MA55593A - Cycles pyridine contenant des dérivés servant d'inhibiteurs de malt1 - Google Patents

Cycles pyridine contenant des dérivés servant d'inhibiteurs de malt1

Info

Publication number
MA55593A
MA55593A MA055593A MA55593A MA55593A MA 55593 A MA55593 A MA 55593A MA 055593 A MA055593 A MA 055593A MA 55593 A MA55593 A MA 55593A MA 55593 A MA55593 A MA 55593A
Authority
MA
Morocco
Prior art keywords
containing derivatives
cycles containing
derivatives serving
malt1 inhibitors
pyridine
Prior art date
Application number
MA055593A
Other languages
English (en)
Inventor
Didier Jean-Claude Berthelot
Gaston Stanislas M Diels
Tianbao Lu
Johannes Wilhelmus J Thuring
Berthold Wroblowski
Tongfei Wu
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of MA55593A publication Critical patent/MA55593A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14Ortho-condensed systems
MA055593A 2019-04-11 2020-04-10 Cycles pyridine contenant des dérivés servant d'inhibiteurs de malt1 MA55593A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201962832608P 2019-04-11 2019-04-11
EP19178959 2019-06-07

Publications (1)

Publication Number Publication Date
MA55593A true MA55593A (fr) 2022-02-16

Family

ID=70224393

Family Applications (1)

Application Number Title Priority Date Filing Date
MA055593A MA55593A (fr) 2019-04-11 2020-04-10 Cycles pyridine contenant des dérivés servant d'inhibiteurs de malt1

Country Status (11)

Country Link
US (1) US20220162187A1 (fr)
EP (1) EP3953345B1 (fr)
JP (1) JP2022528919A (fr)
KR (1) KR20210151880A (fr)
CN (1) CN113677674A (fr)
AU (1) AU2020272156A1 (fr)
CA (1) CA3131856A1 (fr)
ES (1) ES2949871T3 (fr)
MA (1) MA55593A (fr)
MX (1) MX2021012417A (fr)
WO (1) WO2020208222A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022101676A1 (fr) * 2020-11-12 2022-05-19 Monopteros Therapeutics,Inc. Matériaux et procédés de traitement du cancer

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014033447A2 (fr) * 2012-08-29 2014-03-06 Respivert Limited Inhibiteurs de kinase
LT3149001T (lt) 2014-05-28 2019-08-12 Novartis Ag Naujieji pirazolo pirimidino dariniai ir jų panaudojimas kaip malt1 inhibitorių
MD3371190T2 (ro) * 2015-11-06 2022-09-30 Incyte Corp Compuși heterociclici ca inhibitori PI3K-gamma
BR112018009511A2 (pt) * 2015-11-13 2018-11-06 Novartis Ag derivados de pirazolo pirimidina
CN107021963A (zh) * 2016-01-29 2017-08-08 北京诺诚健华医药科技有限公司 吡唑稠环类衍生物、其制备方法及其在治疗癌症、炎症和免疫性疾病上的应用
AU2017302182B2 (en) 2016-07-29 2021-11-04 Lupin Limited Substituted thiazolo-pyridine compounds as MALT1 inhibitors
TWI795381B (zh) 2016-12-21 2023-03-11 比利時商健生藥品公司 作為malt1抑制劑之吡唑衍生物
EP3592731A4 (fr) * 2017-03-08 2020-10-07 Cornell University Inhibiteurs de malt1 et leurs utilisations
WO2018226150A1 (fr) * 2017-06-05 2018-12-13 Medivir Aktiebolag Pyrazolopyrimidine utilisés en tant qu'inhibiteurs de malt-1
CN112585128B (zh) 2018-06-18 2023-02-21 詹森药业有限公司 作为malt1抑制剂的吡唑衍生物
US10888550B2 (en) 2018-06-18 2021-01-12 Janssen Pharmaceutica Nv Pyrazole derivatives as MALT1 inhibitors

Also Published As

Publication number Publication date
KR20210151880A (ko) 2021-12-14
US20220162187A1 (en) 2022-05-26
AU2020272156A1 (en) 2021-10-14
EP3953345B1 (fr) 2023-04-05
EP3953345A1 (fr) 2022-02-16
JP2022528919A (ja) 2022-06-16
MX2021012417A (es) 2021-11-12
CN113677674A (zh) 2021-11-19
ES2949871T3 (es) 2023-10-03
CA3131856A1 (fr) 2020-10-15
WO2020208222A1 (fr) 2020-10-15

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