MA29265B1 - Derives de 3-aryl-1, 2-benzisoxazole, et leur utilisation comme medicaments contre le cancer - Google Patents
Derives de 3-aryl-1, 2-benzisoxazole, et leur utilisation comme medicaments contre le cancerInfo
- Publication number
- MA29265B1 MA29265B1 MA30161A MA30161A MA29265B1 MA 29265 B1 MA29265 B1 MA 29265B1 MA 30161 A MA30161 A MA 30161A MA 30161 A MA30161 A MA 30161A MA 29265 B1 MA29265 B1 MA 29265B1
- Authority
- MA
- Morocco
- Prior art keywords
- aryl
- nr5r6
- nitro
- halogen
- cancer drugs
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/423—Oxazoles condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
L'INVENTION CONCERNE LES NOUVEAUX PRODUITS DE FORMULE (I): DANS LAQUELLE A1 ET A2 REPRÉSENTENT CH OU N; X REPRÉSENTE CRA OU N; Y REPRÉSENTE CRB OU N; R1, R2, R3 ET R4 IDENTIQUES OU DIFFÉRENTS REPRÉSENTENT NOTAMMENT HYDROGÈNE, HALOGÈNE, CYANO, NITRO, TRIFLUOROMÉTHYLE, OR5, SR5, NR5R6, C(O)R5, C(O)OR5, C(O) NR5R6, S(O)R5, S(O)2R5, S(O)NR5R6, S(O)2NR5R6, NR6C(O)R5, NR6C(O)OR5, ALKYLES, ALKÉNYLES, ALKYNYLES, ARYLES, HÉTÉROARYLES, ARALKYLES OU HÉTÉROARALKYLES, TOUS ÉVENTUELLEMENT SUBSTITUÉS; RA REPRÉSENTE NOTAMMENT HALOGÈNE, HYDROXYLE, ALCOXY, NITRO; RB REPRÉSENTE NOTAMMENT HYDROGÈNE, HALOGÈNE, CYANO, NITRO, TRIFLUOROMÉTHYLE, -W-(CI- C3ALKYLE)M- R5 ; R5 ET R6 REPRÉSENTE NOTAMMENT ALKYLE, ARALKYLE OU HÉTÉROARALKYLES ÉVENTUELLEMENT SUBSTITUÉS; CES PRODUITS ÉTANT SOUS TOUTES LES FORMES ISOMÈRES ET LES SELS, À TITRE DE MÉDICAMENTS.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0501801A FR2882361A1 (fr) | 2005-02-22 | 2005-02-22 | Nouveaux derives de 3-aryl-1,2-benzisoxazole, compositions les contenant et leur utilisation |
Publications (1)
Publication Number | Publication Date |
---|---|
MA29265B1 true MA29265B1 (fr) | 2008-02-01 |
Family
ID=35058405
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA30161A MA29265B1 (fr) | 2005-02-22 | 2007-08-23 | Derives de 3-aryl-1, 2-benzisoxazole, et leur utilisation comme medicaments contre le cancer |
Country Status (19)
Country | Link |
---|---|
US (1) | US20080070960A1 (fr) |
EP (1) | EP1861381A1 (fr) |
JP (1) | JP2008531493A (fr) |
KR (1) | KR20070110102A (fr) |
CN (1) | CN101146780A (fr) |
AR (1) | AR053684A1 (fr) |
AU (1) | AU2006217799A1 (fr) |
BR (1) | BRPI0606178A2 (fr) |
CA (1) | CA2597781A1 (fr) |
EA (1) | EA200701798A1 (fr) |
FR (1) | FR2882361A1 (fr) |
IL (1) | IL185166A0 (fr) |
MA (1) | MA29265B1 (fr) |
MX (1) | MX2007010278A (fr) |
NO (1) | NO20074631L (fr) |
TW (1) | TW200640884A (fr) |
UY (1) | UY29390A1 (fr) |
WO (1) | WO2006090052A1 (fr) |
ZA (1) | ZA200707080B (fr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2907453B1 (fr) | 2006-10-24 | 2008-12-26 | Sanofi Aventis Sa | Nouveaux derives du fluorene,compositions les contenant et utilisation |
AR077405A1 (es) | 2009-07-10 | 2011-08-24 | Sanofi Aventis | Derivados del indol inhibidores de hsp90, composiciones que los contienen y utilizacion de los mismos para el tratamiento del cancer |
FR2949467B1 (fr) | 2009-09-03 | 2011-11-25 | Sanofi Aventis | Nouveaux derives de 5,6,7,8-tetrahydroindolizine inhibiteurs d'hsp90, compositions les contenant et utilisation |
US8969343B2 (en) | 2012-12-19 | 2015-03-03 | Quanticel Pharmaceuticals, Inc. | Histone demethylase inhibitors |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6884814B2 (en) * | 2001-12-13 | 2005-04-26 | Wyeth | Phenyl benzisoxazoles as estrogenic agents |
EA009919B1 (ru) * | 2003-02-11 | 2008-04-28 | Вернэлис (Кембридж) Лимитед | Соединения изоксазола |
KR101129215B1 (ko) * | 2003-06-27 | 2012-04-13 | 교와 핫꼬 기린 가부시키가이샤 | Hsp90 패밀리 단백질 저해제 |
CA2536089A1 (fr) * | 2003-08-20 | 2005-03-03 | Eli Lilly And Company | Modulateurs du recepteur active de la proliferation des peroxysomes (ppar) |
-
2005
- 2005-02-22 FR FR0501801A patent/FR2882361A1/fr active Pending
-
2006
- 2006-02-20 EP EP06709343A patent/EP1861381A1/fr not_active Withdrawn
- 2006-02-20 KR KR1020077021865A patent/KR20070110102A/ko not_active Application Discontinuation
- 2006-02-20 BR BRPI0606178-8A patent/BRPI0606178A2/pt not_active IP Right Cessation
- 2006-02-20 CA CA002597781A patent/CA2597781A1/fr not_active Abandoned
- 2006-02-20 MX MX2007010278A patent/MX2007010278A/es not_active Application Discontinuation
- 2006-02-20 EA EA200701798A patent/EA200701798A1/ru unknown
- 2006-02-20 CN CNA2006800095240A patent/CN101146780A/zh active Pending
- 2006-02-20 JP JP2007555668A patent/JP2008531493A/ja active Pending
- 2006-02-20 AR ARP060100604A patent/AR053684A1/es unknown
- 2006-02-20 ZA ZA200707080A patent/ZA200707080B/xx unknown
- 2006-02-20 AU AU2006217799A patent/AU2006217799A1/en not_active Abandoned
- 2006-02-20 WO PCT/FR2006/000375 patent/WO2006090052A1/fr active Application Filing
- 2006-02-21 TW TW095105684A patent/TW200640884A/zh unknown
- 2006-02-22 UY UY29390A patent/UY29390A1/es unknown
-
2007
- 2007-08-09 IL IL185166A patent/IL185166A0/en unknown
- 2007-08-20 US US11/841,128 patent/US20080070960A1/en not_active Abandoned
- 2007-08-23 MA MA30161A patent/MA29265B1/fr unknown
- 2007-09-11 NO NO20074631A patent/NO20074631L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
KR20070110102A (ko) | 2007-11-15 |
ZA200707080B (en) | 2008-11-26 |
EP1861381A1 (fr) | 2007-12-05 |
WO2006090052A1 (fr) | 2006-08-31 |
AR053684A1 (es) | 2007-05-16 |
FR2882361A1 (fr) | 2006-08-25 |
EA200701798A1 (ru) | 2008-02-28 |
BRPI0606178A2 (pt) | 2009-06-02 |
NO20074631L (no) | 2007-11-20 |
CN101146780A (zh) | 2008-03-19 |
US20080070960A1 (en) | 2008-03-20 |
JP2008531493A (ja) | 2008-08-14 |
AU2006217799A1 (en) | 2006-08-31 |
TW200640884A (en) | 2006-12-01 |
MX2007010278A (es) | 2007-11-07 |
CA2597781A1 (fr) | 2006-08-31 |
UY29390A1 (es) | 2006-10-02 |
IL185166A0 (en) | 2007-12-03 |
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