996C2 (ro) * 2009-05-25 2010-07-31 Государственный Университет Молд0 Percloraţi de 5-R-saliciliden-4-feniltiosemicarbazonato(1-)-aquacupru(II) ce posedă proprietăţi de inhibitori ai activităţii enzimei 17 b-HSD (tipul 1)
MD4025C2 (ro) * 2009-08-25 2010-10-31 Владимир КАРАУШ Remediu pentru tratamentul prostatitei şi hiperplaziei prostatei
MD4126C1 (ro) * 2010-11-15 2012-04-30 Государственный Университет Молд0 N,N'-[4,4'-(perfluoro-1,4-fenilendioxi)-bis(4,1-fenilen)]-bis[2-(piridin-2-ilmetilen)hidrazincarbotioamidă] şi utilizarea ei în calitate de inhibitor al proliferării celulelor LNCaP ale cancerului prostatei
MD4132C1 (ro) * 2010-12-13 2012-05-31 Государственный Университет Молд0 Di(µ-S)-bis{cloro-[fenil(piridin-2-il)metanon-tiosemicarbazonato(1-)]cupru} care manifestă proprietatea de inhibare a proliferării celulelor T-47D ale cancerului mamar
MD4349C1 (ro) * 2014-06-23 2015-12-31 Государственный Университет Молд0 Compusul N-(3-metoxifenil)-2-(piridin-2-ilmetilen)-hidrazincarbotioamidă - inhibitor al proliferării celulelor MeW-164 ale melanomului uman

Also Published As

Publication number Publication date
MD3771G2 (ro) 2009-07-31

Similar Documents

Publication Publication Date Title
EA201100125A1 (ru) Производные пирролопиридинилпиримидин-2-иламина
MY160399A (en) Compounds, compositions, and methods for preventing metastasis of cancer cells
CY1120664T1 (el) Χρησεις και συνθεσεις για αντιμετωπιση διαπυητικης ιδρωταδενιτιδας (δι)
ATE553198T1 (de) Behandlung von krebs durch die kombinierte hemmung der proteasom- und telomeraseaktivitäten
EA201491574A1 (ru) Применение car, основанных на icos, для усиления противоопухолевой активности и длительного сохранения car
MX2010008040A (es) Derivados de pirimidina 5-fluoro como fungicidas.
MX2010009765A (es) Moleculas pequeñas que contienen boro como agentes anti-inflamatorios.
MX364002B (es) Compuestos y composiciones activadoras de enzima.
CL2009000687A1 (es) Compuestos derivados de heterociclos nitrogenados de imidazol, inhibidores de la actividad de cinasa raf; composicion farmaceutica; utiles para el tratamiento del cancer, tal como carcinoma de pulmon, pancreatico, de prostata, tiroides, entre otras.
CO7400882A2 (es) Modulación de la expresión de receptores androgénicos
MX366318B (es) Derivados de aminas heterocíclicas que inhiben la transducción de señal mediana por cinasa asociada con el receptor de interleucina-1.
WO2012037155A3 (en) Tyrosine kinase inhibitors
SG195086A1 (en) Compounds containing hydrido-tricyano-borate anions
BR112012021296A2 (pt) imunoconjugados e anticorpos de receptor de folato 1 e usos dos mesmos.
MX391154B (es) Compuestos con actividad anticancer
EA201000004A1 (ru) Производные 6-(пирролопиридинил)пиримидин-2-иламина и их применение для лечения злокачественного новообразования и спида
EA201300442A1 (ru) ПИРРОЛИДИНОНЫ В КАЧЕСТВЕ ИНГИБИТОРОВ MetAP-2
TR201910526T4 (tr) N-sübstitüe sülfoniloksibenzilaminler ve ilgili bileşiklerin kozmetik kullanımı.
EA201492210A1 (ru) Соединения, ингибирующие активность катехол-o-метилтрансферазы
FR2939316B1 (fr) Utilisation cosmetique d'activateurs de l'autophagie des cellules cutanees.
TR201903981T4 (tr) Kanser tedavisi için bileşikler.
WO2013059582A3 (en) Small molecule inhibitors of histone deacteylases
EA201100424A1 (ru) Новые ингибиторы
WO2009114703A3 (en) Combination therapy for the treatment of cancer
MD3771F1 (ro) Inhibitori ai enzimei 17Beta-HSD, stimulatoare a multiplicarii celulelor cancerului prostatei

Legal Events

Date Code Title Description
FG4A Patent for invention issued
KA4A Patent for invention lapsed due to non-payment of fees (with right of restoration)
MM4A Patent for invention definitely lapsed due to non-payment of fees