MA30981B1 - Derives de sulfonyl-phenyl-2h-(1,2,4)oxadiazol-5-one, procedes de preparation associes et utilisation comme medicaments - Google Patents
Derives de sulfonyl-phenyl-2h-(1,2,4)oxadiazol-5-one, procedes de preparation associes et utilisation comme medicamentsInfo
- Publication number
- MA30981B1 MA30981B1 MA31971A MA31971A MA30981B1 MA 30981 B1 MA30981 B1 MA 30981B1 MA 31971 A MA31971 A MA 31971A MA 31971 A MA31971 A MA 31971A MA 30981 B1 MA30981 B1 MA 30981B1
- Authority
- MA
- Morocco
- Prior art keywords
- disorders
- oxadiazol
- sulfonyl
- phenyl
- derivatives
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4245—Oxadiazoles
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
- A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
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- A—HUMAN NECESSITIES
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- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
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- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Diabetes (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Hematology (AREA)
- Dermatology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Endocrinology (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Physical Education & Sports Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Immunology (AREA)
- Vascular Medicine (AREA)
- Oncology (AREA)
- Ophthalmology & Optometry (AREA)
- Communicable Diseases (AREA)
- Psychology (AREA)
- Emergency Medicine (AREA)
- Reproductive Health (AREA)
- Virology (AREA)
Abstract
L'INVENTION PORTE SUR DES SULFONYL-PHÉNYL-OXADIAZOLONES ET SUR LEURS SELS PHYSIOLOGIQUEMENT ACCEPTABLES ET DÉRIVÉS PHYSIOLOGIQUEMENT FONCTIONNELS MONTRANT UNE ACTIVITÉ AGONISTE DE PPARDELTA OU DE PPARDELTA ET PPARGAMMA. ON DÉCRIT DES COMPOSÉS REPRÉSENTÉS PAR LA FORMULE I, DANS LAQUELLE LES RADICAUX SONT TELS QUE DÉFINIS, ET LEURS SELS PHYSIOLOGIQUEMENT ACCEPTABLES ET DES PROCÉDÉS PERMETTANT DE LES PRÉPARER. LES COMPOSÉS SONT APPROPRIÉS POUR LE TRAITEMENT ET/OU LA PRÉVENTION DE TROUBLES DU MÉTABOLISME DES ACIDES GRAS ET DES TROUBLES DE L'UTILISATION DU GLUCOSE AINSI QUE DE TROUBLES DANS LESQUELS LA RÉSISTANCE À L'INSULINE EST MISE EN JEU ET LA DÉMYÉLINISATION ET AUTRES TROUBLES NEURODÉGÉNÉRATIFS DU SYSTÈME NERVEUX CENTRAL ET PÉRIPHÉRIQUE.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP06025880A EP1932843A1 (fr) | 2006-12-14 | 2006-12-14 | Dérivés de sulfonyl-phenyl-2H(1,2,4) oxadiazole-5-one, procédés de préparation de ceux-ci et leur usage sous forme de médicaments |
Publications (1)
Publication Number | Publication Date |
---|---|
MA30981B1 true MA30981B1 (fr) | 2009-12-01 |
Family
ID=37998695
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA31971A MA30981B1 (fr) | 2006-12-14 | 2009-06-10 | Derives de sulfonyl-phenyl-2h-(1,2,4)oxadiazol-5-one, procedes de preparation associes et utilisation comme medicaments |
Country Status (24)
Country | Link |
---|---|
US (1) | US8173674B2 (fr) |
EP (2) | EP1932843A1 (fr) |
JP (1) | JP2010512352A (fr) |
KR (1) | KR20090087922A (fr) |
CN (1) | CN101558064A (fr) |
AR (1) | AR064299A1 (fr) |
AU (1) | AU2007331805A1 (fr) |
BR (1) | BRPI0720416A2 (fr) |
CA (1) | CA2672347A1 (fr) |
CL (1) | CL2007003614A1 (fr) |
CO (1) | CO6210729A2 (fr) |
CR (1) | CR10778A (fr) |
EC (1) | ECSP099409A (fr) |
MA (1) | MA30981B1 (fr) |
MX (1) | MX2009005535A (fr) |
NO (1) | NO20092293L (fr) |
PE (1) | PE20081404A1 (fr) |
RU (1) | RU2009126745A (fr) |
SV (1) | SV2009003293A (fr) |
TN (1) | TN2009000242A1 (fr) |
TW (1) | TW200843749A (fr) |
UY (1) | UY30783A1 (fr) |
WO (1) | WO2008071311A1 (fr) |
ZA (1) | ZA200903160B (fr) |
Families Citing this family (33)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102056921A (zh) * | 2008-06-09 | 2011-05-11 | 赛诺菲-安万特 | 首基为噁二唑酮的增环化n-杂环磺酰胺、其制备方法及其作为药物的用途 |
US8716317B2 (en) * | 2008-06-09 | 2014-05-06 | Sanofi | Sulfonamides with heterocycle and oxadiazolone headgroup, processes for their preparation and their use as pharmaceuticals |
WO2011107494A1 (fr) | 2010-03-03 | 2011-09-09 | Sanofi | Nouveaux dérivés aromatiques de glycoside, médicaments contenants ces composés, et leur utilisation |
US8933024B2 (en) | 2010-06-18 | 2015-01-13 | Sanofi | Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases |
US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
WO2013037390A1 (fr) | 2011-09-12 | 2013-03-21 | Sanofi | Dérivés amides d'acide 6-(4-hydroxyphényl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylique en tant qu'inhibiteurs de kinase |
EP2760862B1 (fr) | 2011-09-27 | 2015-10-21 | Sanofi | Dérivés d'amide d'acide 6-(4-hydroxyphényl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylique utilisés comme inhibiteurs de kinase |
US8859774B2 (en) | 2012-05-25 | 2014-10-14 | Corcept Therapeutics, Inc. | Heteroaryl-ketone fused azadecalin glucocorticoid receptor modulators |
PL3338781T3 (pl) * | 2012-05-25 | 2020-03-31 | Corcept Therapeutics Incorporated | Modulatory receptorów glukokortykoidowych typu azadekaliny skondensowanej z heteroaryloketonem |
WO2017076757A1 (fr) | 2015-11-02 | 2017-05-11 | Basf Se | Utilisation d'oxadiazoles substitués pour lutter contre les champignons phytopathogènes |
EP3165094A1 (fr) | 2015-11-03 | 2017-05-10 | Basf Se | Oxadiazoles substitués pour lutter contre les champignons phytopathogènes |
EP3370525A1 (fr) | 2015-11-04 | 2018-09-12 | Basf Se | Utilisation d'oxadiazoles substitués pour lutter contre les champignons phytopathogènes |
AU2016355949A1 (en) | 2015-11-19 | 2018-05-10 | Basf Se | Substituted oxadiazoles for combating phytopathogenic fungi |
EA201891146A1 (ru) | 2015-11-19 | 2018-12-28 | Басф Се | Замещенные оксадиазолы для борьбы с фитопатогенными грибами |
RU2018138748A (ru) | 2016-04-11 | 2020-05-12 | Басф Се | Замещенные оксадиазолы для борьбы с фитопатогенными грибами |
WO2017211650A1 (fr) | 2016-06-09 | 2017-12-14 | Basf Se | Oxadiazoles substitués pour lutter contre des champignons phytopathogènes |
WO2017211652A1 (fr) | 2016-06-09 | 2017-12-14 | Basf Se | Oxadiazoles substitués pour lutter contre des champignons phytopathogènes |
US20190322631A1 (en) | 2016-12-19 | 2019-10-24 | Basf Se | Substituted oxadiazoles for combating phytopathogenic fungi |
EP3339297A1 (fr) | 2016-12-20 | 2018-06-27 | Basf Se | Oxadiazoles substitués pour lutter contre les champignons phytopathogènes |
EP3600282A4 (fr) | 2017-03-31 | 2020-08-19 | Corcept Therapeutics, Inc. | Modulateurs du récepteur de glucocorticoïdes destinés au traitement du cancer du col de l'utérus |
WO2018219797A1 (fr) | 2017-06-02 | 2018-12-06 | Basf Se | Oxadiazoles substitués utilisés pour lutter contre des champignons phytopathogènes |
US20200190043A1 (en) | 2017-06-19 | 2020-06-18 | Basf Se | 2-[[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]aryloxy](thio)acetamides for combating phytopathogenic fungi |
WO2019002158A1 (fr) | 2017-06-30 | 2019-01-03 | Basf Se | Trifluorométhyloxadiazoles substitués utilisés pour lutter contre des champignons phytopathogènes |
EP3684761A1 (fr) | 2017-09-18 | 2020-07-29 | Basf Se | Trifluorométhyloxadiazoles substitués permettant de lutter contre des champignons phytopathogènes |
WO2019101511A1 (fr) | 2017-11-23 | 2019-05-31 | Basf Se | Trifluorométhyloxadiazoles substitués permettant de lutter contre des champignons phytopathogènes |
US11234971B2 (en) | 2018-12-19 | 2022-02-01 | Corcept Therapeutics Incorporated | Methods of treating cancer comprising administration of a glucocorticoid receptor modulator and a cancer chemotherapy agent |
MX2021007322A (es) | 2018-12-19 | 2021-07-07 | Corcept Therapeutics Inc | Formulaciones farmaceuticas que contienen relacorilant, un compuesto de azadecalina fusionado con heteroaril-cetona. |
US11389432B2 (en) | 2018-12-19 | 2022-07-19 | Corcept Therapeutics Incorporated | Methods of treating cancer comprising administration of a glucocorticoid receptor modulator and a cancer chemotherapy agent |
KR20210118971A (ko) | 2019-02-22 | 2021-10-01 | 코어셉트 쎄라퓨틱스 인코포레이티드 | 헤테로아릴-케톤 융합 아자데칼린 글루코코르티코이드 수용체 조절제인 렐라코릴란트의 치료 용도 |
JP2023522308A (ja) * | 2020-03-31 | 2023-05-30 | エルジー・ケム・リミテッド | 膵島移植保護用組成物 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5641796A (en) * | 1994-11-01 | 1997-06-24 | Eli Lilly And Company | Oral hypoglycemic agents |
DE10222034A1 (de) * | 2002-05-17 | 2003-11-27 | Bayer Ag | Tetrahydroisochinolin-Derivate |
DE10229777A1 (de) * | 2002-07-03 | 2004-01-29 | Bayer Ag | Indolin-Phenylsulfonamid-Derivate |
US20070105959A1 (en) * | 2003-03-11 | 2007-05-10 | Shinya Kusuda | Cynnamyl alcohol derivative compounds and drugs containing the compounds as active ingredient |
US20060258683A1 (en) | 2003-04-07 | 2006-11-16 | Liu Kevin | Para-sulfonyl substituted phenyl compounds as modulators of ppars |
DE10335449A1 (de) | 2003-08-02 | 2005-02-17 | Bayer Healthcare Ag | Bicyclische Indolinsulfonamid-Derivate |
EP1586573B1 (fr) * | 2004-04-01 | 2007-02-07 | Sanofi-Aventis Deutschland GmbH | Oxadiazolones, procédé pour leur préparation, usage comme agents pharmaceutiques |
-
2006
- 2006-12-14 EP EP06025880A patent/EP1932843A1/fr not_active Withdrawn
-
2007
- 2007-11-30 RU RU2009126745/04A patent/RU2009126745A/ru not_active Application Discontinuation
- 2007-11-30 KR KR1020097012309A patent/KR20090087922A/ko not_active Application Discontinuation
- 2007-11-30 EP EP07846915.2A patent/EP2102198B1/fr active Active
- 2007-11-30 MX MX2009005535A patent/MX2009005535A/es not_active Application Discontinuation
- 2007-11-30 BR BRPI0720416-7A patent/BRPI0720416A2/pt not_active IP Right Cessation
- 2007-11-30 CN CNA2007800454445A patent/CN101558064A/zh active Pending
- 2007-11-30 WO PCT/EP2007/010390 patent/WO2008071311A1/fr active Application Filing
- 2007-11-30 JP JP2009540626A patent/JP2010512352A/ja not_active Abandoned
- 2007-11-30 CA CA002672347A patent/CA2672347A1/fr not_active Abandoned
- 2007-11-30 AU AU2007331805A patent/AU2007331805A1/en not_active Abandoned
- 2007-12-12 PE PE2007001772A patent/PE20081404A1/es not_active Application Discontinuation
- 2007-12-12 UY UY30783A patent/UY30783A1/es not_active Application Discontinuation
- 2007-12-12 AR ARP070105563A patent/AR064299A1/es not_active Application Discontinuation
- 2007-12-12 CL CL200703614A patent/CL2007003614A1/es unknown
- 2007-12-12 TW TW096147333A patent/TW200843749A/zh unknown
-
2009
- 2009-05-07 ZA ZA200903160A patent/ZA200903160B/xx unknown
- 2009-05-07 CR CR10778A patent/CR10778A/es not_active Application Discontinuation
- 2009-06-05 CO CO09058528A patent/CO6210729A2/es not_active Application Discontinuation
- 2009-06-09 US US12/480,974 patent/US8173674B2/en not_active Expired - Fee Related
- 2009-06-10 MA MA31971A patent/MA30981B1/fr unknown
- 2009-06-10 SV SV2009003293A patent/SV2009003293A/es unknown
- 2009-06-12 EC EC2009009409A patent/ECSP099409A/es unknown
- 2009-06-12 TN TNP2009000242A patent/TN2009000242A1/fr unknown
- 2009-06-15 NO NO20092293A patent/NO20092293L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
SV2009003293A (es) | 2009-10-27 |
TN2009000242A1 (en) | 2010-10-18 |
BRPI0720416A2 (pt) | 2013-12-31 |
ECSP099409A (es) | 2009-07-31 |
NO20092293L (no) | 2009-09-08 |
CA2672347A1 (fr) | 2008-06-19 |
US20090298871A1 (en) | 2009-12-03 |
CO6210729A2 (es) | 2010-10-20 |
WO2008071311A1 (fr) | 2008-06-19 |
CR10778A (es) | 2009-06-24 |
AU2007331805A1 (en) | 2008-06-19 |
EP2102198A1 (fr) | 2009-09-23 |
JP2010512352A (ja) | 2010-04-22 |
MX2009005535A (es) | 2009-06-05 |
TW200843749A (en) | 2008-11-16 |
EP1932843A1 (fr) | 2008-06-18 |
ZA200903160B (en) | 2010-10-27 |
CL2007003614A1 (es) | 2008-06-20 |
CN101558064A (zh) | 2009-10-14 |
RU2009126745A (ru) | 2011-01-20 |
US8173674B2 (en) | 2012-05-08 |
UY30783A1 (es) | 2008-07-31 |
KR20090087922A (ko) | 2009-08-18 |
AR064299A1 (es) | 2009-03-25 |
EP2102198B1 (fr) | 2015-02-25 |
PE20081404A1 (es) | 2008-11-04 |
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