MC1146A1 - Derives peptidiques et procede pour leur preparation - Google Patents

Derives peptidiques et procede pour leur preparation

Info

Publication number
MC1146A1
MC1146A1 MC771242A MC1242A MC1146A1 MC 1146 A1 MC1146 A1 MC 1146A1 MC 771242 A MC771242 A MC 771242A MC 1242 A MC1242 A MC 1242A MC 1146 A1 MC1146 A1 MC 1146A1
Authority
MC
Monaco
Prior art keywords
alanyl
group
general formula
compound
acid
Prior art date
Application number
MC771242A
Other languages
English (en)
French (fr)
Inventor
C Hassall
F Atherton
P Ringrose
M Hall
R Lambert
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MC1146A1 publication Critical patent/MC1146A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/30Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
    • C07F9/301Acyclic saturated acids which can have further substituents on alkyl
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3808Acyclic saturated acids which can have further substituents on alkyl
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06191Dipeptides containing heteroatoms different from O, S, or N
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0827Tripeptides containing heteroatoms different from O, S, or N
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10Tetrapeptides
    • C07K5/1027Tetrapeptides containing heteroatoms different from O, S, or N
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
MC771242A 1976-05-14 1977-05-13 Derives peptidiques et procede pour leur preparation MC1146A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB20014/76A GB1577232A (en) 1976-05-14 1976-05-14 Peptide derivatives of phosphonic and phosphinic acids

Publications (1)

Publication Number Publication Date
MC1146A1 true MC1146A1 (fr) 1978-01-30

Family

ID=10138919

Family Applications (1)

Application Number Title Priority Date Filing Date
MC771242A MC1146A1 (fr) 1976-05-14 1977-05-13 Derives peptidiques et procede pour leur preparation

Country Status (23)

Country Link
JP (1) JPS52139023A (enExample)
AT (1) AT355740B (enExample)
AU (1) AU511452B2 (enExample)
BE (1) BE854591A (enExample)
CA (1) CA1090785A (enExample)
DE (1) DE2721760A1 (enExample)
DK (1) DK209877A (enExample)
ES (1) ES458748A1 (enExample)
FI (1) FI771518A7 (enExample)
FR (1) FR2351124A1 (enExample)
GB (1) GB1577232A (enExample)
GR (1) GR73010B (enExample)
IL (1) IL52040A (enExample)
IT (1) IT1075484B (enExample)
LU (1) LU77319A1 (enExample)
MC (1) MC1146A1 (enExample)
NL (1) NL7704370A (enExample)
NO (1) NO771717L (enExample)
NZ (1) NZ184047A (enExample)
PH (1) PH14715A (enExample)
PT (1) PT66544B (enExample)
SE (1) SE7705628L (enExample)
ZA (1) ZA772732B (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0002039A1 (en) * 1977-11-19 1979-05-30 Ciba-Geigy Ag Phosphonous acid derivatives, processes for their preparation and their use in combating microorganisms
EP0010067B1 (en) * 1978-10-05 1983-08-31 Ciba-Geigy Ag Process for influencing plant growth
EP0103867B1 (en) * 1982-09-17 1986-12-17 Kyowa Hakko Kogyo Co., Ltd. Phosphorus-containing peptide derivative

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS51639B1 (enExample) * 1971-07-28 1976-01-09
IL48835A (en) * 1975-01-27 1979-05-31 Sparamedica Ag Amino acyl and peptidyl derivatives of phophonic acids, their preparation and pharmaceutical compositions containingthem

Also Published As

Publication number Publication date
LU77319A1 (enExample) 1978-06-26
PT66544B (en) 1979-04-12
ZA772732B (en) 1978-04-26
NZ184047A (en) 1980-04-28
DE2721760A1 (de) 1977-12-01
IL52040A0 (en) 1977-07-31
FR2351124A1 (fr) 1977-12-09
AT355740B (de) 1980-03-25
FI771518A7 (enExample) 1977-11-15
FR2351124B1 (enExample) 1981-02-13
IL52040A (en) 1979-11-30
NL7704370A (nl) 1977-11-16
ATA345877A (de) 1979-08-15
BE854591A (fr) 1977-11-14
SE7705628L (sv) 1977-11-15
AU2500877A (en) 1978-11-16
PT66544A (en) 1977-06-01
DK209877A (da) 1977-11-15
CA1090785A (en) 1980-12-02
IT1075484B (it) 1985-04-22
GR73010B (enExample) 1984-01-24
PH14715A (en) 1981-11-13
ES458748A1 (es) 1978-03-01
GB1577232A (en) 1980-10-22
AU511452B2 (en) 1980-08-21
JPS52139023A (en) 1977-11-19
NO771717L (no) 1977-11-15

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Legal Events

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