KR950011740B1 - 축합된 피리미딘 유도체 - Google Patents

축합된 피리미딘 유도체 Download PDF

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Publication number
KR950011740B1
KR950011740B1 KR1019920015043A KR920015043A KR950011740B1 KR 950011740 B1 KR950011740 B1 KR 950011740B1 KR 1019920015043 A KR1019920015043 A KR 1019920015043A KR 920015043 A KR920015043 A KR 920015043A KR 950011740 B1 KR950011740 B1 KR 950011740B1
Authority
KR
South Korea
Prior art keywords
group
pharmacologically acceptable
acceptable salt
pyrimidine derivative
compound
Prior art date
Application number
KR1019920015043A
Other languages
English (en)
Korean (ko)
Other versions
KR930004307A (ko
Inventor
히로아끼 노무라
도오루 하네다
요시히꼬 고다께
노리히로 우에다
교오스께 기또오
Original Assignee
에자이 가부시끼가이샤
나이또오 하루오
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 에자이 가부시끼가이샤, 나이또오 하루오 filed Critical 에자이 가부시끼가이샤
Publication of KR930004307A publication Critical patent/KR930004307A/ko
Application granted granted Critical
Publication of KR950011740B1 publication Critical patent/KR950011740B1/ko

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
KR1019920015043A 1991-08-21 1992-08-21 축합된 피리미딘 유도체 KR950011740B1 (ko)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
JP91-209252 1991-08-21
JP20925291 1991-08-21
JP91-251548 1991-09-30
JP25154891 1991-09-30
JP92-217670 1992-08-17
JP21767092A JP3144903B2 (ja) 1991-08-21 1992-08-17 縮合ピリミジン誘導体
JP91-217670 1992-08-17

Publications (2)

Publication Number Publication Date
KR930004307A KR930004307A (ko) 1993-03-22
KR950011740B1 true KR950011740B1 (ko) 1995-10-09

Family

ID=27328976

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019920015043A KR950011740B1 (ko) 1991-08-21 1992-08-21 축합된 피리미딘 유도체

Country Status (9)

Country Link
JP (1) JP3144903B2 (fi)
KR (1) KR950011740B1 (fi)
CN (1) CN1070402A (fi)
AU (1) AU655051B2 (fi)
CA (1) CA2076431A1 (fi)
FI (1) FI923697A (fi)
HU (1) HUT70180A (fi)
NO (1) NO923249L (fi)
TW (1) TW202451B (fi)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUT70208A (en) * 1992-09-25 1995-09-28 Lilly Co Eli Process for preparing 5-substituted pyrrolo[2,3-d]-pyrimidines
US20110082158A1 (en) * 2008-10-01 2011-04-07 Aleem Gangjee Selective proton coupled folate transporter and folate receptor, and garftase and/or other folate metabolizing enzymes inhibitor compounds and methods of using the same
US8252804B2 (en) 2008-10-01 2012-08-28 Duquesne University Of The Holy Spirit Selective proton coupled folate transporter and folate receptor, and GARFTase inhibitor compounds and methods of using the same
CN106188060A (zh) * 2015-04-29 2016-12-07 厦门大学 嘧啶并吡咯类化合物、其制备方法、药用组合物及其应用
CN113788834B (zh) * 2021-09-18 2022-11-29 河南奥思恩医药科技有限公司 2,4-二氯-6,7-二氢-5H-吡咯并[3,4-d]嘧啶盐酸盐的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0438261A3 (en) * 1990-01-16 1992-02-26 Takeda Chemical Industries, Ltd. Condensed heterocyclic glutamic acid derivatives, their production and use

Also Published As

Publication number Publication date
FI923697A0 (fi) 1992-08-18
CA2076431A1 (en) 1993-02-22
CN1070402A (zh) 1993-03-31
TW202451B (fi) 1993-03-21
NO923249D0 (no) 1992-08-19
AU2115792A (en) 1993-02-25
NO923249L (no) 1993-02-22
AU655051B2 (en) 1994-12-01
JP3144903B2 (ja) 2001-03-12
FI923697A (fi) 1993-02-22
KR930004307A (ko) 1993-03-22
JPH05186437A (ja) 1993-07-27
HUT70180A (en) 1995-09-28

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E902 Notification of reason for refusal
G160 Decision to publish patent application
E701 Decision to grant or registration of patent right
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