MA55593A - Cycles pyridine contenant des dérivés servant d'inhibiteurs de malt1 - Google Patents
Cycles pyridine contenant des dérivés servant d'inhibiteurs de malt1Info
- Publication number
- MA55593A MA55593A MA055593A MA55593A MA55593A MA 55593 A MA55593 A MA 55593A MA 055593 A MA055593 A MA 055593A MA 55593 A MA55593 A MA 55593A MA 55593 A MA55593 A MA 55593A
- Authority
- MA
- Morocco
- Prior art keywords
- containing derivatives
- cycles containing
- derivatives serving
- malt1 inhibitors
- pyridine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201962832608P | 2019-04-11 | 2019-04-11 | |
EP19178959 | 2019-06-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
MA55593A true MA55593A (fr) | 2022-02-16 |
Family
ID=70224393
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA055593A MA55593A (fr) | 2019-04-11 | 2020-04-10 | Cycles pyridine contenant des dérivés servant d'inhibiteurs de malt1 |
Country Status (11)
Country | Link |
---|---|
US (1) | US20220162187A1 (fr) |
EP (1) | EP3953345B1 (fr) |
JP (1) | JP2022528919A (fr) |
KR (1) | KR20210151880A (fr) |
CN (1) | CN113677674A (fr) |
AU (1) | AU2020272156A1 (fr) |
CA (1) | CA3131856A1 (fr) |
ES (1) | ES2949871T3 (fr) |
MA (1) | MA55593A (fr) |
MX (1) | MX2021012417A (fr) |
WO (1) | WO2020208222A1 (fr) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2022101676A1 (fr) * | 2020-11-12 | 2022-05-19 | Monopteros Therapeutics,Inc. | Matériaux et procédés de traitement du cancer |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2014033447A2 (fr) * | 2012-08-29 | 2014-03-06 | Respivert Limited | Inhibiteurs de kinase |
LT3149001T (lt) | 2014-05-28 | 2019-08-12 | Novartis Ag | Naujieji pirazolo pirimidino dariniai ir jų panaudojimas kaip malt1 inhibitorių |
MD3371190T2 (ro) * | 2015-11-06 | 2022-09-30 | Incyte Corp | Compuși heterociclici ca inhibitori PI3K-gamma |
BR112018009511A2 (pt) * | 2015-11-13 | 2018-11-06 | Novartis Ag | derivados de pirazolo pirimidina |
CN107021963A (zh) * | 2016-01-29 | 2017-08-08 | 北京诺诚健华医药科技有限公司 | 吡唑稠环类衍生物、其制备方法及其在治疗癌症、炎症和免疫性疾病上的应用 |
AU2017302182B2 (en) | 2016-07-29 | 2021-11-04 | Lupin Limited | Substituted thiazolo-pyridine compounds as MALT1 inhibitors |
TWI795381B (zh) | 2016-12-21 | 2023-03-11 | 比利時商健生藥品公司 | 作為malt1抑制劑之吡唑衍生物 |
EP3592731A4 (fr) * | 2017-03-08 | 2020-10-07 | Cornell University | Inhibiteurs de malt1 et leurs utilisations |
WO2018226150A1 (fr) * | 2017-06-05 | 2018-12-13 | Medivir Aktiebolag | Pyrazolopyrimidine utilisés en tant qu'inhibiteurs de malt-1 |
CN112585128B (zh) | 2018-06-18 | 2023-02-21 | 詹森药业有限公司 | 作为malt1抑制剂的吡唑衍生物 |
US10888550B2 (en) | 2018-06-18 | 2021-01-12 | Janssen Pharmaceutica Nv | Pyrazole derivatives as MALT1 inhibitors |
-
2020
- 2020-04-10 KR KR1020217036345A patent/KR20210151880A/ko active Search and Examination
- 2020-04-10 MX MX2021012417A patent/MX2021012417A/es unknown
- 2020-04-10 EP EP20717667.8A patent/EP3953345B1/fr active Active
- 2020-04-10 MA MA055593A patent/MA55593A/fr unknown
- 2020-04-10 ES ES20717667T patent/ES2949871T3/es active Active
- 2020-04-10 JP JP2021559711A patent/JP2022528919A/ja active Pending
- 2020-04-10 US US17/602,885 patent/US20220162187A1/en active Pending
- 2020-04-10 CA CA3131856A patent/CA3131856A1/fr active Pending
- 2020-04-10 WO PCT/EP2020/060307 patent/WO2020208222A1/fr unknown
- 2020-04-10 AU AU2020272156A patent/AU2020272156A1/en active Pending
- 2020-04-10 CN CN202080028070.1A patent/CN113677674A/zh active Pending
Also Published As
Publication number | Publication date |
---|---|
KR20210151880A (ko) | 2021-12-14 |
US20220162187A1 (en) | 2022-05-26 |
AU2020272156A1 (en) | 2021-10-14 |
EP3953345B1 (fr) | 2023-04-05 |
EP3953345A1 (fr) | 2022-02-16 |
JP2022528919A (ja) | 2022-06-16 |
MX2021012417A (es) | 2021-11-12 |
CN113677674A (zh) | 2021-11-19 |
ES2949871T3 (es) | 2023-10-03 |
CA3131856A1 (fr) | 2020-10-15 |
WO2020208222A1 (fr) | 2020-10-15 |
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