MA23735A1 - Preparation et application des derives pyrroliques entant que medicaments - Google Patents

Preparation et application des derives pyrroliques entant que medicaments

Info

Publication number
MA23735A1
MA23735A1 MA24084A MA24084A MA23735A1 MA 23735 A1 MA23735 A1 MA 23735A1 MA 24084 A MA24084 A MA 24084A MA 24084 A MA24084 A MA 24084A MA 23735 A1 MA23735 A1 MA 23735A1
Authority
MA
Morocco
Prior art keywords
medicaments
preparation
application
pyrrol derivatives
pyrrol
Prior art date
Application number
MA24084A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MA23735A1 publication Critical patent/MA23735A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
MA24084A 1994-12-01 1995-12-01 Preparation et application des derives pyrroliques entant que medicaments MA23735A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US08/347,915 US5622948A (en) 1994-12-01 1994-12-01 Pyrrole pyridazine and pyridazinone anti-inflammatory agents

Publications (1)

Publication Number Publication Date
MA23735A1 true MA23735A1 (fr) 1996-07-01

Family

ID=23365840

Family Applications (1)

Application Number Title Priority Date Filing Date
MA24084A MA23735A1 (fr) 1994-12-01 1995-12-01 Preparation et application des derives pyrroliques entant que medicaments

Country Status (19)

Country Link
US (1) US5622948A (fr)
EP (1) EP0714895A1 (fr)
JP (1) JPH08208639A (fr)
KR (1) KR960022506A (fr)
CN (1) CN1066726C (fr)
AR (1) AR001771A1 (fr)
AU (1) AU3906295A (fr)
BR (1) BR9505610A (fr)
CA (1) CA2163490A1 (fr)
CO (1) CO4650183A1 (fr)
CZ (1) CZ316995A3 (fr)
FI (1) FI955783A (fr)
HU (1) HUT75117A (fr)
IL (1) IL116139A0 (fr)
MA (1) MA23735A1 (fr)
NO (1) NO954878L (fr)
PL (1) PL311536A1 (fr)
TR (1) TR199501528A1 (fr)
ZA (1) ZA9510027B (fr)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5622948A (en) * 1994-12-01 1997-04-22 Syntex (U.S.A.) Inc. Pyrrole pyridazine and pyridazinone anti-inflammatory agents
US6231888B1 (en) 1996-01-18 2001-05-15 Perio Products Ltd. Local delivery of non steroidal anti inflammatory drugs (NSAIDS) to the colon as a treatment for colonic polyps
DK0906279T3 (da) * 1996-05-30 2003-02-03 Hoffmann La Roche Pyrrolderivater
CA2205757C (fr) * 1996-05-30 2006-01-24 F. Hoffmann-La Roche Ag Derives de pyridazinone et leur utilisation comme inhibiteurs de la protasglandine g/h synthase i et ii(cox i et ii)
NZ501808A (en) * 1997-08-22 2002-12-20 Abbott Lab Arylpyridazinones and their use as prostaglandin endoperoxide H synthase biosynthesis inhibitors
US6525053B1 (en) 1997-08-22 2003-02-25 Abbott Laboratories Prostaglandin endoperoxide H synthase biosynthesis inhibitors
US6307047B1 (en) * 1997-08-22 2001-10-23 Abbott Laboratories Prostaglandin endoperoxide H synthase biosynthesis inhibitors
EP1007515A1 (fr) * 1997-08-22 2000-06-14 Abbott Laboratories Arylpyridazinones inhibitrices de la biosynthese de la prostaglandine endoperoxyde h synthase
HUP0100072A3 (en) * 1997-10-27 2002-11-28 Reddys Lab Ltd Dr Phenoxazine, phenthiazine derivatives, their use in medicine; process for their preparation and pharmaceutical compositions containing them
US6531152B1 (en) 1998-09-30 2003-03-11 Dexcel Pharma Technologies Ltd. Immediate release gastrointestinal drug delivery system
PL198503B1 (pl) * 1998-10-27 2008-06-30 Abbott Lab Związki pirydazynonowe, kompozycje farmaceutyczne je zawierające oraz ich zastosowanie
US6632451B2 (en) 1999-06-04 2003-10-14 Dexcel Pharma Technologies Ltd. Delayed total release two pulse gastrointestinal drug delivery system
DE60234057D1 (de) 2001-07-25 2009-11-26 Raptor Pharmaceutical Inc Zusammensetzungen und verfahren zur modulation des transports durch die blut-hirn-schranke
EP1539168A2 (fr) * 2002-07-11 2005-06-15 Merck & Co., Inc. Traitement de la douleur neuropathique au moyen de composes 6h-pyrrolo 3,4-d]pyridazine
EP2671507A3 (fr) 2005-04-28 2014-02-19 Proteus Digital Health, Inc. Système pharma-informatique
GB0610680D0 (en) 2006-05-31 2006-07-12 Istituto Di Ricerche D Biolog Therapeutic compounds
US8795627B2 (en) 2007-03-21 2014-08-05 Raptor Pharmaceuticals Inc. Treatment of liver disorders by administration of RAP conjugates
ES2524787T3 (es) 2007-11-15 2014-12-12 Msd Italia S.R.L. Derivados de piridazinona como inhibidores de PARP
DK2398500T3 (da) 2009-02-20 2019-05-13 2 Bbb Medicines B V Glutathion-baseret lægemiddelafgivelsessystem
AU2010245823B2 (en) 2009-05-06 2016-11-24 Laboratory Skin Care, Inc. Dermal delivery compositions comprising active agent-calcium phosphate particle complexes and methods of using the same
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates
EP2527335B1 (fr) 2011-04-26 2013-09-18 King Saud University Dérivés de la triazole comme anti-inflammatoires
KR102233456B1 (ko) 2017-05-31 2021-03-29 주식회사 대웅제약 4-메톡시피롤 유도체의 중간체 제조 방법
KR102233455B1 (ko) 2017-06-21 2021-03-29 주식회사 대웅제약 4-메톡시피롤 유도체의 중간체 제조 방법
WO2022159980A1 (fr) * 2021-01-25 2022-07-28 Athos Therapeutics, Inc. Composés pharmaceutiques et leurs procédés de fabrication et méthodes d'utilisation

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US2316942A (en) * 1937-12-27 1943-04-20 Schlumberger Well Surv Corp Apparatus for measuring temperatures in boreholes
US3586681A (en) * 1967-11-02 1971-06-22 Sandoz Ag 1,4,5,6-tetrahydropyridazines
US3726978A (en) * 1967-11-02 1973-04-10 Sandoz Ag Tetrahydropyridazines and pyridazinones as anti-inflammatory agents
US3752826A (en) * 1970-01-26 1973-08-14 Mcneilab Inc Aroyl substituted pyrroles
US4048191A (en) * 1975-06-27 1977-09-13 Mcneil Laboratories, Incorporated Halo-substituted 1-loweralkyl-5-aroylpyrrole-2-acetic acid compounds
US4089969A (en) * 1976-07-14 1978-05-16 Syntex (U.S.A.) Inc. 5-Aroyl-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof
JPS539788A (en) * 1976-07-14 1978-01-28 Syntex Inc 55aloyll1*22dihydroo3hh pyroro *1*22a* pyroll11 carboxylic acid derivative
US4247551A (en) * 1979-09-17 1981-01-27 Gruppo Lepetit S.P.A. N-Pyrrolyl-pyridazineamines and their use as antihypertensive agents
US4347187A (en) * 1980-10-20 1982-08-31 Syntex (U.S.A.) Inc. Process for preparing 5-aroyl 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acids and novel intermediates therein
IT1150070B (it) * 1980-12-22 1986-12-10 Lepetit Spa Procedimento per preparare derivati n-pirrolipiridazinamminici
AU8509882A (en) * 1981-06-30 1983-01-06 Merck & Co., Inc. Tricyclic derivatives of substituted pyrrole acids
EP0088128A4 (fr) * 1981-09-11 1984-04-06 Diamond Shamrock Corp 4-pyridylpyridazin(2h)-3-ones antiinflammatoires et analgesiques.
US4816454A (en) * 1984-09-21 1989-03-28 Cassella Aktiengesellschaft 4,5-dihydro-3(2H)-pyridazinones and their pharmacological use
GB8501372D0 (en) * 1985-01-18 1985-02-20 Smith Kline French Lab Chemical compounds
US5086052A (en) * 1987-07-17 1992-02-04 Abbott Laboratories Substituted 1,4,5,6-tetrahydro-2H-pyridazin-3-one and -3-thione compounds having lipoxygenase inhibitory activity
US4992441A (en) * 1987-10-14 1991-02-12 Mcneilab, Inc. 1-[[5-[[4-substituted-1-piperazinyl]methyl]-pyrrol-2-yl or furan-2-yl]methyl-2-piperidinones useful in treating schizophrenia
IE913866A1 (en) * 1990-11-28 1992-06-03 Ici Plc Aryl derivatives
CA2144742A1 (fr) * 1992-09-22 1994-03-31 Donald A. Young Cellules de mammiferes transformees de facon stable exprimant une cyclo-oxygenase inflammatoire regulee
US5543297A (en) * 1992-12-22 1996-08-06 Merck Frosst Canada, Inc. Human cyclooxygenase-2 cDNA and assays for evaluating cyclooxygenase-2 activity
US5332736A (en) * 1993-11-01 1994-07-26 Ortho Pharmaceutical Corporation Anti-convulsant aroyl aminoacylpyrroles
US5622948A (en) * 1994-12-01 1997-04-22 Syntex (U.S.A.) Inc. Pyrrole pyridazine and pyridazinone anti-inflammatory agents
KR102081455B1 (ko) * 2017-06-09 2020-04-28 선상규 다중브러시를 이용한 직류발전장치

Also Published As

Publication number Publication date
JPH08208639A (ja) 1996-08-13
HU9503384D0 (en) 1996-01-29
BR9505610A (pt) 1997-09-16
ZA9510027B (en) 1996-06-03
CN1132206A (zh) 1996-10-02
CZ316995A3 (en) 1996-06-12
AR001771A1 (es) 1997-12-10
TR199501528A1 (tr) 1996-11-21
FI955783A0 (fi) 1995-12-01
FI955783A (fi) 1996-06-02
CO4650183A1 (es) 1998-09-03
IL116139A0 (en) 1996-01-31
AU3906295A (en) 1996-06-06
CN1066726C (zh) 2001-06-06
HUT75117A (en) 1997-04-28
KR960022506A (ko) 1996-07-18
CA2163490A1 (fr) 1996-06-02
EP0714895A1 (fr) 1996-06-05
PL311536A1 (en) 1996-06-10
NO954878D0 (no) 1995-11-30
NO954878L (no) 1996-06-03
US5622948A (en) 1997-04-22

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