LU87416A1 - Microgranules charges en une substance active,constitues essentiellement d'un triglyceride d'acides gras satures et leur utilisation par voie topique dans le domaine therapeutique - Google Patents

Microgranules charges en une substance active,constitues essentiellement d'un triglyceride d'acides gras satures et leur utilisation par voie topique dans le domaine therapeutique Download PDF

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Publication number
LU87416A1
LU87416A1 LU87416A LU87416A LU87416A1 LU 87416 A1 LU87416 A1 LU 87416A1 LU 87416 A LU87416 A LU 87416A LU 87416 A LU87416 A LU 87416A LU 87416 A1 LU87416 A1 LU 87416A1
Authority
LU
Luxembourg
Prior art keywords
microgranules
active substance
acid
fatty acids
derivatives
Prior art date
Application number
LU87416A
Other languages
English (en)
French (fr)
Inventor
Jamoulle Jean-Claude
Allec Josiane
Brzokewicz Alain
Shroot Braham
Original Assignee
Cird
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cird filed Critical Cird
Priority to LU87416A priority Critical patent/LU87416A1/fr
Priority to PT92747A priority patent/PT92747A/pt
Priority to FI896321A priority patent/FI896321A0/fi
Priority to ZA899961A priority patent/ZA899961B/xx
Priority to NO89895307A priority patent/NO895307L/no
Priority to DK669789A priority patent/DK669789A/da
Priority to AT89403675T priority patent/ATE90869T1/de
Priority to DE89403675T priority patent/DE68907335T2/de
Priority to DE198989403675T priority patent/DE376852T1/de
Priority to KR1019890019845A priority patent/KR900009058A/ko
Priority to JP1345037A priority patent/JP2731008B2/ja
Priority to ES89403675T priority patent/ES2034951T3/es
Priority to EP89403675A priority patent/EP0376852B1/de
Priority to CA002006834A priority patent/CA2006834A1/fr
Priority to AU47306/89A priority patent/AU617570B2/en
Priority to NZ231982A priority patent/NZ231982A/en
Publication of LU87416A1 publication Critical patent/LU87416A1/fr
Priority to GR91300044T priority patent/GR910300044T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/02Cosmetics or similar toiletry preparations characterised by special physical form
    • A61K8/0241Containing particulates characterized by their shape and/or structure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/37Esters of carboxylic acids
    • A61K8/375Esters of carboxylic acids the alcohol moiety containing more than one hydroxy group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/67Vitamins
    • A61K8/671Vitamin A; Derivatives thereof, e.g. ester of vitamin A acid, ester of retinol, retinol, retinal
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/40Chemical, physico-chemical or functional or structural properties of particular ingredients
    • A61K2800/56Compounds, absorbed onto or entrapped into a solid carrier, e.g. encapsulated perfumes, inclusion compounds, sustained release forms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q7/00Preparations for affecting hair growth

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Birds (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Dermatology (AREA)
  • Emergency Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Cosmetics (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
LU87416A 1988-12-29 1988-12-29 Microgranules charges en une substance active,constitues essentiellement d'un triglyceride d'acides gras satures et leur utilisation par voie topique dans le domaine therapeutique LU87416A1 (fr)

Priority Applications (17)

Application Number Priority Date Filing Date Title
LU87416A LU87416A1 (fr) 1988-12-29 1988-12-29 Microgranules charges en une substance active,constitues essentiellement d'un triglyceride d'acides gras satures et leur utilisation par voie topique dans le domaine therapeutique
DE89403675T DE68907335T2 (de) 1988-12-29 1989-12-28 Im wesentlichen aus Triglyceriden gesättigter Fettsäuren bestehende, mit einem Wirkstoff beladene Mikrogranulate und ihre äusserliche therapeutische Anwendung.
JP1345037A JP2731008B2 (ja) 1988-12-29 1989-12-28 飽和脂肪酸トリグリセリドおよび有効成分含有微細粒並びに局所用製剤
ZA899961A ZA899961B (en) 1988-12-29 1989-12-28 Microgranulates comprising a saturated fatty acid triglyceride and an active substance,and pharmaceutical composition containing them
NO89895307A NO895307L (no) 1988-12-29 1989-12-28 Fylte mikrokapsler.
DK669789A DK669789A (da) 1988-12-29 1989-12-28 Mikrogranulater indeholdende et aktivt stof samt deres anvendelse
AT89403675T ATE90869T1 (de) 1988-12-29 1989-12-28 Im wesentlichen aus triglyceriden gesaettigter fettsaeuren bestehende, mit einem wirkstoff beladene mikrogranulate und ihre aeusserliche therapeutische anwendung.
PT92747A PT92747A (pt) 1988-12-29 1989-12-28 Processo para a preparacao de microgranulados carregados com uma substancia activa, constituidos essencialmente por um triglicerido de acidos gordos saturados e de uma composicao farmceutica que os contem
DE198989403675T DE376852T1 (de) 1988-12-29 1989-12-28 Im wesentlichen aus triglyceriden gesaettigter fettsaeuren bestehende, mit einem wirkstoff beladene mikrogranulate und ihre aeusserliche therapeutische anwendung.
KR1019890019845A KR900009058A (ko) 1988-12-29 1989-12-28 포화지방산 트리글리세리드와 활성기질로 구성되는 미소 과립물과 이를 함유하는 국소처리용 약품조성물
FI896321A FI896321A0 (fi) 1988-12-29 1989-12-28 Mikrogranulat innehaollande aktiv substans, bestaoende huvudsakligen av triglycerid av maettade fettsyror, samt deras anvaendning lokalt inom sjukvaerd.
ES89403675T ES2034951T3 (es) 1988-12-29 1989-12-28 Microgranulados cargados de una substancia activa, constituidos esencialmente por un triglicerido de acidos grasos saturados y su utilizacion por via topica en el campo terapeutico.
EP89403675A EP0376852B1 (de) 1988-12-29 1989-12-28 Im wesentlichen aus Triglyceriden gesättigter Fettsäuren bestehende, mit einem Wirkstoff beladene Mikrogranulate und ihre äusserliche therapeutische Anwendung
CA002006834A CA2006834A1 (fr) 1988-12-29 1989-12-28 Microgranules charges en une substance active, constitues essentiellement d'un triglyceride d'acides gras satures et leur utilisation par voie topique dans le domaine therapeutique
AU47306/89A AU617570B2 (en) 1988-12-29 1989-12-28 Microgranulates comprising a saturated fatty acid triglyceride and an active substance, and topical pharmaceutical compositions containing such microgranulates
NZ231982A NZ231982A (en) 1988-12-29 1990-01-04 Microgranulate compositions containing a therapeutically active agent
GR91300044T GR910300044T1 (en) 1988-12-29 1991-11-15 Microgranules essentially consisting of triglycerides of saturated fatty acids loaded with an active substance, and their topical therapeutical use

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
LU87416A LU87416A1 (fr) 1988-12-29 1988-12-29 Microgranules charges en une substance active,constitues essentiellement d'un triglyceride d'acides gras satures et leur utilisation par voie topique dans le domaine therapeutique

Publications (1)

Publication Number Publication Date
LU87416A1 true LU87416A1 (fr) 1990-07-10

Family

ID=19731128

Family Applications (1)

Application Number Title Priority Date Filing Date
LU87416A LU87416A1 (fr) 1988-12-29 1988-12-29 Microgranules charges en une substance active,constitues essentiellement d'un triglyceride d'acides gras satures et leur utilisation par voie topique dans le domaine therapeutique

Country Status (16)

Country Link
EP (1) EP0376852B1 (de)
JP (1) JP2731008B2 (de)
KR (1) KR900009058A (de)
AT (1) ATE90869T1 (de)
AU (1) AU617570B2 (de)
CA (1) CA2006834A1 (de)
DE (2) DE376852T1 (de)
DK (1) DK669789A (de)
ES (1) ES2034951T3 (de)
FI (1) FI896321A0 (de)
GR (1) GR910300044T1 (de)
LU (1) LU87416A1 (de)
NO (1) NO895307L (de)
NZ (1) NZ231982A (de)
PT (1) PT92747A (de)
ZA (1) ZA899961B (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2649608B1 (fr) * 1989-07-12 1991-10-11 Oreal Composition cosmetique sous forme d'un gel aqueux contenant en suspension des spheroides d'une substance lipidique solide non hydrophile
DE4336407A1 (de) * 1993-10-21 1995-04-27 Rotring Int Gmbh Wasserfeste Kosmetik
FR2721210B1 (fr) * 1994-06-17 1996-08-02 Oreal Composition de nettoyage contenant des grains lipidiques.
US5540920A (en) * 1994-11-22 1996-07-30 Olin Corporation Synergistic biocide composition containing pyrithione plus an additive
US5679648A (en) * 1994-11-30 1997-10-21 The University Hospital Methods for the treatment and prevention of fungal infections by administration of 3'-deoxypurine nucleosides
AT408067B (de) * 1995-03-17 2001-08-27 Gebro Pharma Gmbh Pharmazeutische zusammensetzung zur topischen applizierung und verfahren zu ihrer herstellung
DE19511322C2 (de) * 1995-03-28 1999-09-02 Mann Gerhard Chem Pharm Fab Sterile Augengele mit einem Gehalt an mittelkettigen Triglyceriden und Verfahren zu deren Herstellung
FR2737668B1 (fr) * 1995-08-08 1997-10-31 Rocher Yves Biolog Vegetale Billes a base de substances lipophiles, leur procede de fabrication et leurs applications
JPH09268118A (ja) 1996-04-01 1997-10-14 Kao Corp 肌色改善美容剤
DE19738247C2 (de) * 1997-09-02 2000-02-17 Goldwell Gmbh Haarpflegemittel
DE19952790A1 (de) * 1999-11-03 2001-05-17 Cognis Deutschland Gmbh Verfahren zur Herstellung von Fettstoffgranulaten
GB0015617D0 (en) * 2000-06-26 2000-08-16 Vectura Ltd Improved preparations for dermal delivery of active substances
ITMI20012366A1 (it) * 2001-11-09 2003-05-09 Farmatron Ltd Sistemi terapeutici stabilizzati a rilascio immediato e/o modificato per la somministrazione orale di principi attivi e/o eccipienti e/o ali
US7927034B2 (en) 2002-05-06 2011-04-19 Pharmakodex Limited Application device for topical administration of pharmaceutical compositions and products
US8980235B2 (en) 2003-09-30 2015-03-17 Arch Chemicals, Inc. Coated metal pyrithione particles for treatment of microorganisms
US9861605B2 (en) 2011-10-24 2018-01-09 Stable Solutions Llc Enriched injectable emulsion containing selected fatty acid triglycerides
FR3075635B1 (fr) * 2017-12-22 2019-12-06 Lvmh Recherche Procede de preparation de spheroides anhydres par cryogenie
KR102446371B1 (ko) * 2019-06-11 2022-09-22 대봉엘에스 주식회사 유지 조성물 및 이의 용도

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB543309A (en) * 1940-12-04 1942-02-19 John David Evans Improvements in or relating to drugs
DE2309202A1 (de) * 1973-02-21 1974-08-29 Schering Ag Arzneiformen mit mikroverkapseltem arzneimittelwirkstoff
DE2725924C3 (de) * 1977-06-08 1980-11-06 Hobeg Hochtemperaturreaktor-Brennelement Gmbh, 6450 Hanau Verfahren zur Herstellung kugelförmiger Teilchen aus niedrigschmelzenden organischen Substanzen

Also Published As

Publication number Publication date
AU4730689A (en) 1990-07-05
DE376852T1 (de) 1991-07-04
ZA899961B (en) 1990-10-31
CA2006834A1 (fr) 1990-06-29
AU617570B2 (en) 1991-11-28
JP2731008B2 (ja) 1998-03-25
DE68907335T2 (de) 1994-01-13
KR900009058A (ko) 1990-07-02
JPH02300116A (ja) 1990-12-12
NZ231982A (en) 1991-03-26
ES2034951T3 (es) 1994-10-16
NO895307D0 (no) 1989-12-28
FI896321A0 (fi) 1989-12-28
GR910300044T1 (en) 1991-11-15
EP0376852A1 (de) 1990-07-04
EP0376852B1 (de) 1993-06-23
DK669789D0 (da) 1989-12-28
DK669789A (da) 1990-06-30
PT92747A (pt) 1990-06-29
ATE90869T1 (de) 1993-07-15
ES2034951T1 (es) 1993-04-16
DE68907335D1 (de) 1993-07-29
NO895307L (no) 1990-07-02

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