KR860001030B1 - 6a,10a-트랜스-헥사하이드로디벤조피라논의 제조방법 - Google Patents

6a,10a-트랜스-헥사하이드로디벤조피라논의 제조방법 Download PDF

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Publication number
KR860001030B1
KR860001030B1 KR1019830002130A KR830002130A KR860001030B1 KR 860001030 B1 KR860001030 B1 KR 860001030B1 KR 1019830002130 A KR1019830002130 A KR 1019830002130A KR 830002130 A KR830002130 A KR 830002130A KR 860001030 B1 KR860001030 B1 KR 860001030B1
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KR
South Korea
Prior art keywords
trans
methoxy
reaction
formula
phenol
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Expired
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KR1019830002130A
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English (en)
Korean (ko)
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KR840004737A (ko
Inventor
윌버 라이안 찰스
Original Assignee
일라이 릴리 앤드 캄파니
아더 알. 웨일
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Publication of KR840004737A publication Critical patent/KR840004737A/ko
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Publication of KR860001030B1 publication Critical patent/KR860001030B1/ko
Expired legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/80—Dibenzopyrans; Hydrogenated dibenzopyrans

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Fats And Perfumes (AREA)
  • Pyrane Compounds (AREA)
KR1019830002130A 1982-05-24 1983-05-16 6a,10a-트랜스-헥사하이드로디벤조피라논의 제조방법 Expired KR860001030B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US381,111 1982-05-24
US06/381,111 US4395560A (en) 1982-05-24 1982-05-24 Preparation of 6a,10a-trans-hexahydrodibenzopyranones

Publications (2)

Publication Number Publication Date
KR840004737A KR840004737A (ko) 1984-10-24
KR860001030B1 true KR860001030B1 (ko) 1986-07-28

Family

ID=23503705

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019830002130A Expired KR860001030B1 (ko) 1982-05-24 1983-05-16 6a,10a-트랜스-헥사하이드로디벤조피라논의 제조방법

Country Status (12)

Country Link
US (1) US4395560A (enExample)
EP (1) EP0096480B1 (enExample)
JP (1) JPS58210079A (enExample)
KR (1) KR860001030B1 (enExample)
CA (1) CA1188702A (enExample)
DE (1) DE3378119D1 (enExample)
DK (1) DK210083A (enExample)
GB (1) GB2121038B (enExample)
GR (1) GR79272B (enExample)
HU (1) HU193651B (enExample)
IE (1) IE55184B1 (enExample)
IL (1) IL68626A (enExample)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE247097T1 (de) * 1998-05-04 2003-08-15 Univ Connecticut Analgetische und immunomodulierende cannabinoiden
US7589220B2 (en) * 1998-06-09 2009-09-15 University Of Connecticut Inhibitors of the anandamide transporter
US7897598B2 (en) * 1998-06-09 2011-03-01 Alexandros Makriyannis Inhibitors of the anandamide transporter
US7276613B1 (en) 1998-11-24 2007-10-02 University Of Connecticut Retro-anandamides, high affinity and stability cannabinoid receptor ligands
US7161016B1 (en) 1998-11-24 2007-01-09 University Of Connecticut Cannabimimetic lipid amides as useful medications
US6900236B1 (en) * 1999-10-18 2005-05-31 University Of Connecticut Cannabimimetic indole derivatives
US7393842B2 (en) * 2001-08-31 2008-07-01 University Of Connecticut Pyrazole analogs acting on cannabinoid receptors
US7119108B1 (en) 1999-10-18 2006-10-10 University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
US6943266B1 (en) * 1999-10-18 2005-09-13 University Of Connecticut Bicyclic cannabinoid agonists for the cannabinoid receptor
US8084467B2 (en) * 1999-10-18 2011-12-27 University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
US7741365B2 (en) * 1999-10-18 2010-06-22 University Of Connecticut Peripheral cannabinoid receptor (CB2) selective ligands
MXPA02005103A (es) 1999-10-18 2003-09-25 Alexipharma Inc Ligandos selectivos del receptor de canabinoide (cb2) perifericos.
CA2435409A1 (en) * 2001-01-26 2002-08-01 University Of Connecticut Novel cannabimimetic ligands
WO2002060447A1 (en) 2001-01-29 2002-08-08 University Of Connecticut Receptor selective cannabimimetic aminoalkylindoles
WO2003005960A2 (en) * 2001-07-13 2003-01-23 University Of Connecticut Novel bicyclic and tricyclic cannabinoids
WO2003035005A2 (en) * 2001-10-26 2003-05-01 University Of Connecticut Heteroindanes: a new class of potent cannabimimetic ligands
AU2003265663A1 (en) 2002-08-23 2004-03-11 University Of Connecticut Keto cannabinoids with therapeutic indications
CA2638940C (en) * 2008-08-28 2009-09-15 Dalton Chemical Laboratories Inc. Improved synthesis of hexahydrodibenzopyranones

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT66744B (en) * 1976-07-06 1978-11-27 Lilly Co Eli Process for preparing cis-hexahydrodibenzopyranones
GB1582564A (en) * 1976-07-06 1981-01-14 Lilly Co Eli Dibenzopyrans
US4054583A (en) * 1976-07-06 1977-10-18 Eli Lilly And Company Process for converting 2,7-dihydroxy-5-isopropylidene-9-substituted-2,6-methano-3,4,5,6-tetrahydro-2H-1-benzoxocin to trans-1-hydroxy-3-substituted-6,6-dimethyl-6,6a,7,8,10,10a-hexahydro-9H-dibenzo(b,d)pyran-9-one
US4054581A (en) * 1976-07-06 1977-10-18 Eli Lilly And Company Preparation of cis-1-hydroxy-3-substituted-6,6-dimethyl-6,6a,7,8,10,10a-hexahydro-9H-dibenzo[b,d]pyran-9-ones and intermediates therefor
US4054582A (en) * 1976-07-06 1977-10-18 Eli Lilly And Company Process for converting cis-hexahydrodibenzo[b,d]pyran-9-ones to trans-hexahydrodibenzo[b,d]-pyran-9-ones
CA1096390A (en) * 1976-07-06 1981-02-24 Edward R. Lavagnino PROCESS FOR PREPARING DL-CIS-1-HYDROXY-3-SUBSTITUTED- 6,6-DIMETHYL-6,6.alpha.,7,8,10,10.alpha.-HEXAHYDRO-9H- DIBENZO(B,D,)PYRAN-9-ONES
US4171315A (en) * 1978-03-31 1979-10-16 Eli Lilly And Company Preparation of cis-hexahydrodibenzopyranones

Also Published As

Publication number Publication date
EP0096480B1 (en) 1988-09-28
DK210083D0 (da) 1983-05-11
US4395560A (en) 1983-07-26
JPS58210079A (ja) 1983-12-07
EP0096480A3 (en) 1985-04-03
GB2121038B (en) 1986-01-22
GB2121038A (en) 1983-12-14
GR79272B (enExample) 1984-05-20
DE3378119D1 (en) 1988-11-03
DK210083A (da) 1983-11-25
IE55184B1 (en) 1990-06-20
HU193651B (en) 1987-11-30
CA1188702A (en) 1985-06-11
KR840004737A (ko) 1984-10-24
EP0096480A2 (en) 1983-12-21
IL68626A0 (en) 1983-09-30
IE831115L (en) 1983-11-24
IL68626A (en) 1986-12-31
GB8313470D0 (en) 1983-06-22

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