KR930005587B1 - 세팔로스포린 화합물 - Google Patents

세팔로스포린 화합물 Download PDF

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Publication number
KR930005587B1
KR930005587B1 KR1019900015454A KR900015454A KR930005587B1 KR 930005587 B1 KR930005587 B1 KR 930005587B1 KR 1019900015454 A KR1019900015454 A KR 1019900015454A KR 900015454 A KR900015454 A KR 900015454A KR 930005587 B1 KR930005587 B1 KR 930005587B1
Authority
KR
South Korea
Prior art keywords
methyl
carboxylic acid
dihydroxyphenyl
cepem
fluoro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
KR1019900015454A
Other languages
English (en)
Korean (ko)
Other versions
KR910006299A (ko
Inventor
이사오 나가쿠라
Original Assignee
화이자 인코포레이티드
제이. 트레버 럼
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 화이자 인코포레이티드, 제이. 트레버 럼 filed Critical 화이자 인코포레이티드
Publication of KR910006299A publication Critical patent/KR910006299A/ko
Application granted granted Critical
Publication of KR930005587B1 publication Critical patent/KR930005587B1/ko
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1019900015454A 1989-09-29 1990-09-28 세팔로스포린 화합물 Expired - Fee Related KR930005587B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP254,331 1989-09-29
JP1254331A JPH0699443B2 (ja) 1989-09-29 1989-09-29 セファロスポリン化合物
US1-254331 1989-09-29

Publications (2)

Publication Number Publication Date
KR910006299A KR910006299A (ko) 1991-04-29
KR930005587B1 true KR930005587B1 (ko) 1993-06-23

Family

ID=17263521

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019900015454A Expired - Fee Related KR930005587B1 (ko) 1989-09-29 1990-09-28 세팔로스포린 화합물

Country Status (9)

Country Link
US (1) US5120728A (enExample)
EP (1) EP0420543A3 (enExample)
JP (1) JPH0699443B2 (enExample)
KR (1) KR930005587B1 (enExample)
CA (1) CA2026419A1 (enExample)
FI (1) FI904790A7 (enExample)
IE (1) IE903482A1 (enExample)
PT (1) PT95425A (enExample)
TW (1) TW204352B (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE113050T1 (de) * 1986-11-21 1994-11-15 Ici Pharma Cephalosporine, verfahren zu ihrer herstellung und pharmazeutische präparate.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5692290A (en) * 1979-12-27 1981-07-25 Toyama Chem Co Ltd Preparation of 7-amino-3-substituted methylcephem carboxylic acid, its salt or ester
NZ198350A (en) * 1980-09-25 1985-02-28 Toyama Chemical Co Ltd Cephalosporins and intermediates;pharmaceutical compositions
JPS6251688A (ja) * 1985-08-30 1987-03-06 Taito Pfizer Kk 新規なセフアロスポリン化合物
JPH064643B2 (ja) * 1985-12-20 1994-01-19 ファイザー製薬株式会社 セフアロスポリン化合物
JPS62209082A (ja) * 1986-03-11 1987-09-14 Banyu Pharmaceut Co Ltd セフアロスポリン誘導体
EP0269298B1 (en) * 1986-11-21 1994-10-19 Ici Pharma Cephalosporins, process for their preparation and pharmaceutical compositions
ATE113050T1 (de) * 1986-11-21 1994-11-15 Ici Pharma Cephalosporine, verfahren zu ihrer herstellung und pharmazeutische präparate.

Also Published As

Publication number Publication date
US5120728A (en) 1992-06-09
JPH03118386A (ja) 1991-05-20
FI904790A7 (fi) 1991-03-30
FI904790A0 (fi) 1990-09-28
KR910006299A (ko) 1991-04-29
EP0420543A3 (en) 1992-04-08
CA2026419A1 (en) 1991-03-30
JPH0699443B2 (ja) 1994-12-07
IE903482A1 (en) 1991-04-10
TW204352B (enExample) 1993-04-21
PT95425A (pt) 1991-05-22
EP0420543A2 (en) 1991-04-03

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