MA49618A - Inhibiteurs de la mpo destinés à être utilisés en médecine - Google Patents

Inhibiteurs de la mpo destinés à être utilisés en médecine

Info

Publication number
MA49618A
MA49618A MA049618A MA49618A MA49618A MA 49618 A MA49618 A MA 49618A MA 049618 A MA049618 A MA 049618A MA 49618 A MA49618 A MA 49618A MA 49618 A MA49618 A MA 49618A
Authority
MA
Morocco
Prior art keywords
medicine
mpo inhibitors
mpo
inhibitors
Prior art date
Application number
MA049618A
Other languages
English (en)
Inventor
Hitesh Jayantilal Sanganee
Andrew Whittaker
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of MA49618A publication Critical patent/MA49618A/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Reproductive Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Epidemiology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
MA049618A 2017-07-17 2018-07-12 Inhibiteurs de la mpo destinés à être utilisés en médecine MA49618A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201762533448P 2017-07-17 2017-07-17

Publications (1)

Publication Number Publication Date
MA49618A true MA49618A (fr) 2020-05-27

Family

ID=62904484

Family Applications (1)

Application Number Title Priority Date Filing Date
MA049618A MA49618A (fr) 2017-07-17 2018-07-12 Inhibiteurs de la mpo destinés à être utilisés en médecine

Country Status (15)

Country Link
US (2) US11246870B2 (fr)
EP (1) EP3654983B1 (fr)
JP (1) JP7220193B2 (fr)
KR (1) KR20200029513A (fr)
CN (1) CN110891572B (fr)
AU (1) AU2018304508B2 (fr)
BR (1) BR112019026270A2 (fr)
CA (1) CA3068910A1 (fr)
EA (1) EA202090266A1 (fr)
ES (1) ES2963315T3 (fr)
IL (1) IL272043B (fr)
MA (1) MA49618A (fr)
SG (1) SG11202000086PA (fr)
WO (1) WO2019016074A1 (fr)
ZA (1) ZA202000904B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20200029513A (ko) 2017-07-17 2020-03-18 아스트라제네카 아베 의약에서의 사용을 위한 mpo 억제제
US20240067651A1 (en) * 2019-10-10 2024-02-29 Biohaven Therapeutics Ltd. Prodrugs of myeloperoxidase inhibitors
CN115403584B (zh) * 2021-05-26 2024-04-02 长春金赛药业有限责任公司 2-硫代-2,3-二氢嘧啶-4-酮衍生物、药物组合物及其制备方法和应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2362101A (en) 2000-05-12 2001-11-14 Astrazeneca Ab Treatment of chronic obstructive pulmonary disease
SE0201193D0 (sv) * 2002-04-19 2002-04-19 Astrazeneca Ab Novel use
MY140748A (en) 2004-12-06 2010-01-15 Astrazeneca Ab Novel pyrrolo [3,2-d] pyrimidin-4-one derivatives and their use in therapy
US20090081177A1 (en) 2005-07-05 2009-03-26 Fertility Technologies Pty Ltd Methods and compositions for improving pregnancy outcome
AR066936A1 (es) 2007-06-13 2009-09-23 Astrazeneca Ab 3 - (2r - tetrahidrofuril - metil) - 2 - tioxantina. composiciones farmaceuticas.
US20090054468A1 (en) 2007-08-23 2009-02-26 Astrazeneca Ab New Use 938
JP5757604B2 (ja) 2010-02-05 2015-07-29 ヒガシマル醤油株式会社 ミエロペルオキシダーゼ阻害剤
US9616063B2 (en) 2014-12-01 2017-04-11 Astrazeneca Ab 1-[2-(aminomethyl)benzyl]-2-thioxo-1,2,3,5-tetrahydro-4H-pyrrolo[3,2-d]pyrimidin-4-ones as inhibitors of myeloperoxidase
US11241406B2 (en) 2015-08-28 2022-02-08 Nature's Sunshine Products, Inc. Compositions and methods for acutley raising nitric oxide levels
KR20200029513A (ko) 2017-07-17 2020-03-18 아스트라제네카 아베 의약에서의 사용을 위한 mpo 억제제

Also Published As

Publication number Publication date
AU2018304508B2 (en) 2021-06-10
US11246870B2 (en) 2022-02-15
EP3654983B1 (fr) 2023-08-30
EP3654983A1 (fr) 2020-05-27
ES2963315T3 (es) 2024-03-26
AU2018304508A1 (en) 2020-02-27
IL272043B (en) 2022-09-01
ZA202000904B (en) 2023-04-26
US11738027B2 (en) 2023-08-29
IL272043A (en) 2020-03-31
US20220160715A1 (en) 2022-05-26
EA202090266A1 (ru) 2020-06-05
CA3068910A1 (fr) 2019-01-24
KR20200029513A (ko) 2020-03-18
CN110891572A (zh) 2020-03-17
WO2019016074A1 (fr) 2019-01-24
JP2020527137A (ja) 2020-09-03
SG11202000086PA (en) 2020-02-27
US20200206226A1 (en) 2020-07-02
NZ761505A (en) 2023-09-29
CN110891572B (zh) 2023-08-15
JP7220193B2 (ja) 2023-02-09
BR112019026270A2 (pt) 2020-06-30

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